133 related articles for article (PubMed ID: 7205880)
1. Importance of the aromatic ring in adrenergic amines. 5. Nonaromatic analogues of phenylethanolamine as inhibitors of phenylethanolamine N-methyltransferase: role of hydrophobic and steric interactions.
Vincek WC; Aldrich CS; Borchardt RT; Grunewald GL
J Med Chem; 1981 Jan; 24(1):7-12. PubMed ID: 7205880
[No Abstract] [Full Text] [Related]
2. Importance of the aromatic ring in adrenergic amines. 6. Nonaromatic analogues of phenylethanolamine as inhibitors of phenylethanolamine N-methyltransferase: role of pi-electronic and steric interactions.
Davis DP; Borchardt RT; Grunewald GL
J Med Chem; 1981 Jan; 24(1):12-6. PubMed ID: 7205869
[TBL] [Abstract][Full Text] [Related]
3. Importance of the aromatic ring in adrenergic amines. Nonaromatic analoques of phenylethanolamine as substrates for phenylethanolamine N-methyltransferase.
Grunewald GL; Grindel JM; Vincek WC; Borchardt RT
Mol Pharmacol; 1975 Sep; 11(5):694-9. PubMed ID: 1237082
[No Abstract] [Full Text] [Related]
4. Conformational and steric aspects of phenylethanolamine and phenylethylamine analogues as substrates or inhibitors of phenylethanolamine N-methyltransferase.
Grunewald GL; Ye Q; Sall DJ; Criscione KR; Wise B
Mol Pharmacol; 1989 Jan; 35(1):93-7. PubMed ID: 2913486
[TBL] [Abstract][Full Text] [Related]
5. Importance of the aromatic ring in adrenergic amines. 8. 2-(Aminomethyl)-trans-2-decalols as inhibitors of norepinephrine N-methyltransferase.
Rafferty MF; Krass P; Borchardt RT; Grunewald GL
J Med Chem; 1982 Oct; 25(10):1250-2. PubMed ID: 7143367
[TBL] [Abstract][Full Text] [Related]
6. Importance of the aromatic ring in adrenergic amines. 7. Comparison of the stereoselectivity of norepinephrine N-methyltransferase for aromatic vs. nonaromatic substrates and inhibitors.
Rafferty MF; Wilson DS; Monn JA; Krass P; Borchardt RT; Grunewald GL
J Med Chem; 1982 Oct; 25(10):1198-204. PubMed ID: 7143356
[TBL] [Abstract][Full Text] [Related]
7. Quantitative structure-activity relationship studies of non-aromatic analogues of ethanolamine as inhibitors of phenylethanolamine N-methyltransferase.
Singh P
Arzneimittelforschung; 1985; 35(1):21-3. PubMed ID: 4039148
[TBL] [Abstract][Full Text] [Related]
8. Substrate and inhibitor kinetics of bovine phenylethanolamine-N-methyltransferase.
Hoffman AR; Ciaranello RD; Axelrod J
Biochem Pharmacol; 1975 Feb; 24(4):544-6. PubMed ID: 1167462
[No Abstract] [Full Text] [Related]
9. Regulation of phenylethanolamine N-methyl transferase.
Fuller RW; Roush BW; Molloy BB
Adv Enzyme Regul; 1974; 12():311-41. PubMed ID: 4462384
[No Abstract] [Full Text] [Related]
10. Conformational requirements of substrates for activity with phenylethanolamine N-methyltransferase.
Grunewald GL; Ye Q; Kieffer L; Monn JA
J Med Chem; 1988 Jan; 31(1):169-71. PubMed ID: 3336016
[TBL] [Abstract][Full Text] [Related]
11. Inhibitors of phenylethanolamine N-methyltransferase and epinephrine biosynthesis. 1. Chloro-substituted 1,2,3,4-tetrahydroisoquinolines.
Bondinell WE; Chapin FW; Girard GR; Kaiser C; Krog AJ; Pavloff AM; Schwartz MS; Silvestri JS; Vaidya PD; Lam BL; Wellman GR; Pendleton RG
J Med Chem; 1980 May; 23(5):506-11. PubMed ID: 7381849
[TBL] [Abstract][Full Text] [Related]
12. The remarkable substrate activity for phenylethanolamine N-methyltransferase of some conformationally defined phenylethylamines lacking a side-chain hydroxyl group. Conformationally defined adrenergic agents. 6.
Rafferty MF; Grunewald GL
Mol Pharmacol; 1982 Jul; 22(1):127-32. PubMed ID: 7121446
[No Abstract] [Full Text] [Related]
13. Conformational preference for the binding of biaryl substrates and inhibitors to the active site of phenylethanolamine N-methyltransferase.
Grunewald GL; Carter AE; Sall DJ; Monn JA
J Med Chem; 1988 Jan; 31(1):60-5. PubMed ID: 3336033
[TBL] [Abstract][Full Text] [Related]
14. Effects of sodium chloride on phenylethanolamine N-methyltransferase activity.
Cubeddu X L; Vargas AM
Mol Pharmacol; 1977 Jan; 13(1):172-80. PubMed ID: 13293
[No Abstract] [Full Text] [Related]
15. Inhibition in vitro of norepinephrine N-methyltransferase by 2-aminotetralins, analogs of phenylethylamines with rigid conformation.
Fuller RW; Molloy BB
Biochem Pharmacol; 1977 Mar; 26(5):446-7. PubMed ID: 849338
[No Abstract] [Full Text] [Related]
16. Brief cortisol exposure elevates adrenal phenylethanolamine N-methyltransferase after a necessary lag period.
Betito K; Diorio J; Boksa P
Eur J Pharmacol; 1993 Jul; 238(2-3):273-82. PubMed ID: 8405097
[TBL] [Abstract][Full Text] [Related]
17. Binding orientation of amphetamine and norfenfluramine analogues in the benzonorbornene and benzobicyclo[3.2.1]octane ring systems at the active site of phenylethanolamine N-methyltransferase (PNMT).
Grunewald GL; Markovich KM; Sall DJ
J Med Chem; 1987 Dec; 30(12):2191-208. PubMed ID: 3681889
[TBL] [Abstract][Full Text] [Related]
18. Importance of the aromatic ring in adrenergic amines. 2. Synthesis and adrenergic activity of some nonaromatic six- and eight-membered ring analogs of beta-phenylethanolamine.
Grunewald GL; Grindel JM; Patil PN; Salman KN
J Med Chem; 1976 Jan; 19(1):10-6. PubMed ID: 1534
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and evaluation of 3-substituted analogues of 1,2,3,4-tetrahydroisoquinoline as inhibitors of phenylethanolamine N-methyltransferase.
Grunewald GL; Sall DJ; Monn JA
J Med Chem; 1988 Apr; 31(4):824-30. PubMed ID: 3351861
[TBL] [Abstract][Full Text] [Related]
20. Tetrahydrothiadiazoloisoquinolines: synthesis and inhibition of phenylethanolamine-N-methyltransferase.
Girard GR; Bondinell WE; Hillegass LM; Holden KG; Pendleton RG; Uzinskas I
J Med Chem; 1989 Jul; 32(7):1566-71. PubMed ID: 2738892
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
