39 related articles for article (PubMed ID: 8182707)
1. Synthesis and in vitro evaluation of 9-anilino-3,6-diaminoacridines active against a multidrug-resistant strain of the malaria parasite Plasmodium falciparum.
Gamage SA; Tepsiri N; Wilairat P; Wojcik SJ; Figgitt DP; Ralph RK; Denny WA
J Med Chem; 1994 May; 37(10):1486-94. PubMed ID: 8182707
[TBL] [Abstract][Full Text] [Related]
2. 3,6-Diamino-4-(2-halophenyl)-2-benzoylthieno[2,3-b]pyridine-5-carbonitriles are selective inhibitors of Plasmodium falciparum glycogen synthase kinase-3.
Fugel W; Oberholzer AE; Gschloessl B; Dzikowski R; Pressburger N; Preu L; Pearl LH; Baratte B; Ratin M; Okun I; Doerig C; Kruggel S; Lemcke T; Meijer L; Kunick C
J Med Chem; 2013 Jan; 56(1):264-75. PubMed ID: 23214499
[TBL] [Abstract][Full Text] [Related]
3. New 4-(N-cinnamoylbutyl)aminoacridines as potential multi-stage antiplasmodial leads.
Fonte M; Fontinha D; Moita D; Caño-Prades O; Avalos-Padilla Y; Fernàndez-Busquets X; Prudêncio M; Gomes P; Teixeira C
Eur J Med Chem; 2023 Oct; 258():115575. PubMed ID: 37390511
[TBL] [Abstract][Full Text] [Related]
4. In vitro Plasmodium falciparum drug sensitivity assay: inhibition of parasite growth by incorporation of stomatocytogenic amphiphiles into the erythrocyte membrane.
Ziegler HL; Staerk D; Christensen J; Hviid L; Hägerstrand H; Jaroszewski JW
Antimicrob Agents Chemother; 2002 May; 46(5):1441-6. PubMed ID: 11959580
[TBL] [Abstract][Full Text] [Related]
5. Development of diaminoquinazoline histone lysine methyltransferase inhibitors as potent blood-stage antimalarial compounds.
Sundriyal S; Malmquist NA; Caron J; Blundell S; Liu F; Chen X; Srimongkolpithak N; Jin J; Charman SA; Scherf A; Fuchter MJ
ChemMedChem; 2014 Oct; 9(10):2360-2373. PubMed ID: 25044750
[TBL] [Abstract][Full Text] [Related]
6. A class of pantothenic acid analogs inhibits Plasmodium falciparum pantothenate kinase and represses the proliferation of malaria parasites.
Spry C; Chai CL; Kirk K; Saliba KJ
Antimicrob Agents Chemother; 2005 Nov; 49(11):4649-57. PubMed ID: 16251308
[TBL] [Abstract][Full Text] [Related]
7. Antimalarial activities of polyhydroxyphenyl and hydroxamic acid derivatives.
Holland KP; Elford HL; Bracchi V; Annis CG; Schuster SM; Chakrabarti D
Antimicrob Agents Chemother; 1998 Sep; 42(9):2456-8. PubMed ID: 9736585
[TBL] [Abstract][Full Text] [Related]
8. Structure-Activity Relationship of a Pyrrole Based Series of PfPKG Inhibitors as Anti-Malarials.
Gilleran JA; Ashraf K; Delvillar M; Eck T; Fondekar R; Miller EB; Hutchinson A; Dong A; Seitova A; De Souza ML; Augeri D; Halabelian L; Siekierka J; Rotella DP; Gordon J; Childers WE; Grier MC; Staker BL; Roberge JY; Bhanot P
J Med Chem; 2024 Mar; 67(5):3467-3503. PubMed ID: 38372781
[TBL] [Abstract][Full Text] [Related]
9. Plasmodium falciparum topoisomerases: Emerging targets for anti-malarial therapy.
Dar A; Godara P; Prusty D; Bashir M
Eur J Med Chem; 2024 Feb; 265():116056. PubMed ID: 38171145
[TBL] [Abstract][Full Text] [Related]
10. Oudemansin and 9-methoxystrobilurin derivatives with antimalarial activity from cultures of the basidiomycete
Palasarn S; Pruksatrakul T; Choowong W; Wiriyathanawudhiwong N; Boonpratuang T; Surawatanawong P; Thongpanchang C; Isaka M
Org Biomol Chem; 2023 Oct; 21(39):7944-7953. PubMed ID: 37740400
[TBL] [Abstract][Full Text] [Related]
11. Optimization of diastereomeric dihydropyridines as antimalarials.
Van Horn KS; Zhao Y; Parvatkar PT; Maier J; Mutka T; Lacrue A; Brockmeier F; Ebert D; Wu W; Casandra DR; Namelikonda N; Yacoub J; Sigal M; Knapp S; Floyd D; Waterson D; Burrows JN; Duffy J; DeRisi JL; Kyle DE; Guy RK; Manetsch R
Eur J Med Chem; 2024 Jun; 275():116599. PubMed ID: 38909569
[TBL] [Abstract][Full Text] [Related]
12. Reaction hijacking inhibition of
Xie SC; Wang Y; Morton CJ; Metcalfe RD; Dogovski C; Pasaje CFA; Dunn E; Luth MR; Kumpornsin K; Istvan ES; Park JS; Fairhurst KJ; Ketprasit N; Yeo T; Yildirim O; Bhebhe MN; Klug DM; Rutledge PJ; Godoy LC; Dey S; De Souza ML; Siqueira-Neto JL; Du Y; Puhalovich T; Amini M; Shami G; Loesbanluechai D; Nie S; Williamson N; Jana GP; Maity BC; Thomson P; Foley T; Tan DS; Niles JC; Han BW; Goldberg DE; Burrows J; Fidock DA; Lee MCS; Winzeler EA; Griffin MDW; Todd MH; Tilley L
Res Sq; 2023 Jul; ():. PubMed ID: 37546892
[TBL] [Abstract][Full Text] [Related]
13. Improved synthesis of antiplasmodial 4-aminoacridines and 4,9-diaminoacridines.
Fonte M; Teixeira C; Gomes P
RSC Adv; 2024 Feb; 14(9):6253-6261. PubMed ID: 38375018
[TBL] [Abstract][Full Text] [Related]
14. An efficient three-component synthesis of highly functionalized tetrahydroacenaphtho[1,2-b]indolone derivatives catalyzed by L-proline.
Zhang JJ; Feng X; Liu XC; Huang ZB; Shi DQ
Mol Divers; 2014 Nov; 18(4):727-36. PubMed ID: 25151274
[TBL] [Abstract][Full Text] [Related]
15. Docking studies, synthesis, characterization and evaluation of their antioxidant and cytotoxic activities of some novel isoxazole-substituted 9-anilinoacridine derivatives.
Kalirajan R; Rafick MH; Sankar S; Jubie S
ScientificWorldJournal; 2012; 2012():165258. PubMed ID: 22593663
[TBL] [Abstract][Full Text] [Related]
16. Synthesis of novel Eu(III) luminescent probe based on 9- acridinecarboxylic acid skelton for sensing of ds-DNA.
Azab HA; Hussein BH; El-Falouji AI
J Fluoresc; 2012 Mar; 22(2):639-49. PubMed ID: 22065175
[TBL] [Abstract][Full Text] [Related]
17. Acridine and acridinones: old and new structures with antimalarial activity.
Valdés AF
Open Med Chem J; 2011; 5():11-20. PubMed ID: 21673977
[TBL] [Abstract][Full Text] [Related]
18. Synthesis and anti-intestinal nematode activity of variously substituted benzonaphthyridine derivatives.
Duan LP; Wen AD; Wu NB; Tao Y; Zhang HB
Molecules; 2011 Feb; 16(2):1593-602. PubMed ID: 21321530
[TBL] [Abstract][Full Text] [Related]
19. Antimalarial drug targets in Plasmodium falciparum predicted by stage-specific metabolic network analysis.
Huthmacher C; Hoppe A; Bulik S; Holzhütter HG
BMC Syst Biol; 2010 Aug; 4():120. PubMed ID: 20807400
[TBL] [Abstract][Full Text] [Related]
20. Antimalarial 9-anilinoacridine compounds directed at hematin.
Auparakkitanon S; Noonpakdee W; Ralph RK; Denny WA; Wilairat P
Antimicrob Agents Chemother; 2003 Dec; 47(12):3708-12. PubMed ID: 14638470
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]