These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

129 related articles for article (PubMed ID: 6259354)

  • 1. Synthesis and stereochemistry of 7-phenyl-2-propionanilidobenzo[a]quinolizidine derivatives. Structural probes of fentanyl analgesics.
    Maryanoff BE; McComsey DF; Taylor RJ; Gardocki JF
    J Med Chem; 1981 Jan; 24(1):79-88. PubMed ID: 6259354
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Stereoisomers of N-[1-hydroxy-(2-phenylethyl)-3-methyl-4-piperidyl]- N-phenylpropanamide: synthesis, stereochemistry, analgesic activity, and opioid receptor binding characteristics.
    Wang ZX; Zhu YC; Jin WQ; Chen XJ; Chen J; Ji RY; Chi ZQ
    J Med Chem; 1995 Sep; 38(18):3652-9. PubMed ID: 7658453
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Studies on synthesis and relationship between analgesic activity and receptor affinity for 3-methyl fentanyl derivatives.
    Jin WQ; Xu H; Zhu YC; Fang SN; Xia XL; Huang ZM; Ge BL; Chi ZQ
    Sci Sin; 1981 May; 24(5):710-20. PubMed ID: 6264594
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Potential affinity labels for the opiate receptor based on fentanyl and related compounds.
    Maryanoff BE; Simon EJ; Gioannini T; Gorissen H
    J Med Chem; 1982 Aug; 25(8):913-9. PubMed ID: 6288945
    [TBL] [Abstract][Full Text] [Related]  

  • 5. New 4-(heteroanilido)piperidines, structurally related to the pure opioid agonist fentanyl, with agonist and/or antagonist properties.
    Bagley JR; Wynn RL; Rudo FG; Doorley BM; Spencer HK; Spaulding T
    J Med Chem; 1989 Mar; 32(3):663-71. PubMed ID: 2563773
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Molecular structure of two conformationally restrained fentanyl analogues: cis- and trans-isomers of N-(3-methyl-1-[2-(1,2,3,4-tetrahydro)naphthyl] -4-piperidinyl)-N-phenylpropanamide.
    Klein CL; Stevens ED; Fifer EK; Borne RF
    J Pharm Sci; 1985 Nov; 74(11):1147-51. PubMed ID: 4087172
    [TBL] [Abstract][Full Text] [Related]  

  • 7. [Synthesis and analgesic activity of non-aryl analogues of 4-methoxycarbonyl fentanyl].
    Wen ST; Yang YL; Shao HZ; Zhang KG; Li YL; Chen JS
    Yao Xue Xue Bao; 1993; 28(3):181-7. PubMed ID: 8103617
    [TBL] [Abstract][Full Text] [Related]  

  • 8. [Studies on structure-activity relationships and receptor binding feature for 3-methylfentanyl derivatives].
    Weng JH; Xu XR; Zhu YC; Zhou J; Xu H; Chi ZQ
    Yao Xue Xue Bao; 1990; 25(3):178-85. PubMed ID: 2173349
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Probes for narcotic receptor mediated phenomena. 15. (3S,4S)-(+)-trans-3-methylfentanyl isothiocyanate, a potent site-directed acylating agent for the delta opioid receptors in vitro.
    Kim CH; Rothman RB; Jacobson AE; Mattson MV; Bykov V; Streaty RA; Klee WA; George C; Long JB; Rice KC
    J Med Chem; 1989 Jun; 32(6):1392-8. PubMed ID: 2542560
    [TBL] [Abstract][Full Text] [Related]  

  • 10. [Synthesis and pharmacological activities of the 1-substituted 4-methoxycarbonyl fentanyl derivatives].
    Yi M; Zhu GZ; Li JG; Chen JS
    Yao Xue Xue Bao; 1992; 27(10):734-7. PubMed ID: 1363456
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and analgesic activity of stereoisomers of cis-fluoro-ohmefentanyl.
    Yong Z; Hao W; Weifang Y; Qiyuan D; Xinjian C; Wenqiao J; Youcheng Z
    Pharmazie; 2003 May; 58(5):300-2. PubMed ID: 12779044
    [TBL] [Abstract][Full Text] [Related]  

  • 12. New heteroaryl derivatives of fentanyl.
    Llama EF; del Campo C; Capo M
    J Pharm Pharmacol; 1991 Jan; 43(1):68-9. PubMed ID: 1676069
    [TBL] [Abstract][Full Text] [Related]  

  • 13. "Carba"-analogues of fentanyl are opioid receptor agonists.
    Weltrowska G; Chung NN; Lemieux C; Guo J; Lu Y; Wilkes BC; Schiller PW
    J Med Chem; 2010 Apr; 53(7):2875-81. PubMed ID: 20218625
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and pharmacological evaluation of a series of new 3-methyl-1,4-disubstituted-piperidine analgesics.
    Lalinde N; Moliterni J; Wright D; Spencer HK; Ossipov MH; Spaulding TC; Rudo FG
    J Med Chem; 1990 Oct; 33(10):2876-82. PubMed ID: 2170652
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Probes for narcotic receptor mediated phenomena. 12. cis-(+)-3-Methylfentanyl isothiocyanate, a potent site-directed acylating agent for delta opioid receptors. Synthesis, absolute configuration, and receptor enantioselectivity.
    Burke TR; Jacobson AE; Rice KC; Silverton JV; Simonds WF; Streaty RA; Klee WA
    J Med Chem; 1986 Jun; 29(6):1087-93. PubMed ID: 3012085
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis and Biological Evaluation of Fentanyl Analogues Modified at Phenyl Groups with Alkyls.
    Qin Y; Ni L; Shi J; Zhu Z; Shi S; Lam AL; Magiera J; Sekar S; Kuo A; Smith MT; Li T
    ACS Chem Neurosci; 2019 Jan; 10(1):201-208. PubMed ID: 30179508
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Molecular docking reveals a novel binding site model for fentanyl at the mu-opioid receptor.
    Subramanian G; Paterlini MG; Portoghese PS; Ferguson DM
    J Med Chem; 2000 Feb; 43(3):381-91. PubMed ID: 10669565
    [TBL] [Abstract][Full Text] [Related]  

  • 18. [Synthesis and analgesic activity of 1-substituted derivatives of 4-methoxycarbonyl-4-N-propionylanilinepiperidine].
    Yang YL; Zhu XW; Zhu GZ; Yang ZJ; Li Y; Zhao SY; Chen CH; Zhang KG
    Yao Xue Xue Bao; 1990; 25(4):253-9. PubMed ID: 1980781
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthetic 1,4-disubstituted-1,4-dihydro-5H-tetrazol-5-one derivatives of fentanyl: alfentanil (R 39209), a potent, extremely short-acting narcotic analgesic.
    Janssens F; Torremans J; Janssen PA
    J Med Chem; 1986 Nov; 29(11):2290-7. PubMed ID: 2878076
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Structure-activity studies of fentanyl.
    Casy AF; Huckstep MR
    J Pharm Pharmacol; 1988 Sep; 40(9):605-8. PubMed ID: 2907025
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.