111 related articles for article (PubMed ID: 6562904)
1. Suicide inactivation of chymotrypsin by benzoxazinones.
Hedstrom L; Moorman AR; Dobbs J; Abeles RH
Biochemistry; 1984 Apr; 23(8):1753-9. PubMed ID: 6562904
[TBL] [Abstract][Full Text] [Related]
2. A new class of heterocyclic serine protease inhibitors. Inhibition of human leukocyte elastase, porcine pancreatic elastase, cathepsin G, and bovine chymotrypsin A alpha with substituted benzoxazinones, quinazolines, and anthranilates.
Teshima T; Griffin JC; Powers JC
J Biol Chem; 1982 May; 257(9):5085-91. PubMed ID: 7040392
[TBL] [Abstract][Full Text] [Related]
3. Inhibition of serine proteases by benzoxazinones: effects of electron withdrawal and 5-substitution.
Spencer RW; Copp LJ; Bonaventura B; Tam TF; Liak TJ; Billedeau RJ; Krantz A
Biochem Biophys Res Commun; 1986 Nov; 140(3):928-33. PubMed ID: 3535800
[TBL] [Abstract][Full Text] [Related]
4. Design and synthesis of 4H-3,1-benzoxazin-4-ones as potent alternate substrate inhibitors of human leukocyte elastase.
Krantz A; Spencer RW; Tam TF; Liak TJ; Copp LJ; Thomas EM; Rafferty SP
J Med Chem; 1990 Feb; 33(2):464-79. PubMed ID: 2299617
[TBL] [Abstract][Full Text] [Related]
5. Inhibition of human chymase by 2-amino-3,1-benzoxazin-4-ones.
Neumann U; Schechter NM; Gütschow M
Bioorg Med Chem; 2001 Apr; 9(4):947-54. PubMed ID: 11354678
[TBL] [Abstract][Full Text] [Related]
6. Inhibition of chymotrypsin and pancreatic elastase by 4H-3,1-benzoxazin-4-ones.
Neumann U; Stürzebecher J; Leistner S; Vieweg H
J Enzyme Inhib; 1991; 4(3):227-32. PubMed ID: 2037867
[TBL] [Abstract][Full Text] [Related]
7. Mechanism of inactivation of chymotrypsin by 5-butyl-3H-1,3-oxazine-2,6-dione.
Weidmann B; Abeles RH
Biochemistry; 1984 May; 23(11):2373-6. PubMed ID: 6548151
[TBL] [Abstract][Full Text] [Related]
8. Substituted isatoic anhydrides: selective inactivators of trypsin-like serine proteases.
Gelb MH; Abeles RH
J Med Chem; 1986 Apr; 29(4):585-9. PubMed ID: 3514913
[TBL] [Abstract][Full Text] [Related]
9. N-[2,2-dimethyl-3-(N-(4-cyanobenzoyl)amino)nonanoyl]-L-phenylalanine ethyl ester as a stable ester-type inhibitor of chymotrypsin-like serine proteases: structural requirements for potent inhibition of alpha-chymotrypsin.
Iijima K; Katada J; Yasuda E; Uno I; Hayashi Y
J Med Chem; 1999 Jan; 42(2):312-23. PubMed ID: 9925737
[TBL] [Abstract][Full Text] [Related]
10. Inhibition of cathepsin G by 4H-3,1-benzoxazin-4-ones.
Gütschow M; Neumann U
Bioorg Med Chem; 1997 Oct; 5(10):1935-42. PubMed ID: 9370038
[TBL] [Abstract][Full Text] [Related]
11. Proline-valine pseudo peptide enol lactones. Effective and selective inhibitors of chymotrypsin and human leukocyte elastase.
Reed PE; Katzenellenbogen JA
J Biol Chem; 1991 Jan; 266(1):13-21. PubMed ID: 1985887
[TBL] [Abstract][Full Text] [Related]
12. Inhibition of serine proteases by peptidyl fluoromethyl ketones.
Imperiali B; Abeles RH
Biochemistry; 1986 Jul; 25(13):3760-7. PubMed ID: 3527255
[TBL] [Abstract][Full Text] [Related]
13. Novel thieno[2,3-d][1,3]oxazin-4-ones as inhibitors of human leukocyte elastase.
Gütschow M; Neumann U
J Med Chem; 1998 May; 41(10):1729-40. PubMed ID: 9572899
[TBL] [Abstract][Full Text] [Related]
14. Inactivation of proteases and esterases by halomethylated derivatives of dihydrocoumarins.
Béchet JJ; Dupaix A; Roucous C; Bonamy AM
Biochimie; 1977; 59(3):241-6. PubMed ID: 889930
[TBL] [Abstract][Full Text] [Related]
15. Novel inactivators of serine proteases based on 6-chloro-2-pyrone.
Westkaemper RB; Abeles RH
Biochemistry; 1983 Jun; 22(13):3256-64. PubMed ID: 6411120
[TBL] [Abstract][Full Text] [Related]
16. Mechanism for slow-binding inhibition of human leukocyte elastase by valine-derived benzoxazinones.
Stein RL; Strimpler AM; Viscarello BR; Wildonger RA; Mauger RC; Trainor DA
Biochemistry; 1987 Jun; 26(13):4126-30. PubMed ID: 3651441
[TBL] [Abstract][Full Text] [Related]
17. Mechanism of inhibition of human leucocyte elastase by monocyclic beta-lactams.
Chabin R; Green BG; Gale P; Maycock AL; Weston H; Dorn CP; Finke PE; Hagmann WK; Hale JJ; MacCoss M
Biochemistry; 1993 Aug; 32(34):8970-80. PubMed ID: 8364042
[TBL] [Abstract][Full Text] [Related]
18. O'-(epoxyalkyl)tyrosines and (epoxyalkyl)phenylalanine as irreversible inactivators of serine proteases: synthesis and inhibition mechanism.
Tous G; Bush A; Tous A; Jordan F
J Med Chem; 1990 Jun; 33(6):1620-34. PubMed ID: 2187995
[TBL] [Abstract][Full Text] [Related]
19. 2-amino-4H-3,1-benzoxazin-4-ones as inhibitors of C1r serine protease.
Hays SJ; Caprathe BW; Gilmore JL; Amin N; Emmerling MR; Michael W; Nadimpalli R; Nath R; Raser KJ; Stafford D; Watson D; Wang K; Jaen JC
J Med Chem; 1998 Mar; 41(7):1060-7. PubMed ID: 9544206
[TBL] [Abstract][Full Text] [Related]
20. Inhibition of human sputum elastase by 7-substituted 5-methyl-2-isopropylamino-4H-3,1-benzoxazin-4-ones.
Uejima Y; Oshida J; Kawabata H; Kokubo M; Kato Y; Fujii K
Biochem Pharmacol; 1994 Jul; 48(2):426-8. PubMed ID: 8053939
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]