203 related articles for article (PubMed ID: 8544181)
1. Syntheses and antimalarial activities of N-substituted 11-azaartemisinins.
Torok DS; Ziffer H; Meshnick SR; Pan XQ; Ager A
J Med Chem; 1995 Dec; 38(26):5045-50. PubMed ID: 8544181
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and antimalarial activities of fluoroalkyl derivatives of dihydroartemisinin.
Thanh Nga TT; Ménage C; Bégué JP; Bonnet-Delpon D; Gantier JC; Pradines B; Doury JC; Thac TD
J Med Chem; 1998 Oct; 41(21):4101-8. PubMed ID: 9767645
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and antimalarial activities of base-catalyzed adducts of 11-azaartemisinin.
Mekonnen B; Weiss E; Katz E; Ma J; Ziffer H; Kyle DE
Bioorg Med Chem; 2000 May; 8(5):1111-6. PubMed ID: 10882021
[TBL] [Abstract][Full Text] [Related]
4. Structure-activity relationships of the antimalarial agent artemisinin. 2. Effect of heteroatom substitution at O-11: synthesis and bioassay of N-alkyl-11-aza-9-desmethylartemisinins.
Avery MA; Bonk JD; Chong WK; Mehrotra S; Miller R; Milhous W; Goins DK; Venkatesan S; Wyandt C; Khan I
J Med Chem; 1995 Dec; 38(26):5038-44. PubMed ID: 8544180
[TBL] [Abstract][Full Text] [Related]
5. Antimalarial activity of new dihydroartemisinin derivatives. 7. 4-(p-substituted phenyl)-4(R or S)-[10(alpha or beta)-dihydroartemisininoxy]butyric acids.
Lin AJ; Zikry AB; Kyle DE
J Med Chem; 1997 Apr; 40(9):1396-400. PubMed ID: 9135037
[TBL] [Abstract][Full Text] [Related]
6. Structure-activity relationships of the antimalarial agent artemisinin. 7. Direct modification of (+)-artemisinin and in vivo antimalarial screening of new, potential preclinical antimalarial candidates.
Avery MA; Alvim-Gaston M; Vroman JA; Wu B; Ager A; Peters W; Robinson BL; Charman W
J Med Chem; 2002 Sep; 45(19):4321-35. PubMed ID: 12213073
[TBL] [Abstract][Full Text] [Related]
7. Syntheses and antimalarial activities of 10-substituted deoxoartemisinins.
Ma J; Katz E; Kyle DE; Ziffer H
J Med Chem; 2000 Nov; 43(22):4228-32. PubMed ID: 11063619
[TBL] [Abstract][Full Text] [Related]
8. Antimalarial activity of novel ring-contracted artemisinin derivatives.
Venugopalan B; Bapat CP; Karnik PJ; Chatterjee DK; Iyer N; Lepcha D
J Med Chem; 1995 May; 38(11):1922-7. PubMed ID: 7783124
[TBL] [Abstract][Full Text] [Related]
9. Structure-activity relationships of lactone ring-opened analogs of the antimalarial 1,2,4-trioxane artemisinin.
Posner GH; McGarvey DJ; Oh CH; Kumar N; Meshnick SR; Asawamahasadka W
J Med Chem; 1995 Feb; 38(4):607-12. PubMed ID: 7861408
[TBL] [Abstract][Full Text] [Related]
10. Synthesis of new artemisinin analogues from artemisinic acid modified at C-3 and C-13 and their antimalarial activity.
Han J; Lee JG; Min SS; Park SH; Angerhofer CK; Cordell GA; Kim SU
J Nat Prod; 2001 Sep; 64(9):1201-5. PubMed ID: 11575956
[TBL] [Abstract][Full Text] [Related]
11. Convenient access both to highly antimalaria-active 10-arylaminoartemisinins, and to 10-alkyl ethers including artemether, arteether, and artelinate.
Haynes RK; Chan HW; Ho WY; Ko CK; Gerena L; Kyle DE; Peters W; Robinson BL
Chembiochem; 2005 Apr; 6(4):659-67. PubMed ID: 15812783
[TBL] [Abstract][Full Text] [Related]
12. Fluoroartemisinin: trifluoromethyl analogues of artemether and artesunate.
Magueur G; Crousse B; Charneau S; Grellier P; Bégué JP; Bonnet-Delpon D
J Med Chem; 2004 May; 47(10):2694-9. PubMed ID: 15115411
[TBL] [Abstract][Full Text] [Related]
13. Synthesis and antimalarial activity of some 9-substituted artemisinin derivatives.
Acton N; Karle JM; Miller RE
J Med Chem; 1993 Aug; 36(17):2552-7. PubMed ID: 8355254
[TBL] [Abstract][Full Text] [Related]
14. Structure and antimalarial activity of adducts of 11-azaartemisinin with conjugated terminal acetylenes.
Katz E; Ma J; Kyle D; Ziffer H
Bioorg Med Chem Lett; 1999 Oct; 9(20):2969-72. PubMed ID: 10571157
[TBL] [Abstract][Full Text] [Related]
15. Synthesis, antimalarial activity, biomimetic iron(II) chemistry, and in vivo metabolism of novel, potent C-10-phenoxy derivatives of dihydroartemisinin.
O'Neill PM; Miller A; Bishop LP; Hindley S; Maggs JL; Ward SA; Roberts SM; Scheinmann F; Stachulski AV; Posner GH; Park BK
J Med Chem; 2001 Jan; 44(1):58-68. PubMed ID: 11141088
[TBL] [Abstract][Full Text] [Related]
16. Mechanism-based design of parasite-targeted artemisinin derivatives: synthesis and antimalarial activity of benzylamino and alkylamino ether analogues of artemisinin.
O'Neill PM; Bishop LP; Storr RC; Hawley SR; Maggs JL; Ward SA; Park BK
J Med Chem; 1996 Oct; 39(22):4511-4. PubMed ID: 8893847
[TBL] [Abstract][Full Text] [Related]
17. Antimalarial activity of new water-soluble dihydroartemisinin derivatives. 3. Aromatic amine analogues.
Lin AJ; Li LQ; Klayman DL; George CF; Flippen-Anderson JL
J Med Chem; 1990 Sep; 33(9):2610-4. PubMed ID: 2202831
[TBL] [Abstract][Full Text] [Related]
18. Structure-activity relationships of the antimalarial agent artemisinin. 4. Effect of substitution at C-3.
Avery MA; Mehrotra S; Bonk JD; Vroman JA; Goins DK; Miller R
J Med Chem; 1996 Jul; 39(15):2900-6. PubMed ID: 8709124
[TBL] [Abstract][Full Text] [Related]
19. Correlation of antimalarial activity of artemisinin derivatives with binding affinity with ferroprotoporphyrin IX.
Paitayatat S; Tarnchompoo B; Thebtaranonth Y; Yuthavong Y
J Med Chem; 1997 Feb; 40(5):633-8. PubMed ID: 9057849
[TBL] [Abstract][Full Text] [Related]
20. C-16 artemisinin derivatives and their antimalarial and cytotoxic activities: syntheses of artemisinin monomers, dimers, trimers, and tetramers by nucleophilic additions to artemisitene.
Ekthawatchai S; Kamchonwongpaisan S; Kongsaeree P; Tarnchompoo B; Thebtaranonth Y; Yuthavong Y
J Med Chem; 2001 Dec; 44(26):4688-95. PubMed ID: 11741486
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]