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6. Aryl and cycloalkyl analogues of AMPA: synthetic, pharmacological and stereochemical aspects. Skjaerbaek N; Brehm L; Johansen TN; Hansen LM; Nielsen B; Ebert B; Søby KK; Stensbøl TB; Falch E; Krogsgaard-Larsen P Bioorg Med Chem; 1998 Jan; 6(1):119-31. PubMed ID: 9502111 [TBL] [Abstract][Full Text] [Related]
7. Resolution, absolute stereochemistry and molecular pharmacology of the enantiomers of ATPA. Stensbøl TB; Borre L; Johansen TN; Egebjerg J; Madsen U; Ebert B; Krogsgaard-Larsen P Eur J Pharmacol; 1999 Sep; 380(2-3):153-62. PubMed ID: 10513575 [TBL] [Abstract][Full Text] [Related]
8. Excitatory amino acid receptor ligands: resolution, absolute stereochemistry, and enantiopharmacology of 2-amino-3-(4-butyl-3-hydroxyisoxazol-5-yl)propionic acid. Johansen TN; Ebert B; Bräuner-Osborne H; Didriksen M; Christensen IT; Søby KK; Madsen U; Krogsgaard-Larsen P; Brehm L J Med Chem; 1998 Mar; 41(6):930-9. PubMed ID: 9526567 [TBL] [Abstract][Full Text] [Related]
9. Ionotropic excitatory amino acid receptor ligands. Synthesis and pharmacology of a new amino acid AMPA antagonist. Madsen U; Sløk FA; Stensbøl TB; Bräuner-Osborne H; Lützhøft HH; Poulsen MV; Eriksen L; Krogsgaard-Larsen P Eur J Med Chem; 2000 Jan; 35(1):69-76. PubMed ID: 10733604 [TBL] [Abstract][Full Text] [Related]
10. Pharmacology and toxicology of ATOA, an AMPA receptor antagonist and a partial agonist at GluR5 receptors. Wahl P; Frandsen A; Madsen U; Schousboe A; Krogsgaard-Larsen P Neuropharmacology; 1998; 37(10-11):1205-10. PubMed ID: 9849658 [TBL] [Abstract][Full Text] [Related]
11. Characterization of the binding of [3H]NS 257, a novel competitive AMPA receptor antagonist, to rat brain membranes and brain sections. Nielsen EO; Johansen TH; Wätjen F; Drejer J J Neurochem; 1995 Sep; 65(3):1264-73. PubMed ID: 7543932 [TBL] [Abstract][Full Text] [Related]
12. Heteroaryl analogues of AMPA. Synthesis and quantitative structure-activity relationships. Bang-Andersen B; Lenz SM; Skjaerbaek N; Søby KK; Hansen HO; Ebert B; Bøgesø KP; Krogsgaard-Larsen P J Med Chem; 1997 Aug; 40(18):2831-42. PubMed ID: 9288165 [TBL] [Abstract][Full Text] [Related]
13. Differentiation of in vivo effects of AMPA and NMDA receptor ligands using drug discrimination methods and convulsant/anticonvulsant activity. Arnt J; Sánchez C; Lenz SM; Madsen U; Krogsgaard-Larsen P Eur J Pharmacol; 1995 Oct; 285(3):289-97. PubMed ID: 8575516 [TBL] [Abstract][Full Text] [Related]
14. Synthesis and structure-activity studies on acidic amino acids and related diacids as NMDA receptor ligands. Johansen TN; Frydenvang K; Ebert B; Krogsgaard-Larsen P; Madsen U J Med Chem; 1994 Sep; 37(20):3252-62. PubMed ID: 7523673 [TBL] [Abstract][Full Text] [Related]
15. Structural determinants for AMPA agonist activity of aryl or heteroaryl substituted AMPA analogues. Synthesis and pharmacology. Sørensen US; Falch E; Stensbøl TB; Jaroszewski JW; Madsen U; Krogsgaard-Larsen P Arch Pharm (Weinheim); 2001 Feb; 334(2):62-8. PubMed ID: 11268776 [TBL] [Abstract][Full Text] [Related]
16. Novel class of amino acid antagonists at non-N-methyl-D-aspartic acid excitatory amino acid receptors. Synthesis, in vitro and in vivo pharmacology, and neuroprotection. Krogsgaard-Larsen P; Ferkany JW; Nielsen EO; Madsen U; Ebert B; Johansen JS; Diemer NH; Bruhn T; Beattie DT; Curtis DR J Med Chem; 1991 Jan; 34(1):123-30. PubMed ID: 1825114 [TBL] [Abstract][Full Text] [Related]
17. Structural determinants of AMPA agonist activity in analogues of 2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid: synthesis and pharmacology. Bang-Andersen B; Ahmadian H; Lenz SM; Stensbøl TB; Madsen U; Bøgesø KP; Krogsgaard-Larsen P J Med Chem; 2000 Dec; 43(25):4910-8. PubMed ID: 11124000 [TBL] [Abstract][Full Text] [Related]
18. Excitatory amino acid receptor antagonists: resolution, absolute stereochemistry, and pharmacology of (S)- and (R)-2-amino-2-(5-tert-butyl-3-hydroxyisoxazol-4-yl)acetic acid (ATAA). Johansen TN; Frydenvang K; Ebert B; Madsen U; Krogsgaard-Larsen P Chirality; 1997; 9(5-6):529-36. PubMed ID: 9329180 [TBL] [Abstract][Full Text] [Related]