257 related articles for article (PubMed ID: 8071813)
1. Morpholinoalkyl ester prodrugs of diclofenac: synthesis, in vitro and in vivo evaluation.
Tammara VK; Narurkar MM; Crider AM; Khan MA
J Pharm Sci; 1994 May; 83(5):644-8. PubMed ID: 8071813
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and evaluation of morpholinoalkyl ester prodrugs of indomethacin and naproxen.
Tammara VK; Narurkar MM; Crider AM; Khan MA
Pharm Res; 1993 Aug; 10(8):1191-9. PubMed ID: 8415407
[TBL] [Abstract][Full Text] [Related]
3. Cyclic amide derivatives as potential prodrugs II: N-hydroxymethylsuccinimide- / isatin esters of some NSAIDs as prodrugs with an improved therapeutic index.
Mahfouz NM; Omar FA; Aboul-Fadl T
Eur J Med Chem; 1999; 34(7-8):551-62. PubMed ID: 11278041
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, chemical and enzymatic hydrolysis, and bioavailability evaluation in rabbits of metronidazole amino acid ester prodrugs with enhanced water solubility.
Mahfouz NM; Hassan MA
J Pharm Pharmacol; 2001 Jun; 53(6):841-8. PubMed ID: 11428660
[TBL] [Abstract][Full Text] [Related]
5. Oligoethylene ester derivatives of ketoprofen, naproxen and diclofenac as oral prodrugs: a pharmacological evaluation.
Bonina F; Puglia C; Santagati NA; Saija A; Tomaino A; Tita B
Pharmazie; 2002 Aug; 57(8):552-5. PubMed ID: 12227196
[TBL] [Abstract][Full Text] [Related]
6. Prodrugs of 2',3'-dideoxyinosine (DDI): improved oral bioavailability via hydrophobic esters.
Kawaguchi T; Hasegawa T; Seki T; Juni K; Morimoto Y; Miyakawa A; Saneyoshi M
Chem Pharm Bull (Tokyo); 1992 May; 40(5):1338-40. PubMed ID: 1394659
[TBL] [Abstract][Full Text] [Related]
7. Vitamin K prodrugs: 1. Synthesis of amino acid esters of menahydroquinone-4 and enzymatic reconversion to an active form.
Takata J; Karube Y; Hanada M; Matsunaga K; Matsushima Y; Sendo T; Aoyama T
Pharm Res; 1995 Jan; 12(1):18-23. PubMed ID: 7724483
[TBL] [Abstract][Full Text] [Related]
8. Evaluation of a targeted prodrug strategy of enhance oral absorption of poorly water-soluble compounds.
Chan OH; Schmid HL; Stilgenbauer LA; Howson W; Horwell DC; Stewart BH
Pharm Res; 1998 Jul; 15(7):1012-8. PubMed ID: 9688053
[TBL] [Abstract][Full Text] [Related]
9. The physicochemical properties, plasma enzymatic hydrolysis, and nasal absorption of acyclovir and its 2'-ester prodrugs.
Shao Z; Park GB; Krishnamoorthy R; Mitra AK
Pharm Res; 1994 Feb; 11(2):237-42. PubMed ID: 8165182
[TBL] [Abstract][Full Text] [Related]
10. Pharmacokinetics of indomethacin ester prodrugs: gastrointestinal and hepatic toxicity and the hydrolytic capacity of various tissues in rats.
Ogiso T; Iwaki M; Tanino T; Nagai T; Ueda Y; Muraoka O; Tanabe G
Biol Pharm Bull; 1996 Sep; 19(9):1178-83. PubMed ID: 8889037
[TBL] [Abstract][Full Text] [Related]
11. Prodrugs of peptides. 18. Synthesis and evaluation of various esters of desmopressin (dDAVP).
Kahns AH; Buur A; Bundgaard H
Pharm Res; 1993 Jan; 10(1):68-74. PubMed ID: 8430062
[TBL] [Abstract][Full Text] [Related]
12. Synthesis and in vitro/in vivo evaluation of novel oral N-alkyl- and N,N-dialkyl-carbamate esters of entacapone.
Savolainen J; Leppanen J; Forsberg M; Taipale H; Nevalainen T; Huuskonen J; Gynther J; Mannisto PT; Jarvinen T
Life Sci; 2000; 67(2):205-16. PubMed ID: 10901288
[TBL] [Abstract][Full Text] [Related]
13. Synthesis, enzymatic hydrolysis and physico-chemical properties of N-substituted 4-(aminomethyl)benzoate diester prodrugs of ganciclovir.
Jensen E; Bundgaard H
Acta Pharm Nord; 1991; 3(4):243-7. PubMed ID: 1781915
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and pharmacological evaluation of oligoethylene ester derivatives as indomethacin oral prodrugs.
De Caprariis P; Palagiano F; Bonina F; Montenegro L; D'Amico M; Rossi F
J Pharm Sci; 1994 Nov; 83(11):1578-81. PubMed ID: 7891278
[TBL] [Abstract][Full Text] [Related]
15. Synthesis and in-vitro/in-vivo evaluation of orally administered entacapone prodrugs.
Leppänen J; Savolainen J; Nevalainen T; Forsberg M; Huuskonen J; Taipale H; Gynther J; Männistö PT; Järvinen T
J Pharm Pharmacol; 2001 Nov; 53(11):1489-98. PubMed ID: 11732751
[TBL] [Abstract][Full Text] [Related]
16. Prodrugs of 2',3'-didehydro-3'-deoxythymidine.
Hasegawa T; Seki T; Juni K; Saneyoshi M; Kawaguchi T
J Pharm Sci; 1993 Dec; 82(12):1232-6. PubMed ID: 8308702
[TBL] [Abstract][Full Text] [Related]
17. Water-soluble, solution-stable, and biolabile N-substituted (aminomethyl)benzoate ester prodrugs of acyclovir.
Bundgaard H; Jensen E; Falch E
Pharm Res; 1991 Sep; 8(9):1087-93. PubMed ID: 1788153
[TBL] [Abstract][Full Text] [Related]
18. Permeation of buprenorphine and its 3-alkyl-ester prodrugs through human skin.
Stinchcomb AL; Paliwal A; Dua R; Imoto H; Woodard RW; Flynn GL
Pharm Res; 1996 Oct; 13(10):1519-23. PubMed ID: 8899844
[TBL] [Abstract][Full Text] [Related]
19. In vitro and in vivo study of water-soluble prodrugs of dexanabinol.
Pop E; Rachwal S; Vlasak J; Biegon A; Zharikova A; Prokai L
J Pharm Sci; 1999 Nov; 88(11):1156-60. PubMed ID: 10564064
[TBL] [Abstract][Full Text] [Related]
20. Bisphosphonate prodrugs: synthesis and in vitro evaluation of novel acyloxyalkyl esters of clodronic acid.
Niemi R; Vepsäläinen J; Taipale H and ; Järvinen T
J Med Chem; 1999 Dec; 42(24):5053-8. PubMed ID: 10585214
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]