These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
195 related articles for article (PubMed ID: 8667368)
41. Synthesis and structure-activity studies on N-[5-(1H-imidazol-4-yl)-5,6,7,8-tetrahydro-1-naphthalenyl]methanesulfonamide, an imidazole-containing alpha(1A)-adrenoceptor agonist. Altenbach RJ; Khilevich A; Kolasa T; Rohde JJ; Bhatia PA; Patel MV; Searle XB; Yang F; Bunnelle WH; Tietje K; Bayburt EK; Carroll WA; Meyer MD; Henry R; Buckner SA; Kuk J; Daza AV; Milicic IV; Cain JC; Kang CH; Ireland LM; Carr TL; Miller TR; Hancock AA; Nakane M; Esbenshade TA; Brune ME; O'Neill AB; Gauvin DM; Katwala SP; Holladay MW; Brioni JD; Sullivan JP J Med Chem; 2004 Jun; 47(12):3220-35. PubMed ID: 15163201 [TBL] [Abstract][Full Text] [Related]
42. 3-Phenyl analogues of 2-[[[2-(2,6-dimethoxyphenoxy)ethyl]amino]-methyl]-1,4-benzodioxan (WB 4101) as highly selective alpha 1-adrenoceptor antagonists. Quaglia W; Pigini M; Giannella M; Melchiorre C J Med Chem; 1990 Nov; 33(11):2946-8. PubMed ID: 1977906 [No Abstract] [Full Text] [Related]
43. AMPA receptor agonists: resolution, configurational assignment, and pharmacology of (+)-(S)- and (-)-(R)-2-amino-3-[3-hydroxy-5-(2-pyridyl)-isoxazol-4-yl]-propionic acid (2-Py-AMPA). Johansen TN; Ebert B; Falch E; Krogsgaard-Larsen P Chirality; 1997; 9(3):274-80. PubMed ID: 9176992 [TBL] [Abstract][Full Text] [Related]
44. De novo design, synthesis, and biological activities of high-affinity and selective non-peptide agonists of the delta-opioid receptor. Liao S; Alfaro-Lopez J; Shenderovich MD; Hosohata K; Lin J; Li X; Stropova D; Davis P; Jernigan KA; Porreca F; Yamamura HI; Hruby VJ J Med Chem; 1998 Nov; 41(24):4767-76. PubMed ID: 9822547 [TBL] [Abstract][Full Text] [Related]
45. Characterization of the binding site of the histamine H3 receptor. 1. Various approaches to the synthesis of 2-(1H-imidazol-4-yl)cyclopropylamine and histaminergic activity of (1R,2R)- and (1S,2S)-2-(1H-imidazol-4-yl)-cyclopropylamine. De Esch IJ; Vollinga RC; Goubitz K; Schenk H; Appelberg U; Hacksell U; Lemstra S; Zuiderveld OP; Hoffmann M; Leurs R; Menge WM; Timmerman H J Med Chem; 1999 Apr; 42(7):1115-22. PubMed ID: 10197956 [TBL] [Abstract][Full Text] [Related]
46. Absolute configuration and biological activity of mequitamium iodide enantiomers. Di Bugno C; Dapporto P; Giorgi R; Manzini S; Paoli P; Subissi A; Arcamone F Chirality; 1994; 6(5):382-8. PubMed ID: 8068497 [TBL] [Abstract][Full Text] [Related]
47. Absolute configuration of glycerol derivatives. 4. Synthesis and pharmacological activity of chiral 2-alkylaminomethylbenzodioxans, competitive alpha-adrenergic antagonists. Nelson WL; Wennerstrom JE; Dyer DC; Engel JE J Med Chem; 1977 Jul; 20(7):880-5. PubMed ID: 17749 [TBL] [Abstract][Full Text] [Related]
48. Analogues of prazosin that bear a benextramine-related polyamine backbone exhibit different antagonism toward alpha1-adrenoreceptor subtypes. Bolognesi ML; Marucci G; Angeli P; Buccioni M; Minarini A; Rosini M; Tumiatti V; Melchiorre C J Med Chem; 2001 Feb; 44(3):362-71. PubMed ID: 11462977 [TBL] [Abstract][Full Text] [Related]
49. Structure-activity relationships in 1,4-benzodioxan-related compounds. Investigation on the role of the dehydrodioxane ring on alpha 1-adrenoreceptor blocking activity. Pigini M; Brasili L; Giannella M; Giardinà D; Gulini U; Quaglia W; Melchiorre C J Med Chem; 1988 Dec; 31(12):2300-4. PubMed ID: 2903932 [TBL] [Abstract][Full Text] [Related]
50. 2-[[[2-(2,6-Dimethoxyphenoxy)ethyl]amino]-methyl] -1,4-benzoxathian: a new antagonist with high potency and selectivity toward alpha 1-adrenoreceptors. Melchiorre C; Brasili L; Giardinà D; Pigini M; Strappaghetti G J Med Chem; 1984 Dec; 27(12):1535-6. PubMed ID: 6150111 [No Abstract] [Full Text] [Related]
51. Stereoselectivity at alpha-adrenoreceptor subtypes: observations with the enantiomers of WB 4101 separated through their amides of N-tosyl-(S)-proline. Andrisano V; Marucci G; Melchiorre C; Tumiatti V Chirality; 1992; 4(1):16-20. PubMed ID: 1353682 [TBL] [Abstract][Full Text] [Related]
52. [Synthesis and alpha-adrenolytic activities of 2-(1,4-benzodioxan-2-yl- methyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline derivatives]. Glusa E; Grüner H; Hagen A; Lohmann D; Foken H Pharmazie; 1990 Jun; 45(6):408-10. PubMed ID: 1976262 [TBL] [Abstract][Full Text] [Related]
53. Design, synthesis and alpha1-adrenoreceptor blocking activity of new arylpiperazines containing acetophenone substituents. Huang JJ; Huang YJ; Zhu L; Yuan M; Huang L Pharmazie; 2014 Aug; 69(8):578-84. PubMed ID: 25158567 [TBL] [Abstract][Full Text] [Related]
54. Alpha-adrenoreceptor reagents. 3. Synthesis of some 2-substituted 1,4-benzodioxans as selective presynaptic alpha 2-adrenoreceptor antagonists. Stillings MR; Chapleo CB; Butler RC; Davis JA; England CD; Myers M; Myers PL; Tweddle N; Welbourn AP; Doxey JC J Med Chem; 1985 Aug; 28(8):1054-62. PubMed ID: 2862284 [TBL] [Abstract][Full Text] [Related]
55. New 2-substituted 2,3,3a,4-tetrahydro-1H-imidazo[5,1-c] [1,4]benzoxazin-1-ones as alpha 2-adrenoceptor antagonists. Melloni P; Banzatti C; Heidempergher F; Marazzi G; Ricciardi S; Vaghi F; Varasi M Farmaco; 1991 Sep; 46(9):1011-21. PubMed ID: 1687241 [TBL] [Abstract][Full Text] [Related]
56. Design, synthesis, and structure-activity relationships of phthalimide-phenylpiperazines: a novel series of potent and selective alpha(1)(a)-adrenergic receptor antagonists. Kuo GH; Prouty C; Murray WV; Pulito V; Jolliffe L; Cheung P; Varga S; Evangelisto M; Wang J J Med Chem; 2000 Jun; 43(11):2183-95. PubMed ID: 10841797 [TBL] [Abstract][Full Text] [Related]
57. alpha-adrenoreceptor reagents. 1. Synthesis of some 1,4-benzodioxans as selective presynaptic alpha 2-adrenoreceptor antagonists and potential antidepressants. Chapleo CB; Myers PL; Butler RC; Doxey JC; Roach AG; Smith CF J Med Chem; 1983 Jun; 26(6):823-31. PubMed ID: 6133953 [TBL] [Abstract][Full Text] [Related]
58. Structure-activity relationship study on alpha1 adrenergic receptor antagonists from beer. Wakimoto T; Nitta M; Kasahara K; Chiba T; Ye Y; Tsuji K; Kan T; Nukaya H; Ishiguro M; Koike M; Yokoo Y; Suwa Y Bioorg Med Chem Lett; 2009 Oct; 19(20):5905-8. PubMed ID: 19762239 [TBL] [Abstract][Full Text] [Related]
59. Structure--activity relationships among novel phenoxybenzamine-related beta-chloroethylamines. Giardinà D; Crucianelli M; Angeli P; Buccioni M; Gulini U; Marucci G; Sagratini G; Melchiorre C Bioorg Med Chem; 2002 May; 10(5):1291-303. PubMed ID: 11886792 [TBL] [Abstract][Full Text] [Related]
60. Rigid analogues of the α2-adrenergic blocker atipamezole: small changes, big consequences. Vacher B; Funes P; Chopin P; Cussac D; Heusler P; Tourette A; Marien M J Med Chem; 2010 Oct; 53(19):6986-95. PubMed ID: 20809632 [TBL] [Abstract][Full Text] [Related] [Previous] [Next] [New Search]