These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
125 related articles for article (PubMed ID: 8388216)
1. Benzodiazepine receptor affinity and interaction of new indole derivatives. Da Settimo A; Primofiore G; Da Settimo F; Lucacchini A; Martini C; Senatore G Farmaco; 1993 Feb; 48(2):285-95. PubMed ID: 8388216 [TBL] [Abstract][Full Text] [Related]
2. Synthesis, structure-activity relationships, and molecular modeling studies of N-(indol-3-ylglyoxylyl)benzylamine derivatives acting at the benzodiazepine receptor. Da Settimo A; Primofiore G; Da Settimo F; Marini AM; Novellino E; Greco G; Martini C; Giannaccini G; Lucacchini A J Med Chem; 1996 Dec; 39(26):5083-91. PubMed ID: 8978839 [TBL] [Abstract][Full Text] [Related]
3. Benzodiazepine receptor affinity and interaction of some N-(indol-3-ylglyoxylyl)amine derivatives. Bianucci AM; Da Settimo A; Da Settimo F; Primofiore G; Martini C; Giannaccini G; Lucacchini A J Med Chem; 1992 Jun; 35(12):2214-20. PubMed ID: 1319492 [TBL] [Abstract][Full Text] [Related]
4. N'-Phenylindol-3-ylglyoxylohydrazide derivatives: synthesis, structure-activity relationships, molecular modeling studies, and pharmacological action on brain benzodiazepine receptors. Da Settimo A; Primofiore G; Da Settimo F; Marini AM; Novellino E; Greco G; Gesi M; Martini C; Giannaccini G; Lucacchini A J Med Chem; 1998 Sep; 41(20):3821-30. PubMed ID: 9748357 [TBL] [Abstract][Full Text] [Related]
5. Synthesis and benzodiazepine receptor affinity of N-(indol-3-ylglyoxylyl)-dipeptide derivatives. Structural requirements for inverse agonist/antagonist receptor interactions. Da Settimo A; Primofiore G; Da Settimo F; Bianucci A; Martini C; Senatore G; Lucacchini A Drug Des Discov; 1993; 10(3):199-211. PubMed ID: 8268392 [TBL] [Abstract][Full Text] [Related]
6. Specific inhibition of benzodiazepine receptor binding by some N-(2-methyl or 1,2-dimethylindol-3-ylglyoxylyl)amino acid derivatives. Primofiore G; Marini AM; Da Settimo F; Salvadori C; Martini C; Lucacchini A; Giannaccini G Farmaco; 1990 Mar; 45(3):341-51. PubMed ID: 2166528 [TBL] [Abstract][Full Text] [Related]
7. N-(indol-3-ylglyoxylyl)amino acid ester derivatives. Synthesis and interaction properties at the benzodiazepine receptor. Primofiore G; Da Settimo F; Marini AM; La Motta C; Martini C; Senatore G; Lucacchini A Farmaco; 1995 Jan; 50(1):5-12. PubMed ID: 7702721 [TBL] [Abstract][Full Text] [Related]
8. Novel N-(arylalkyl)indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships. Primofiore G; Settimo FD; Taliani S; Marini AM; Novellino E; Greco G; Lavecchia A; Besnard F; Trincavelli L; Costa B; Martini C J Med Chem; 2001 Jul; 44(14):2286-97. PubMed ID: 11428922 [TBL] [Abstract][Full Text] [Related]
9. Synthesis and serotonergic activity of substituted 2, N-benzylcarboxamido-5-(2-ethyl-1-dioxoimidazolidinyl)-N, N-dimethyltryptamine derivatives: novel antagonists for the vascular 5-HT(1B)-like receptor. Moloney GP; Martin GR; Mathews N; Milne A; Hobbs H; Dodsworth S; Sang PY; Knight C; Williams M; Maxwell M; Glen RC J Med Chem; 1999 Jul; 42(14):2504-26. PubMed ID: 10411472 [TBL] [Abstract][Full Text] [Related]
10. Synthesis of 3-(2'-furoyl)indole derivatives as potential new ligands at the benzodiazepine receptor, structurally more restrained analogues of indoleglyoxylylamides. Da Settimo A; Primofiore G; Da Settimo F; Marini AM; Novellino E; Greco G; Martini C; Senatore G; Lucacchini A Farmaco; 1995 May; 50(5):311-20. PubMed ID: 7626165 [TBL] [Abstract][Full Text] [Related]
11. Isosteric replacement of amide by ester function. Synthesis and benzodiazepine receptor affinity of indol-3-ylglyoxylyl ester derivatives. Da Settimo A; Primofiore G; Marini AM; Da Settimo F; Nuti V; Martini C; Trincavelli L; Lucacchini A Farmaco; 1997; 52(6-7):421-8. PubMed ID: 9372593 [TBL] [Abstract][Full Text] [Related]
12. Novel N-substituted indol-3-ylglyoxylamides probing the LDi and L1/L2 lipophilic regions of the benzodiazepine receptor site in search for subtype-selective ligands. Primofiore G; Taliani S; Da Settimo F; Marini AM; La Motta C; Simorini F; Patrizi MP; Sergianni V; Novellino E; Greco G; Cosimelli B; Calderone V; Montali M; Besnard F; Martini C J Med Chem; 2007 Apr; 50(7):1627-34. PubMed ID: 17335185 [TBL] [Abstract][Full Text] [Related]
13. High affinity central benzodiazepine receptor ligands: synthesis and biological evaluation of a series of phenyltriazolobenzotriazindione derivatives. Primofiore G; Da Settimo F; Taliani S; Salerno S; Novellino E; Greco G; Cosimelli B; Besnard F; Costa B; Montali M; Martini C J Med Chem; 2005 Apr; 48(8):2936-43. PubMed ID: 15828832 [TBL] [Abstract][Full Text] [Related]
15. Refinement of the benzodiazepine receptor site topology by structure-activity relationships of new N-(heteroarylmethyl)indol-3-ylglyoxylamides. Primofiore G; Da Settimo F; Marini AM; Taliani S; La Motta C; Simorini F; Novellino E; Greco G; Cosimelli B; Ehlardo M; Sala A; Besnard F; Montali M; Martini C J Med Chem; 2006 Apr; 49(8):2489-95. PubMed ID: 16610792 [TBL] [Abstract][Full Text] [Related]
16. Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423) at wild type and recombinant GABAA receptors. Cox ED; Diaz-Arauzo H; Huang Q; Reddy MS; Ma C; Harris B; McKernan R; Skolnick P; Cook JM J Med Chem; 1998 Jul; 41(14):2537-52. PubMed ID: 9651158 [TBL] [Abstract][Full Text] [Related]
17. Studies on annelated 1,4-benzothiazines and 1,5-benzothiazepines. X--Synthesis and inhibition of benzodiazepine receptor binding of new 1,4-thiazine and 1,5-thiazepine polycondensed heterocycles with steroidal structure. Grandolini G; Ambrogi V; Perioli L; Giannaccini G; Lucacchini A; Martini C Farmaco; 1996 Mar; 51(3):203-7. PubMed ID: 8688143 [TBL] [Abstract][Full Text] [Related]
18. 2,3-Dihydro-2-oxo-1H-benzimidazole-1-carboxamides with selective affinity for the 5-HT(4) receptor: synthesis and structure-affinity and structure-activity relationships of a new series of partial agonist and antagonist derivatives. Tapia I; Alonso-Cires L; López-Tudanca PL; Mosquera R; Labeaga L; Innerárity A; Orjales A J Med Chem; 1999 Jul; 42(15):2870-80. PubMed ID: 10425096 [TBL] [Abstract][Full Text] [Related]
19. Synthesis of new 6H-indolo[2,3-b] [1,8]naphthyridines and their specific inhibition of benzodiazepine receptor. Da Settimo A; Primofiore G; Ferrarini PL; Mori C; Martini C; Pennacchi E; Lucacchini A Farmaco Sci; 1986 Aug; 41(8):577-85. PubMed ID: 3017748 [TBL] [Abstract][Full Text] [Related]
20. New 2,3-substituted 4,7-dihydro-6-(1'H-pyrazol-3'-yl)pyrazolo[1,5-a] pyrimidin-7-ones and related compounds: synthesis and benzodiazepine receptor binding study. Selleri S; Bruni F; Costanzo A; Guerrini G; Casilli ML; Giusti L; Lucacchini A; Martini C Farmaco; 1995 Oct; 50(10):679-87. PubMed ID: 8590575 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]