BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

128 related articles for article (PubMed ID: 8545542)

  • 21. Medicinal chemistry of indolylglyoxylamide GABAA/BzR high affinity ligands: identification of novel anxiolytic/non sedative agents.
    Salerno S; Da Settimo F; Taliani S; Simorini F; La Motta C; Fornaciari G; Marini AM
    Curr Top Med Chem; 2012; 12(4):286-311. PubMed ID: 22204484
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Synthetic and computer-assisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors.
    Wong G; Koehler KF; Skolnick P; Gu ZQ; Ananthan S; Schönholzer P; Hunkeler W; Zhang W; Cook JM
    J Med Chem; 1993 Jun; 36(13):1820-30. PubMed ID: 8390574
    [TBL] [Abstract][Full Text] [Related]  

  • 23. Synthesis and structure-activity relationships of 3,5-disubstituted 4,5-dihydro-6H-imidazo[1,5-a][1,4]benzodiazepin-6-ones at diazepam-sensitive and diazepam-insensitive benzodiazepine receptors.
    Ananthan S; Clayton SD; Ealick SE; Wong G; Evoniuk GE; Skolnick P
    J Med Chem; 1993 Feb; 36(4):479-90. PubMed ID: 8386247
    [TBL] [Abstract][Full Text] [Related]  

  • 24. Electrophysiology of benzodiazepine receptor ligands: multiple mechanisms and sites of action.
    Polc P
    Prog Neurobiol; 1988; 31(5):349-423. PubMed ID: 2851856
    [TBL] [Abstract][Full Text] [Related]  

  • 25. Relationship between benzodiazepine receptor occupancy and potentiation of gamma-aminobutyric acid-stimulated chloride flux in vitro of four ligands of differing intrinsic efficacies.
    Facklam M; Schoch P; Haefely WE
    J Pharmacol Exp Ther; 1992 Jun; 261(3):1106-12. PubMed ID: 1318370
    [TBL] [Abstract][Full Text] [Related]  

  • 26. Synthesis of benzo-fused benzodiazepines employed as probes of the agonist pharmacophore of benzodiazepine receptors.
    Zhang W; Koehler KF; Harris B; Skolnick P; Cook JM
    J Med Chem; 1994 Mar; 37(6):745-57. PubMed ID: 8145224
    [TBL] [Abstract][Full Text] [Related]  

  • 27. 3D-pharmacophores of flavonoid binding at the benzodiazepine GABA(A) receptor site using 4D-QSAR analysis.
    Hong X; Hopfinger AJ
    J Chem Inf Comput Sci; 2003; 43(1):324-36. PubMed ID: 12546568
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Geometrically constrained derivatives of indolylglyoxylamides as ligands binding the GABAA/BzR complex.
    Sartini S; Morelli M; Simorini F; Taliani S; Salerno S; Marini AM; Da Settimo F; La Motta C
    Curr Top Med Chem; 2012; 12(4):312-20. PubMed ID: 22204489
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Synthesis, structure-activity relationships, and molecular modeling studies of N-(indol-3-ylglyoxylyl)benzylamine derivatives acting at the benzodiazepine receptor.
    Da Settimo A; Primofiore G; Da Settimo F; Marini AM; Novellino E; Greco G; Martini C; Giannaccini G; Lucacchini A
    J Med Chem; 1996 Dec; 39(26):5083-91. PubMed ID: 8978839
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Bidirectional modulation of cortical acetylcholine efflux by infusion of benzodiazepine receptor ligands into the basal forebrain.
    Moore H; Sarter M; Bruno JP
    Neurosci Lett; 1995 Apr; 189(1):31-4. PubMed ID: 7603619
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Determinants of recognition of ligands binding to benzodiazepine receptor/GABA(A) receptors initiating sedation.
    Harris DL; DeLorey TM; He X; Cook JM; Loew GH
    Eur J Pharmacol; 2000 Aug; 401(3):271-87. PubMed ID: 10936485
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Structure-activity relationships of 1,2,4-triazolo[1,5-a] quinoxalines and their 1-deaza analogues imidazo[1,2-a]quinoxalines at the benzodiazepine receptor.
    Catarzi D; Cecchi L; Colotta V; Melani F; Filacchioni G; Martini C; Giusti L; Lucacchini A
    J Med Chem; 1994 Sep; 37(18):2846-50. PubMed ID: 8071933
    [TBL] [Abstract][Full Text] [Related]  

  • 33. New 2,3-substituted 4,7-dihydro-6-(1'H-pyrazol-3'-yl)pyrazolo[1,5-a] pyrimidin-7-ones and related compounds: synthesis and benzodiazepine receptor binding study.
    Selleri S; Bruni F; Costanzo A; Guerrini G; Casilli ML; Giusti L; Lucacchini A; Martini C
    Farmaco; 1995 Oct; 50(10):679-87. PubMed ID: 8590575
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Development of radioligands for in vivo imaging of GABA(A)-benzodiazepine receptors.
    Katsifis A; Kassiou M
    Mini Rev Med Chem; 2004 Oct; 4(8):909-21. PubMed ID: 15544552
    [TBL] [Abstract][Full Text] [Related]  

  • 35. GABA A/Bz receptor subtypes as targets for selective drugs.
    Da Settimo F; Taliani S; Trincavelli ML; Montali M; Martini C
    Curr Med Chem; 2007; 14(25):2680-701. PubMed ID: 17979718
    [TBL] [Abstract][Full Text] [Related]  

  • 36. The story of flumazenil.
    Haefely W; Hunkeler W
    Eur J Anaesthesiol Suppl; 1988; 2():3-13. PubMed ID: 2842141
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Benzodiazepine receptor binding activity of 8-substituted-9-(3-substituted-benzyl)-6-(dimethylamino)-9H-purines.
    Kelley JL; McLean EW; Linn JA; Krochmal MP; Ferris RM; Howard JL
    J Med Chem; 1990 Jan; 33(1):196-202. PubMed ID: 1967311
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Novel 3-aroylpyrazolo[5,1-c][1,2,4]benzotriazine 5-oxides 8-substituted, ligands at GABAA/benzodiazepine receptor complex: synthesis, pharmacological and molecular modeling studies.
    Guerrini G; Ciciani G; Cambi G; Bruni F; Selleri S; Melani F; Montali M; Martini C; Ghelardini C; Norcini M; Costanzo A
    Bioorg Med Chem; 2008 Apr; 16(8):4471-89. PubMed ID: 18325771
    [TBL] [Abstract][Full Text] [Related]  

  • 39. 2-Aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones: novel rigid planar benzodiazepine receptor ligands.
    Campagna F; Carotti A; Casini G; Palluotto F; Genchi G; De Sarro GB
    Bioorg Med Chem; 1993 Dec; 1(6):437-46. PubMed ID: 8087565
    [TBL] [Abstract][Full Text] [Related]  

  • 40. Benzodiazepine receptor ligands. 8: synthesis and pharmacological evaluation of new pyrazolo[5,1-c] [1,2,4]benzotriazine 5-oxide 3- and 8-disubstituted: high affinity ligands endowed with inverse-agonist pharmacological efficacy.
    Guerrini G; Costanzo A; Ciciani G; Bruni F; Selleri S; Costagli C; Besnard F; Costa B; Martini C; De Siena G; Malmberg-Aiello P
    Bioorg Med Chem; 2006 Feb; 14(3):758-75. PubMed ID: 16214350
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 7.