These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
6. Excitatory amino acid receptor antagonists: resolution, absolute stereochemistry, and pharmacology of (S)- and (R)-2-amino-2-(5-tert-butyl-3-hydroxyisoxazol-4-yl)acetic acid (ATAA). Johansen TN; Frydenvang K; Ebert B; Madsen U; Krogsgaard-Larsen P Chirality; 1997; 9(5-6):529-36. PubMed ID: 9329180 [TBL] [Abstract][Full Text] [Related]
7. Synthesis and structure-activity studies on acidic amino acids and related diacids as NMDA receptor ligands. Johansen TN; Frydenvang K; Ebert B; Krogsgaard-Larsen P; Madsen U J Med Chem; 1994 Sep; 37(20):3252-62. PubMed ID: 7523673 [TBL] [Abstract][Full Text] [Related]
8. Novel class of amino acid antagonists at non-N-methyl-D-aspartic acid excitatory amino acid receptors. Synthesis, in vitro and in vivo pharmacology, and neuroprotection. Krogsgaard-Larsen P; Ferkany JW; Nielsen EO; Madsen U; Ebert B; Johansen JS; Diemer NH; Bruhn T; Beattie DT; Curtis DR J Med Chem; 1991 Jan; 34(1):123-30. PubMed ID: 1825114 [TBL] [Abstract][Full Text] [Related]
9. Aryl and cycloalkyl analogues of AMPA: synthetic, pharmacological and stereochemical aspects. Skjaerbaek N; Brehm L; Johansen TN; Hansen LM; Nielsen B; Ebert B; Søby KK; Stensbøl TB; Falch E; Krogsgaard-Larsen P Bioorg Med Chem; 1998 Jan; 6(1):119-31. PubMed ID: 9502111 [TBL] [Abstract][Full Text] [Related]
10. Differentiation of in vivo effects of AMPA and NMDA receptor ligands using drug discrimination methods and convulsant/anticonvulsant activity. Arnt J; Sánchez C; Lenz SM; Madsen U; Krogsgaard-Larsen P Eur J Pharmacol; 1995 Oct; 285(3):289-97. PubMed ID: 8575516 [TBL] [Abstract][Full Text] [Related]
11. Resolution, absolute stereochemistry and molecular pharmacology of the enantiomers of ATPA. Stensbøl TB; Borre L; Johansen TN; Egebjerg J; Madsen U; Ebert B; Krogsgaard-Larsen P Eur J Pharmacol; 1999 Sep; 380(2-3):153-62. PubMed ID: 10513575 [TBL] [Abstract][Full Text] [Related]
12. Heteroaryl analogues of AMPA. Synthesis and quantitative structure-activity relationships. Bang-Andersen B; Lenz SM; Skjaerbaek N; Søby KK; Hansen HO; Ebert B; Bøgesø KP; Krogsgaard-Larsen P J Med Chem; 1997 Aug; 40(18):2831-42. PubMed ID: 9288165 [TBL] [Abstract][Full Text] [Related]
14. (S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid, a potent and selective agonist at the GluR5 subtype of ionotropic glutamate receptors. Synthesis, modeling, and molecular pharmacology. Brehm L; Greenwood JR; Hansen KB; Nielsen B; Egebjerg J; Stensbøl TB; Bräuner-Osborne H; Sløk FA; Kronborg TT; Krogsgaard-Larsen P J Med Chem; 2003 Apr; 46(8):1350-8. PubMed ID: 12672235 [TBL] [Abstract][Full Text] [Related]
15. Excitatory amino acid receptor ligands. Synthesis and biological activity of 3-isoxazolol amino acids structurally related to homoibotenic acid. Christensen IT; Ebert B; Madsen U; Nielsen B; Brehm L; Krogsgaard-Larsen P J Med Chem; 1992 Sep; 35(19):3512-9. PubMed ID: 1383544 [TBL] [Abstract][Full Text] [Related]
16. N-methyl-D-aspartic acid receptor agonists: resolution, absolute stereochemistry, and pharmacology of the enantiomers of 2-amino-2-(3-hydroxy-5-methyl-4-isoxazolyl)acetic acid. Madsen U; Frydenvang K; Ebert B; Johansen TN; Brehm L; Krogsgaard-Larsen P J Med Chem; 1996 Jan; 39(1):183-90. PubMed ID: 8568805 [TBL] [Abstract][Full Text] [Related]
17. Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2H- tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3- and GluR4-preferring AMPA receptor agonist. Vogensen SB; Jensen HS; Stensbøl TB; Frydenvang K; Bang-Andersen B; Johansen TN; Egebjerg J; Krogsgaard-Larsen P Chirality; 2000 Nov; 12(10):705-13. PubMed ID: 11054828 [TBL] [Abstract][Full Text] [Related]
18. Kynurenic acid analogues with improved affinity and selectivity for the glycine site on the N-methyl-D-aspartate receptor from rat brain. Foster AC; Kemp JA; Leeson PD; Grimwood S; Donald AE; Marshall GR; Priestley T; Smith JD; Carling RW Mol Pharmacol; 1992 May; 41(5):914-22. PubMed ID: 1375317 [TBL] [Abstract][Full Text] [Related]
19. Synthesis of 1,4,7,8,9,10-hexahydro-9-methyl-6-nitropyrido[3,4-f]- quinoxaline-2,3-dione and related quinoxalinediones: characterization of alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (and N-methyl-D-aspartate) receptor and anticonvulsant activity. Bigge CF; Malone TC; Boxer PA; Nelson CB; Ortwine DF; Schelkun RM; Retz DM; Lescosky LJ; Borosky SA; Vartanian MG J Med Chem; 1995 Sep; 38(19):3720-40. PubMed ID: 7562904 [TBL] [Abstract][Full Text] [Related]
20. Effects of thiocyanate and AMPA receptor ligands on (S)-5-fluorowillardiine, (S)-AMPA and (R,S)-AMPA binding. Hawkinson JE; Espitia SA Eur J Pharmacol; 1997 Jun; 329(2-3):213-21. PubMed ID: 9226415 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]