84 related articles for article (PubMed ID: 7578807)
1. Synthesis and biodistribution of [4-14C]-5-bromo-6-methoxy-5,6-dihydro-prodrug derivatives of 5-ethyl-2'-deoxyuridine.
Cheraghali AM; Morin KW; Kumar R; Knaus EE; Wiebe LI
Drug Des Discov; 1994 Jul; 12(1):53-61. PubMed ID: 7578807
[TBL] [Abstract][Full Text] [Related]
2. In vivo biodistribution, pharmacokinetic parameters, and brain uptake of 5-halo-y-methoxy(or ethoxy)-5,6-dihydro-3'-azido-3'-deoxythymidine diastereomers as potential prodrugs of 3'-azido-3'-deoxythymidine.
Wang L; Morin KW; Kumar R; Cheraghali M; Todd KG; Baker GB; Knaus EE; Wiebe LI
J Med Chem; 1996 Feb; 39(4):826-33. PubMed ID: 8632406
[TBL] [Abstract][Full Text] [Related]
3. Accumulation of 5-ethyl-2'-deoxyuridine and its 5,6-dihydro prodrugs in murine lung and its potential clinical application.
Cheraghali AM; Morin KW; Kumar R; Knaus EE; Wiebe LI
J Pharm Pharmacol; 1995 Jul; 47(7):595-600. PubMed ID: 8568628
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, biotransformation, pharmacokinetics, and antiviral properties of 5-ethyl-5-halo-6-methoxy-5,6-dihydro-2'-deoxyuridine diastereomers.
Cheraghali AM; Kumar R; Wang L; Knaus EE; Wiebe LI
Biochem Pharmacol; 1994 Apr; 47(9):1615-25. PubMed ID: 8185676
[TBL] [Abstract][Full Text] [Related]
5. Pharmacokinetics and bioavailability of 5-ethyl-2'-deoxyuridine and its novel (5R,6R)-5-bromo-6-ethoxy-5,6-dihydro prodrugs in mice.
Cheraghali AM; Kumar R; Knaus EE; Wiebe LI
Drug Metab Dispos; 1995 Feb; 23(2):223-6. PubMed ID: 7736915
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and antiviral activity of 5-ethyl-5-halo-6-alkoxy-(or azido)-5,6-dihydro-2'-deoxyuridine diastereomers as potential prodrugs to 5-ethyl-2'-deoxyuridine.
Kumar R; Wiebe LI; Knaus EE
Arch Pharm (Weinheim); 1997 Aug; 330(8):259-63. PubMed ID: 9361522
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and antiviral (HIV-1, HBV) activities of 5-halo-6-methoxy(or azido)-5,6-dihydro-3'-fluoro-3'-deoxythymidine diastereomers. Potential prodrugs to 3'-fluoro-3'-deoxythymidine.
Kumar R; Wang L; Wiebe LI; Knaus EE
J Med Chem; 1994 Oct; 37(21):3554-60. PubMed ID: 7932583
[TBL] [Abstract][Full Text] [Related]
8. Evaluation of 4'-[methyl-14C]thiothymidine for in vivo DNA synthesis imaging.
Toyohara J; Kumata K; Fukushi K; Irie T; Suzuki K
J Nucl Med; 2006 Oct; 47(10):1717-22. PubMed ID: 17015909
[TBL] [Abstract][Full Text] [Related]
9. Synthesis, in vitro biological stability, and anti-HIV activity of 5-halo-6-alkoxy(or azido)-5,6-dihydro-3'-azido-3'-deoxythymidine diastereomers as potential prodrugs to 3'-azido-3'-deoxythymidine (AZT).
Kumar R; Wang L; Wiebe LI; Knaus EE
J Med Chem; 1994 Dec; 37(25):4297-306. PubMed ID: 7996541
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and biological activity of 5-(2,2-difluorocyclopropyl)-2'-deoxyuridine deoxyuridine diastereomers.
Tandon M; Singh S; Xu L; Kumar P; Wiebe LI; Knaus EE; Gati WP; Tempest ML
Drug Des Discov; 1992; 9(1):79-91. PubMed ID: 1333829
[TBL] [Abstract][Full Text] [Related]
11. [Pharmacokinetic studies of 14C-labeled epervudine in rats].
Dereszlay I; Vereczkey L
Acta Pharm Hung; 1993 Jul; 63(4):222-6. PubMed ID: 8379338
[TBL] [Abstract][Full Text] [Related]
12. Synthesis of the diastereomers of 5-(2,2-dichlorocyclopropyl)- and 5-(2-chlorocyclopropyl)-2'-deoxyuridine, and the antiviral and cytotoxic activity of these and bromo analogues.
Tandon M; Singh S; Wiebe LI; Knaus EE; Gati WP; Tempest ML
Drug Des Deliv; 1991 Jul; 7(4):295-307. PubMed ID: 1657019
[TBL] [Abstract][Full Text] [Related]
13. Synthesis of 5-[1-hydroxy(or methoxy)-2-bromo(or chloro)ethyl]-2'-deoxyuridines and related halohydrin analogues with antiviral and cytotoxic activity.
Kumar R; Wiebe LI; Hall TW; Knaus EE; Tovell DR; Tyrrell DL; Allen TM; Fathi-Afshar R
J Med Chem; 1989 May; 32(5):941-4. PubMed ID: 2709380
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and enzymatic transformations of 5-halo-6-methoxy-5,6-dihydro derivatives of 5-[1-methoxy-2-halo (or 2,2-dihalo)ethyl]-2'-deoxyuridines as potential herpes simplex virus inhibitors.
Kumar R
J Enzyme Inhib Med Chem; 2003 Jun; 18(3):273-8. PubMed ID: 14506919
[TBL] [Abstract][Full Text] [Related]
15. Pharmacological studies on 5-methoxymethyl-2'-deoxyuridine: a new antiviral agent.
Meldrum JB; Gupta VS; Taneja AK; Sisodia CS
J Pharmacol Exp Ther; 1981 Feb; 216(2):275-80. PubMed ID: 7463349
[TBL] [Abstract][Full Text] [Related]
16. 5-Bromo (or chloro)-6-azido-5,6-dihydro-2' -deoxyuridine and -thymidine derivatives with potent antiviral activity.
Kumar R
Bioorg Med Chem Lett; 2002 Feb; 12(3):275-8. PubMed ID: 11814776
[TBL] [Abstract][Full Text] [Related]
17. Prodrugs of 5-ethyl-2'-deoxyuridine, I. Syntheses and antiviral activities of some 5'-O-acyl derivatives.
Keppeler K; Kiefer G; De Clercq E
Arch Pharm (Weinheim); 1984 Oct; 317(10):867-73. PubMed ID: 6517672
[No Abstract] [Full Text] [Related]
18. Prodrugs of 5-ethyl-2'-deoxyuridine, II. Syntheses and antiviral activities of 5'- and 3'-ester derivatives.
Kiefer G; Keppeler K; De Clercq E
Arch Pharm (Weinheim); 1986 Feb; 319(2):154-60. PubMed ID: 3010900
[No Abstract] [Full Text] [Related]
19. Labelling and biological evaluation of [(11)C]methoxy-Sch225336: a radioligand for the cannabinoid-type 2 receptor.
Evens N; Bosier B; Lavey BJ; Kozlowski JA; Vermaelen P; Baudemprez L; Busson R; Lambert DM; Van Laere K; Verbruggen AM; Bormans GM
Nucl Med Biol; 2008 Oct; 35(7):793-800. PubMed ID: 18848664
[TBL] [Abstract][Full Text] [Related]
20. Distribution of carbon-14 and associated radiation dose in rat fetal brain and liver after maternal injection of [14C]thymidine.
Takahashi S; Kubota Y; Koshimoto C; Sato H; Hatashita S
Radiat Res; 1994 Oct; 140(1):10-6. PubMed ID: 7938442
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
