116 related articles for article (PubMed ID: 8216669)
1. Tricyclic heteroaromatic systems 1,2,4-triazolo[1,5-a]quinoxalines: synthesis and benzodiazepine receptor activity.
Catarzi D; Cecchi L; Colotta V; Melani F; Filacchioni G; Martini C; Giusti L; Lucacchini A
Farmaco; 1993 Aug; 48(8):1065-78. PubMed ID: 8216669
[TBL] [Abstract][Full Text] [Related]
2. Tricyclic heteroaromatic systems pyrazolo[1,5-a]quinoxalines: synthesis and benzodiazepine receptor activity.
Colotta V; Cecchi L; Catarzi D; Conti G; Filacchioni G; Martini C; Giusti L; Lucacchini A
Farmaco; 1993 Aug; 48(8):1051-63. PubMed ID: 8216668
[TBL] [Abstract][Full Text] [Related]
3. Tricyclic heteroaromatic systems. 2-Phenyl-1,2,4-triazolo[1,5-c][1,3]benzoxazin-5-one: a novel benzodiazepine receptor ligand.
Catarzi D; Cecchi L; Colotta V; Filacchioni ; Martini C; Giusti L; Lucacchini A; Valle G
Farmaco; 1994 Feb; 49(2):89-92. PubMed ID: 8003185
[TBL] [Abstract][Full Text] [Related]
4. Studies on annelated 1,4-benzothiazines and 1,5-benzothiazepines. X--Synthesis and inhibition of benzodiazepine receptor binding of new 1,4-thiazine and 1,5-thiazepine polycondensed heterocycles with steroidal structure.
Grandolini G; Ambrogi V; Perioli L; Giannaccini G; Lucacchini A; Martini C
Farmaco; 1996 Mar; 51(3):203-7. PubMed ID: 8688143
[TBL] [Abstract][Full Text] [Related]
5. Tricyclic heteroaromatic systems. 1,2,4-triazolo[4,3-a]quinoxalines and 1,2,4-Triazino[4,3-a]quinoxalines: synthesis and central benzodiazepine receptor activity.
Colotta V; Catarzi D; Varano F; Cecchi L; Filacchioni G; Galli A; Costagli C
Arch Pharm (Weinheim); 1997 Dec; 330(12):387-91. PubMed ID: 9474898
[TBL] [Abstract][Full Text] [Related]
6. Structure-activity relationships of 1,2,4-triazolo[1,5-a] quinoxalines and their 1-deaza analogues imidazo[1,2-a]quinoxalines at the benzodiazepine receptor.
Catarzi D; Cecchi L; Colotta V; Melani F; Filacchioni G; Martini C; Giusti L; Lucacchini A
J Med Chem; 1994 Sep; 37(18):2846-50. PubMed ID: 8071933
[TBL] [Abstract][Full Text] [Related]
7. 1,2,4-Triazolo[1,5-a]quinoxaline derivatives: synthesis and biological evaluation as adenosine receptor antagonists.
Catarzi D; Colotta V; Varano F; Filacchioni G; Martini C; Trincavelli L; Lucacchini A
Farmaco; 2004 Feb; 59(2):71-81. PubMed ID: 14871498
[TBL] [Abstract][Full Text] [Related]
8. 4-amido-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones as new potent and selective human A3 adenosine receptor antagonists. synthesis, pharmacological evaluation, and ligand-receptor modeling studies.
Lenzi O; Colotta V; Catarzi D; Varano F; Filacchioni G; Martini C; Trincavelli L; Ciampi O; Varani K; Marighetti F; Morizzo E; Moro S
J Med Chem; 2006 Jun; 49(13):3916-25. PubMed ID: 16789747
[TBL] [Abstract][Full Text] [Related]
9. Reaction of 1-aminophthalazines with alpha-halocarbonyl compounds: imidazo[2,1-a]phthalazines and their benzodiazepine receptor activities.
Catarzi D; Cecchi L; Colotta V; Conti G; Melani F; Filacchioni G; Martini C; Giusti L; Lucacchini A
Farmaco; 1993 Apr; 48(4):447-57. PubMed ID: 8395173
[TBL] [Abstract][Full Text] [Related]
10. Studies on annelated 1,4-benzothiazines and 1,5-benzothiazepines. VII. Synthesis and inhibition of benzodiazepine receptor binding of some 4,5-dihydro-tetrazolo[5,1-d]-1,5-benzothiazepines and 5-phenyl-s-triazolo[3,4-d]-1,5-benzothiazepines.
Ambrogi V; Grandolini G; Perioli L; Giusti L; Lucacchini A; Martini C
Farmaco; 1993 May; 48(5):665-76. PubMed ID: 8393678
[TBL] [Abstract][Full Text] [Related]
11. Specific inhibition of benzodiazepine receptor binding by some N-(2-methyl or 1,2-dimethylindol-3-ylglyoxylyl)amino acid derivatives.
Primofiore G; Marini AM; Da Settimo F; Salvadori C; Martini C; Lucacchini A; Giannaccini G
Farmaco; 1990 Mar; 45(3):341-51. PubMed ID: 2166528
[TBL] [Abstract][Full Text] [Related]
12. Studies on annelated 1,4-benzothiazines and 1,5-benzothiazepines. VIII-Synthesis and inhibition of benzodiazepine receptor binding of some derivatives of triazino[3,4-c]-1,4-benzothiazine and triazino[3,4-d]-1,5-benzothiazepine, two new heterocyclic ring systems.
Perioli L; Ambrogi V; Grandolini G; Giusti L; Lucacchini A; Martini C
Farmaco; 1994 Apr; 49(4):245-51. PubMed ID: 8049004
[TBL] [Abstract][Full Text] [Related]
13. 1,2,4-Triazolo[1,5-a]quinoxaline as a versatile tool for the design of selective human A3 adenosine receptor antagonists: synthesis, biological evaluation, and molecular modeling studies of 2-(hetero)aryl- and 2-carboxy-substituted derivatives.
Catarzi D; Colotta V; Varano F; Lenzi O; Filacchioni G; Trincavelli L; Martini C; Montopoli C; Moro S
J Med Chem; 2005 Dec; 48(25):7932-45. PubMed ID: 16335918
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and biological evaluation of analogues of 7-chloro-4,5-dihydro-4- oxo-8-(1,2,4-triazol-4-yl)-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylic acid (TQX-173) as novel selective AMPA receptor antagonists.
Catarzi D; Colotta V; Varano F; Calabri FR; Filacchioni G; Galli A; Costagli C; CarlĂ V
J Med Chem; 2004 Jan; 47(1):262-72. PubMed ID: 14695840
[TBL] [Abstract][Full Text] [Related]
15. Tricyclic heteroaromatic systems. Synthesis of 1,3 and 1,2 disubstituted [1]benzopyrano[4,3-b]pyrrol-4-ones and structure-activity relationships as benzodiazepine receptor ligands.
Colotta V; Cecchi L; Melani F; Filacchioni G; Martini C; Gelli S; Lucacchini A
Farmaco; 1991 Oct; 46(10):1139-54. PubMed ID: 1667727
[TBL] [Abstract][Full Text] [Related]
16. 1,2,4-triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A3 adenosine receptor antagonists: synthesis, pharmacological, and ligand-receptor modeling studies.
Colotta V; Catarzi D; Varano F; Calabri FR; Lenzi O; Filacchioni G; Martini C; Trincavelli L; Deflorian F; Moro S
J Med Chem; 2004 Jul; 47(14):3580-90. PubMed ID: 15214785
[TBL] [Abstract][Full Text] [Related]
17. Altered GABA(A)-benzodiazepine receptor number and pharmacology in the adult guinea pig cerebral cortex after chronic prenatal ethanol exposure.
Bailey CD; Brien JF; Reynolds JN
Alcohol Clin Exp Res; 1999 Nov; 23(11):1816-24. PubMed ID: 10591599
[TBL] [Abstract][Full Text] [Related]
18. Synthesis and binding activity of some pyrazolo[1,5-c]quinazolines as tools to verify an optional binding site of a benzodiazepine receptor ligand.
Colotta V; Catarzi D; Varano F; Filacchioni G; Cecchi L; Galli A; Costagli C
J Med Chem; 1996 Jul; 39(15):2915-21. PubMed ID: 8709126
[TBL] [Abstract][Full Text] [Related]
19. 3-phenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[3,4-a]phthalazines and analogues: high-affinity gamma-aminobutyric acid-A benzodiazepine receptor ligands with alpha 2, alpha 3, and alpha 5-subtype binding selectivity over alpha 1.
Carling RW; Moore KW; Street LJ; Wild D; Isted C; Leeson PD; Thomas S; O'Connor D; McKernan RM; Quirk K; Cook SM; Atack JR; Wafford KA; Thompson SA; Dawson GR; Ferris P; Castro JL
J Med Chem; 2004 Mar; 47(7):1807-22. PubMed ID: 15027873
[TBL] [Abstract][Full Text] [Related]
20. Synthesis of 7-(2-dimethylaminovinyl) derivatives of pyrazolo[1,5-a] pyrimidines, as precursors of new tricyclic series. Binding studies of BDZ receptor.
Bruni F; Costanzo A; Selleri S; Guerrini G; Giusti L; Martini C; Lucacchini A
Farmaco; 1993 Feb; 48(2):309-19. PubMed ID: 8388217
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]