BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

148 related articles for article (PubMed ID: 8230105)

  • 1. Efficient inhibition of human leukocyte elastase and cathepsin G by saccharin derivatives.
    Groutas WC; Houser-Archield N; Chong LS; Venkataraman R; Epp JB; Huang H; McClenahan JJ
    J Med Chem; 1993 Oct; 36(21):3178-81. PubMed ID: 8230105
    [TBL] [Abstract][Full Text] [Related]  

  • 2. The Gabriel-Colman rearrangement in biological systems: design, synthesis and biological evaluation of phthalimide and saccharin derivatives as potential mechanism-based inhibitors of human leukocyte elastase, cathepsin G and proteinase 3.
    Groutas WC; Chong LS; Venkataraman R; Epp JB; Kuang R; Houser-Archield N; Hoidal JR
    Bioorg Med Chem; 1995 Feb; 3(2):187-93. PubMed ID: 7796053
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Amino acid-derived phthalimide and saccharin derivatives as inhibitors of human leukocyte elastase, cathepsin G, and proteinase 3.
    Groutas WC; Chong LS; Venkataraman R; Kuang R; Epp JB; Houser-Archield N; Huang H; Hoidal JR
    Arch Biochem Biophys; 1996 Aug; 332(2):335-40. PubMed ID: 8806743
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Mechanism-based inhibition of human leukocyte elastase and cathepsin G by substituted dihydrouracils.
    Groutas WC; Huang H; Epp JB; Venkataraman R; McClenahan JJ; Tagusagawa F
    Biochim Biophys Acta; 1994 Nov; 1227(3):130-6. PubMed ID: 7986820
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Novel potential mechanism-based inhibitors of human leukocyte elastase and cathepsin G: derivatives of isothiazolidin-3-one.
    Groutas WC; Chong LS; Venkataraman R
    Biochem Biophys Res Commun; 1993 Dec; 197(2):730-9. PubMed ID: 8267609
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design, synthesis and biological evaluation of succinimide derivatives as potential mechanism-based inhibitors of human leukocyte elastase, cathepsin G and proteinase 3.
    Groutas WC; Brubaker MJ; Chong LS; Venkataraman R; Huang H; Epp JB; Kuang R; Hoidal JR
    Bioorg Med Chem; 1995 Apr; 3(4):375-81. PubMed ID: 8581420
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Substituted 3-oxo-1,2,5-thiadiazolidine 1,1-dioxides: a new class of potential mechanism-based inhibitors of human leukocyte elastase and cathepsin G.
    Groutas WC; Kuang R; Venkataraman R
    Biochem Biophys Res Commun; 1994 Jan; 198(1):341-9. PubMed ID: 8292039
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Design, synthesis, and in vitro inhibitory activity toward human leukocyte elastase, cathepsin G, and proteinase 3 of saccharin-derived sulfones and congeners.
    Groutas WC; Epp JB; Venkataraman R; Kuang R; Truong TM; McClenahan JJ; Prakash O
    Bioorg Med Chem; 1996 Sep; 4(9):1393-400. PubMed ID: 8894097
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Isoxazoline derivatives as potential inhibitors of the proteolytic enzymes human leukocyte elastase, cathepsin G and proteinase 3: a structure-activity relationship study.
    Groutas WC; Venkataraman R; Chong LS; Yoder JE; Epp JB; Stanga MA; Kim EH
    Bioorg Med Chem; 1995 Feb; 3(2):125-8. PubMed ID: 7796046
    [No Abstract]   [Full Text] [Related]  

  • 10. Novel anthraquinone inhibitors of human leukocyte elastase and cathepsin G.
    Zembower DE; Kam CM; Powers JC; Zalkow LH
    J Med Chem; 1992 May; 35(9):1597-605. PubMed ID: 1578486
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of a trihexacontapeptide corresponding to the sequence 8-70 of eglin c and studies on the relationship between the structure and the inhibitory activity against human leukocyte elastase, cathepsin G and alpha-chymotrypsin.
    Okada Y; Tsuboi S; Tsuda Y; Nagamatsu Y; Yamamoto J
    FEBS Lett; 1990 Oct; 272(1-2):113-6. PubMed ID: 2226822
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Mechanism-based inhibitors of serine proteinases based on the Gabriel-Colman rearrangement.
    Groutas WC; Chong LS; Venkataraman R; Epp JB; Kuang RZ; Brubaker MJ; Houser-Archield N; Huang H; McClenahan JJ
    Biochem Biophys Res Commun; 1993 Aug; 194(3):1491-9. PubMed ID: 8352807
    [TBL] [Abstract][Full Text] [Related]  

  • 13. The inhibition of human neutrophil elastase and cathepsin G by peptidyl 1,2-dicarbonyl derivatives.
    Mehdi S; Angelastro MR; Burkhart JP; Koehl JR; Peet NP; Bey P
    Biochem Biophys Res Commun; 1990 Jan; 166(2):595-600. PubMed ID: 2302225
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Interaction of the human leukocyte proteinases elastase and cathepsin G with gold, silver and copper compounds.
    Baici A; Camus A; Marsich N
    Biochem Pharmacol; 1984 Jun; 33(12):1859-65. PubMed ID: 6428416
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Inhibition of the human leukocyte endopeptidases elastase and cathepsin G and of porcine pancreatic elastase by N-oleoyl derivatives of heparin.
    Baici A; Diczházi C; Neszmélyi A; Móczár E; Hornebeck W
    Biochem Pharmacol; 1993 Nov; 46(9):1545-9. PubMed ID: 8240409
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Stereoselective synthesis of peptidyl trifluoromethyl alcohols and ketones: inhibitory potency against human leucocyte elastase, cathepsin G, porcine pancreatic elastase and HIV-1 protease.
    Amour A; Reboud-Ravaux M; de Rosny E; Abouabdellah A; Bégue JP; Bonnet-Delpon D; Le Gall M
    J Pharm Pharmacol; 1998 Jun; 50(6):593-600. PubMed ID: 9680068
    [TBL] [Abstract][Full Text] [Related]  

  • 17. The kinetic mechanism of inhibition of human leukocyte elastase by MR889, a new cyclic thiolic compound.
    Baici A; Pelloso R; Hörler D
    Biochem Pharmacol; 1990 Mar; 39(5):919-24. PubMed ID: 2310417
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Inhibition of human leukocyte elastase, cathepsin G, chymotrypsin A alpha, and porcine pancreatic elastase with substituted isobenzofuranones and benzopyrandiones.
    Hemmi K; Harper JW; Powers JC
    Biochemistry; 1985 Apr; 24(8):1841-8. PubMed ID: 3848330
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Ionic inhibitors of human leukocyte elastase: pyridinium and phenyl carboxylate derivatives of 3-alkyl-N-hydroxysuccinimide.
    Groutas WC; Stanga MA; Castrisos JC; Schatz EJ; Brubaker MJ
    J Pharm Sci; 1990 Oct; 79(10):886-8. PubMed ID: 2280356
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Retardation by the soybean Bowman-Birk inhibitor of elastin hydrolysis catalyzed by leukocyte proteinases.
    Tikhonova TV; Gladysheva IP; Larionova NI
    FEBS Lett; 1995 Apr; 362(2):225-8. PubMed ID: 7720877
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.