113 related articles for article (PubMed ID: 7961978)
1. Discovery and structure-function analysis of alpha-melanocyte-stimulating hormone antagonists.
Jayawickreme CK; Quillan JM; Graminski GF; Lerner MR
J Biol Chem; 1994 Nov; 269(47):29846-54. PubMed ID: 7961978
[TBL] [Abstract][Full Text] [Related]
2. Cyclic lactam alpha-melanotropin analogues of Ac-Nle4-cyclo[Asp5, D-Phe7,Lys10] alpha-melanocyte-stimulating hormone-(4-10)-NH2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin receptors.
Hruby VJ; Lu D; Sharma SD; Castrucci AL; Kesterson RA; al-Obeidi FA; Hadley ME; Cone RD
J Med Chem; 1995 Sep; 38(18):3454-61. PubMed ID: 7658432
[TBL] [Abstract][Full Text] [Related]
3. Discovery and structure-activity relationships of novel alpha-melanocyte-stimulating hormone inhibitors.
Sawyer TK; Staples DJ; Castrucci AM; Hadley ME
Pept Res; 1989; 2(1):140-6. PubMed ID: 2562482
[TBL] [Abstract][Full Text] [Related]
4. Design, synthesis, and biological activities of a potent and selective alpha-melanotropin antagonist.
al-Obeidi F; Hruby VJ; Hadley ME; Sawyer TK; Castrucci AM
Int J Pept Protein Res; 1990 Mar; 35(3):228-34. PubMed ID: 2162330
[TBL] [Abstract][Full Text] [Related]
5. Structure-activity relationships of cyclic lactam analogues of alpha-melanocyte-stimulating hormone (alpha-MSH) targeting the human melanocortin-3 receptor.
Mayorov AV; Cai M; Palmer ES; Dedek MM; Cain JP; Van Scoy AR; Tan B; Vagner J; Trivedi D; Hruby VJ
J Med Chem; 2008 Jan; 51(2):187-95. PubMed ID: 18088090
[TBL] [Abstract][Full Text] [Related]
6. Potent and prolonged acting cyclic lactam analogues of alpha-melanotropin: design based on molecular dynamics.
Al-Obeidi F; Castrucci AM; Hadley ME; Hruby VJ
J Med Chem; 1989 Dec; 32(12):2555-61. PubMed ID: 2555512
[TBL] [Abstract][Full Text] [Related]
7. Biological and conformational examination of stereochemical modifications using the template melanotropin peptide, Ac-Nle-c[Asp-His-Phe-Arg-Trp-Ala-Lys]-NH2, on human melanocortin receptors.
Haskell-Luevano C; Nikiforovich G; Sharma SD; Yang YK; Dickinson C; Hruby VJ; Gantz I
J Med Chem; 1997 May; 40(11):1738-48. PubMed ID: 9171884
[TBL] [Abstract][Full Text] [Related]
8. Alpha-melanotropin: the minimal active sequence in the lizard skin bioassay.
Castrucci AM; Hadley ME; Sawyer TK; Wilkes BC; al-Obeidi F; Staples DJ; de Vaux AE; Dym O; Hintz MF; Riehm JP
Gen Comp Endocrinol; 1989 Jan; 73(1):157-63. PubMed ID: 2537778
[TBL] [Abstract][Full Text] [Related]
9. alpha-Melanotropin: the minimal active sequence in the frog skin bioassay.
Hruby VJ; Wilkes BC; Hadley ME; Al-Obeidi F; Sawyer TK; Staples DJ; de Vaux AE; Dym O; Castrucci AM; Hintz MF
J Med Chem; 1987 Nov; 30(11):2126-30. PubMed ID: 2822931
[TBL] [Abstract][Full Text] [Related]
10. Alpha-melanocyte stimulating hormone message and inhibitory sequences: comparative structure-activity studies on melanocytes.
Sawyer TK; Staples DJ; Castrucci AM; Hadley ME; al-Obeidi FA; Cody WL; Hruby VJ
Peptides; 1990; 11(2):351-7. PubMed ID: 2162535
[TBL] [Abstract][Full Text] [Related]
11. Design of potent linear alpha-melanotropin 4-10 analogues modified in positions 5 and 10.
Al-Obeidi F; Hruby VJ; Castrucci AM; Hadley ME
J Med Chem; 1989 Jan; 32(1):174-9. PubMed ID: 2535874
[TBL] [Abstract][Full Text] [Related]
12. Isolation and structural characterization of peptides related to alpha- and gamma-melanocyte-stimulating hormone (MSH) from the frog brain.
Bunel DT; Conlon JM; Chartrel N; Tonon MC; Vaudry H
Brain Res Mol Brain Res; 1992 Sep; 15(1-2):1-7. PubMed ID: 1331655
[TBL] [Abstract][Full Text] [Related]
13. [half-Cys4,half-Cys10]-alpha-Melanocyte-stimulating hormone: a cyclic alpha-melanotropin exhibiting superagonist biological activity.
Sawyer TK; Hruby VJ; Darman PS; Hadley ME
Proc Natl Acad Sci U S A; 1982 Mar; 79(6):1751-5. PubMed ID: 6281785
[TBL] [Abstract][Full Text] [Related]
14. Structure activity studies of the melanocortin-4 receptor by in vitro mutagenesis: identification of agouti-related protein (AGRP), melanocortin agonist and synthetic peptide antagonist interaction determinants.
Haskell-Luevano C; Cone RD; Monck EK; Wan YP
Biochemistry; 2001 May; 40(20):6164-79. PubMed ID: 11352754
[TBL] [Abstract][Full Text] [Related]
15. Three-dimensional molecular models of the hMC1R melanocortin receptor: complexes with melanotropin peptide agonists.
Haskell-Luevano C; Sawyer TK; Trumpp-Kallmeyer S; Bikker JA; Humblet C; Gantz I; Hruby VJ
Drug Des Discov; 1996 Dec; 14(3):197-211. PubMed ID: 9017363
[TBL] [Abstract][Full Text] [Related]
16. Melanin concentrating hormone. V. Isolation and characterization of alpha-melanocyte-stimulating hormone from frog pituitary glands.
Tonon MC; Desrues L; Lazure C; Jenks BG; Chrétien M; Vaudry H
Life Sci; 1989; 45(13):1155-61. PubMed ID: 2552247
[TBL] [Abstract][Full Text] [Related]
17. Chimeric NDP-MSH and MTII melanocortin peptides with agouti-related protein (AGRP) Arg-Phe-Phe amino acids possess agonist melanocortin receptor activity.
Joseph CG; Wilczynski A; Holder JR; Xiang Z; Bauzo RM; Scott JW; Haskell-Luevano C
Peptides; 2003 Dec; 24(12):1899-908. PubMed ID: 15127941
[TBL] [Abstract][Full Text] [Related]
18. Discovery of an alpha-melanotropin antagonist effective in vivo.
Castrucci AM; Sherbrooke WC; Sawyer TK; Staples DJ; Tuma MC; Hadley ME
Peptides; 1994; 15(4):627-32. PubMed ID: 7937337
[TBL] [Abstract][Full Text] [Related]
19. Peripheral analgesic activities of peptides related to alpha-melanocyte stimulating hormone and interleukin-1 beta 193-195.
Poole S; Bristow AF; Lorenzetti BB; Das RE; Smith TW; Ferreira SH
Br J Pharmacol; 1992 Jun; 106(2):489-92. PubMed ID: 1327383
[TBL] [Abstract][Full Text] [Related]
20. Development of potent gastrin-releasing peptide antagonists having a D-Pro-psi(CH2NH)-Phe-NH2 C terminus.
Leban JJ; Kull FC; Landavazo A; Stockstill B; McDermed JD
Proc Natl Acad Sci U S A; 1993 Mar; 90(5):1922-6. PubMed ID: 8446610
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
