These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

144 related articles for article (PubMed ID: 7597074)

  • 21. Carbonic anhydrase inhibitors: the first on-resin screening of a 4-sulfamoylphenylthiourea library.
    Innocenti A; Casini A; Alcaro MC; Papini AM; Scozzafava A; Supuran CT
    J Med Chem; 2004 Oct; 47(21):5224-9. PubMed ID: 15456265
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors.
    Mishra CB; Kumari S; Angeli A; Monti SM; Buonanno M; Prakash A; Tiwari M; Supuran CT
    J Enzyme Inhib Med Chem; 2016; 31(sup2):174-179. PubMed ID: 27314170
    [TBL] [Abstract][Full Text] [Related]  

  • 23. Discovery of novel spiro-piperidine derivatives as highly potent and selective melanin-concentrating hormone 1 receptor antagonists.
    Suzuki T; Moriya M; Sakamoto T; Suga T; Kishino H; Takahashi H; Ishikawa M; Nagai K; Imai Y; Sekino E; Ito M; Iwaasa H; Ishihara A; Tokita S; Kanatani A; Sato N; Fukami T
    Bioorg Med Chem Lett; 2009 Jun; 19(11):3072-7. PubMed ID: 19403308
    [TBL] [Abstract][Full Text] [Related]  

  • 24. Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms.
    Buemi MR; De Luca L; Ferro S; Bruno E; Ceruso M; Supuran CT; Pospíšilová K; Brynda J; Řezáčová P; Gitto R
    Eur J Med Chem; 2015 Sep; 102():223-32. PubMed ID: 26276436
    [TBL] [Abstract][Full Text] [Related]  

  • 25. The effects of some bromophenols on human carbonic anhydrase isoenzymes.
    Taslimi P; Gülçin İ; Öztaşkın N; Çetinkaya Y; Göksu S; Alwasel SH; Supuran CT
    J Enzyme Inhib Med Chem; 2016 Aug; 31(4):603-7. PubMed ID: 26133541
    [TBL] [Abstract][Full Text] [Related]  

  • 26. Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c.
    Carta F; Maresca A; Covarrubias AS; Mowbray SL; Jones TA; Supuran CT
    Bioorg Med Chem Lett; 2009 Dec; 19(23):6649-54. PubMed ID: 19846301
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Synthesis and evaluation of N-heteroarylsubstituted triazolosulfonamides as carbonic anhydrase inhibitors.
    Balci A; Arslan M; Nixha AR; Bilen C; Ergun A; Gençer N
    J Enzyme Inhib Med Chem; 2015 Jun; 30(3):377-82. PubMed ID: 25068730
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity.
    Congiu C; Onnis V; Deplano A; Balboni G; Dedeoglu N; Supuran CT
    Bioorg Med Chem Lett; 2015 Sep; 25(18):3850-3. PubMed ID: 26233435
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Carbonic anhydrase inhibitors: Synthesis, molecular docking, cytotoxic and inhibition of the human carbonic anhydrase isoforms I, II, IX, XII with novel benzenesulfonamides incorporating pyrrole, pyrrolopyrimidine and fused pyrrolopyrimidine moieties.
    Ghorab MM; Alsaid MS; Ceruso M; Nissan YM; Supuran CT
    Bioorg Med Chem; 2014 Jul; 22(14):3684-95. PubMed ID: 24878360
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Carbonic anhydrase inhibitors. Regioselective synthesis of novel series 1-substituted 1,4-dihydro-4-oxo-3-pyridinesulfonamides and their inhibition of the human cytosolic isozymes I and II and transmembrane cancer-associated isozymes IX and XII.
    Brzozowski Z; Sławiński J; Vullo D; Supuran CT
    Eur J Med Chem; 2012 Oct; 56():282-91. PubMed ID: 22910138
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Carbonic anhydrase inhibitors. Inhibition of human cytosolic isoforms I and II with (reduced) Schiff's bases incorporating sulfonamide, carboxylate and carboxymethyl moieties.
    Nasr G; Cristian A; Barboiu M; Vullo D; Winum JY; Supuran CT
    Bioorg Med Chem; 2014 May; 22(10):2867-74. PubMed ID: 24746465
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Carbonic anhydrase inhibitors: thioxolone versus sulfonamides for obtaining isozyme-selective inhibitors?
    Innocenti A; Maresca A; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2008 Jul; 18(14):3938-41. PubMed ID: 18572406
    [TBL] [Abstract][Full Text] [Related]  

  • 33. Novel indolin-2-one-based sulfonamides as carbonic anhydrase inhibitors: Synthesis, in vitro biological evaluation against carbonic anhydrases isoforms I, II, IV and VII and molecular docking studies.
    Eldehna WM; Al-Ansary GH; Bua S; Nocentini A; Gratteri P; Altoukhy A; Ghabbour H; Ahmed HY; Supuran CT
    Eur J Med Chem; 2017 Feb; 127():521-530. PubMed ID: 28109946
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Synthesis and evaluation of 4-alkoxy-[1'-cyclobutyl-spiro(3,4-dihydrobenzopyran-2,4'-piperidine)] analogues as histamine-3 receptor antagonists.
    Becknell NC; Dandu RR; Lyons JA; Aimone LD; Raddatz R; Hudkins RL
    Bioorg Med Chem Lett; 2012 Jan; 22(1):186-9. PubMed ID: 22153342
    [TBL] [Abstract][Full Text] [Related]  

  • 35. Carbonic anhydrase inhibitors: Inhibition of the new membrane-associated isoform XV with phenols.
    Innocenti A; Hilvo M; Scozzafava A; Parkkila S; Supuran CT
    Bioorg Med Chem Lett; 2008 Jun; 18(12):3593-6. PubMed ID: 18501600
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase.
    Bozdag M; Carta F; Vullo D; Isik S; AlOthman Z; Osman SM; Scozzafava A; Supuran CT
    J Enzyme Inhib Med Chem; 2016; 31(1):132-6. PubMed ID: 25669351
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII.
    D'Ascenzio M; Carradori S; De Monte C; Secci D; Ceruso M; Supuran CT
    Bioorg Med Chem; 2014 Mar; 22(6):1821-31. PubMed ID: 24560739
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Flow synthesis and biological activity of aryl sulfonamides as selective carbonic anhydrase IX and XII inhibitors.
    Rosatelli E; Carotti A; Ceruso M; Supuran CT; Gioiello A
    Bioorg Med Chem Lett; 2014 Aug; 24(15):3422-5. PubMed ID: 24948563
    [TBL] [Abstract][Full Text] [Related]  

  • 39. Multicomponent chemistry in the synthesis of carbonic anhydrase inhibitors.
    Kalinin S; Supuran CT; Krasavin M
    J Enzyme Inhib Med Chem; 2016; 31(sup4):185-199. PubMed ID: 27784162
    [TBL] [Abstract][Full Text] [Related]  

  • 40. Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with N-hydroxysulfamides--a new zinc-binding function in the design of inhibitors.
    Winum JY; Innocenti A; Nasr J; Montero JL; Scozzafava A; Vullo D; Supuran CT
    Bioorg Med Chem Lett; 2005 May; 15(9):2353-8. PubMed ID: 15837324
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 8.