These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

142 related articles for article (PubMed ID: 8003439)

  • 1. 1-Carbamoylalkyl-2-phenylindoles: relationship between side chain structure and estrogen antagonism.
    von Angerer E; Biberger C; Holler E; Koop R; Leichtl S
    J Steroid Biochem Mol Biol; 1994 May; 49(1):51-62. PubMed ID: 8003439
    [TBL] [Abstract][Full Text] [Related]  

  • 2. 2-Phenylindoles with sulfur containing side chains. Estrogen receptor affinity, antiestrogenic potency, and antitumor activity.
    Biberger C; von Angerer E
    J Steroid Biochem Mol Biol; 1996 Apr; 58(1):31-43. PubMed ID: 8809184
    [TBL] [Abstract][Full Text] [Related]  

  • 3. 1-Benzyl-2-phenylindole- and 1,2-diphenylindole-based antiestrogens. Estimation of agonist and antagonist activities in transfection assays.
    Biberger C; von Angerer E
    J Steroid Biochem Mol Biol; 1998 Mar; 64(5-6):277-85. PubMed ID: 9618029
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and biological activities of thioether derivatives related to the antiestrogens tamoxifen and ICI 164384.
    Auger S; Mérand Y; Pelletier JD; Poirier D; Labrie F
    J Steroid Biochem Mol Biol; 1995 Jun; 52(6):547-65. PubMed ID: 7779759
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Studies on heterocycle-based pure estrogen antagonists.
    Von Angerer E; Biberger C; Leichtl S
    Ann N Y Acad Sci; 1995 Jun; 761():176-91. PubMed ID: 7625720
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Altered expression of estrogen-regulated genes in a tamoxifen-resistant and ICI 164,384 and ICI 182,780 sensitive human breast cancer cell line, MCF-7/TAMR-1.
    Lykkesfeldt AE; Madsen MW; Briand P
    Cancer Res; 1994 Mar; 54(6):1587-95. PubMed ID: 8137264
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Hydroxylated polychlorinated biphenyls (PCBs) as estrogens and antiestrogens: structure-activity relationships.
    Connor K; Ramamoorthy K; Moore M; Mustain M; Chen I; Safe S; Zacharewski T; Gillesby B; Joyeux A; Balaguer P
    Toxicol Appl Pharmacol; 1997 Jul; 145(1):111-23. PubMed ID: 9221830
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Structure-activity relationships of nonisomerizable derivatives of tamoxifen: importance of hydroxyl group and side chain positioning for biological activity.
    Murphy CS; Parker CJ; McCague R; Jordan VC
    Mol Pharmacol; 1991 Mar; 39(3):421-8. PubMed ID: 2005879
    [TBL] [Abstract][Full Text] [Related]  

  • 9. 1-(aminoalkyl)-2-phenylindoles as novel pure estrogen antagonists.
    von Angerer E; Knebel N; Kager M; Ganss B
    J Med Chem; 1990 Sep; 33(9):2635-40. PubMed ID: 2391702
    [TBL] [Abstract][Full Text] [Related]  

  • 10. A new antiestrogen, 2-(4-hydroxy-phenyl)-3-methyl-1-[4-(2-piperidin-1-yl-ethoxy)-benzyl]-1H-indol-5-ol hydrochloride (ERA-923), inhibits the growth of tamoxifen-sensitive and -resistant tumors and is devoid of uterotropic effects in mice and rats.
    Greenberger LM; Annable T; Collins KI; Komm BS; Lyttle CR; Miller CP; Satyaswaroop PG; Zhang Y; Frost P
    Clin Cancer Res; 2001 Oct; 7(10):3166-77. PubMed ID: 11595711
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Antiestrogenic properties of keoxifene, trans-4-hydroxytamoxifen, and ICI 164384, a new steroidal antiestrogen, in ZR-75-1 human breast cancer cells.
    Poulin R; Merand Y; Poirier D; Levesque C; Dufour JM; Labrie F
    Breast Cancer Res Treat; 1989 Oct; 14(1):65-76. PubMed ID: 2605344
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and biological activity of 17 alpha-alkynylamide derivatives of estradiol.
    Poirier D; Labrie C; Mérand Y; Labrie F
    J Steroid Biochem Mol Biol; 1991 Jun; 38(6):759-74. PubMed ID: 2064992
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Action of "pure" antiestrogens in inhibiting estrogen receptor action.
    Parker MG
    Breast Cancer Res Treat; 1993; 26(2):131-7. PubMed ID: 8219250
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Human estrogen receptor ligand activity inversion mutants: receptors that interpret antiestrogens as estrogens and estrogens as antiestrogens and discriminate among different antiestrogens.
    Montano MM; Ekena K; Krueger KD; Keller AL; Katzenellenbogen BS
    Mol Endocrinol; 1996 Mar; 10(3):230-42. PubMed ID: 8833652
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and biological evaluation of stilbene-based pure estrogen antagonists.
    Walter G; Liebl R; von Angerer E
    Bioorg Med Chem Lett; 2004 Sep; 14(18):4659-63. PubMed ID: 15324884
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Depletion of estrogen receptor in human breast tumor cells by a novel substituted indole that does not bind to the hormone binding domain.
    Bitonti AJ; Dumont JA; Salituro FG; McDonald IA; Jarvi ET; Frey LM; Wright PS; Baumann RJ
    J Steroid Biochem Mol Biol; 1996 Apr; 58(1):21-30. PubMed ID: 8809183
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Human breast cancer cell lines resistant to pure anti-estrogens are sensitive to tamoxifen treatment.
    Lykkesfeldt AE; Larsen SS; Briand P
    Int J Cancer; 1995 May; 61(4):529-34. PubMed ID: 7759159
    [TBL] [Abstract][Full Text] [Related]  

  • 18. 3-Alkyl-2-phenylbenzo[b]thiophenes: nonsteroidal estrogen antagonists with mammary tumor inhibiting activity.
    von Angerer E; Erber S
    J Steroid Biochem Mol Biol; 1992 Mar; 41(3-8):557-62. PubMed ID: 1562527
    [TBL] [Abstract][Full Text] [Related]  

  • 19. A potent specific pure antiestrogen with clinical potential.
    Wakeling AE; Dukes M; Bowler J
    Cancer Res; 1991 Aug; 51(15):3867-73. PubMed ID: 1855205
    [TBL] [Abstract][Full Text] [Related]  

  • 20. 2-Phenylbenzo[b]thiophene-based antiestrogens with mammary tumor inhibiting activity.
    Leichtl S; von Angerer E
    Arch Pharm (Weinheim); 1998 Sep; 331(9):283-9. PubMed ID: 9793483
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.