These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

109 related articles for article (PubMed ID: 8770391)

  • 1. Affinity probes for the GABA-gated chloride channel: selection of 5e-tert-butyl-2e-[4-(substituted-ethynyl)phenyl]-1,3-dithianes and optimization of linker moiety.
    Li QX; Casida JE
    Bioorg Med Chem; 1995 Dec; 3(12):1667-74. PubMed ID: 8770391
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Affinity probes for the GABA-gated chloride channel: 5e-tert-butyl-2e-[4-(substituted-ethynyl)phenyl]-1,3-dithianes with photoactivatable, fluorescent, biotin, agarose and protein substituents.
    Li QX; Casida JE
    Bioorg Med Chem; 1995 Dec; 3(12):1675-84. PubMed ID: 8770392
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Structure-activity studies leading to potent chloride channel blockers: 5e-tert-Butyl-2-[4-(substituted-ethynyl)phenyl]-1,3-dithianes.
    Li QX; Casida JE
    Bioorg Med Chem; 1994 Dec; 2(12):1423-34. PubMed ID: 7788306
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Photoactivatable 2-(4'-azidotetrafluorophenyl)-5-tert-butyl-1,3-dithiane-bis- sulfone and related compounds as candidate irreversible probes for the GABA-gated chloride channels.
    Kapfer I; Hawkinson JE; Casida JE; Goeldner MP
    J Med Chem; 1994 Jan; 37(1):133-40. PubMed ID: 8289186
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Characterization of [3H]ethynylbicycloorthobenzoate ([3H]EBOB) binding and the action of insecticides on the gamma-aminobutyric acid-gated chloride channel in cultured cerebellar granule neurons.
    Huang J; Casida JE
    J Pharmacol Exp Ther; 1996 Dec; 279(3):1191-6. PubMed ID: 8968340
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis of carbon-11-, fluorine-18-, and iodine-125-labeled GABAA-gated chloride ion channel blockers: substituted 5-tert-butyl-2-phenyl-1,3-dithianes and -dithiane oxides.
    Snyder SE; Kume A; Jung YW; Connor SE; Sherman PS; Albin RL; Wieland DM; Kilbourn MR
    J Med Chem; 1995 Jul; 38(14):2663-71. PubMed ID: 7629805
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Drosophila GABA-gated chloride channel: modified [3H]EBOB binding site associated with Ala-->Ser or Gly mutants of Rdl subunit.
    Cole LM; Roush RT; Casida JE
    Life Sci; 1995; 56(10):757-65. PubMed ID: 7885191
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Actions of cyclic esters, S-esters, and amides of phenyl- and phenylthiophosphonic acids on mammalian and insect GABA-gated chloride channels.
    Ozoe Y; Niina K; Matsumoto K; Ikeda I; Mochida K; Ogawa C; Matsuno A; Miki M; Yanagi K
    Bioorg Med Chem; 1998 Jan; 6(1):73-83. PubMed ID: 9502107
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Binding kinetics of gamma-aminobutyric acidA receptor noncompetitive antagonists: trioxabicyclooctane, dithiane, and cyclodiene insecticide-induced slow transition to blocked chloride channel conformation.
    Hawkinson JE; Casida JE
    Mol Pharmacol; 1992 Dec; 42(6):1069-76. PubMed ID: 1282663
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Avermectin B1a binds to high- and low-affinity sites with dual effects on the gamma-aminobutyric acid-gated chloride channel of cultured cerebellar granule neurons.
    Huang J; Casida JE
    J Pharmacol Exp Ther; 1997 Apr; 281(1):261-6. PubMed ID: 9103505
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Insecticide action at the GABA-gated chloride channel: recognition, progress, and prospects.
    Casida JE
    Arch Insect Biochem Physiol; 1993; 22(1-2):13-23. PubMed ID: 7679302
    [TBL] [Abstract][Full Text] [Related]  

  • 12. 5-[4-(3,3-Dimethylbutoxycarbonyl)phenyl]-4-pentynoic acid and its derivatives inhibit ionotropic gamma-aminobutyric acid receptors by binding to the 4'-ethynyl-4-n-propylbicycloorthobenzoate site.
    Hamano H; Nagata K; Fukada TN; Shimotahira H; Ju XL; Ozoe Y
    Bioorg Med Chem; 2000 Mar; 8(3):665-74. PubMed ID: 10732984
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Comparative photoaffinity labeling study between azidophenyl, difluoroazidophenyl, and tetrafluoroazidophenyl derivatives for the GABA-gated chloride channels.
    Kapfer I; Jacques P; Toubal H; Goeldner MP
    Bioconjug Chem; 1995; 6(1):109-14. PubMed ID: 7711096
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Effects of [3H]-BIDN, a novel bicyclic dinitrile radioligand for GABA-gated chloride channels of insects and vertebrates.
    Rauh JJ; Benner E; Schnee ME; Cordova D; Holyoke CW; Howard MH; Bai D; Buckingham SD; Hutton ML; Hamon A; Roush RT; Sattelle DB
    Br J Pharmacol; 1997 Aug; 121(7):1496-505. PubMed ID: 9257933
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and structure-activity relationships of 1-phenyl-1H-1,2,3-triazoles as selective insect GABA receptor antagonists.
    Alam MS; Kajiki R; Hanatani H; Kong X; Ozoe F; Matsui Y; Matsumura F; Ozoe Y
    J Agric Food Chem; 2006 Feb; 54(4):1361-72. PubMed ID: 16478261
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Inhibition of GABA-gated chloride channels by 12,14-dichlorodehydroabietic acid in mammalian brain.
    Nicholson RA; Lees G; Zheng J; Verdon B
    Br J Pharmacol; 1999 Mar; 126(5):1123-32. PubMed ID: 10204999
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Differential blocking actions of 4'-ethynyl-4-n-propylbicycloorthobenzoate (EBOB) and gamma-hexachlorocyclohexane (gamma-HCH) on gamma-aminobutyric acid- and glutamate-induced responses of American cockroach neurons.
    Ihara M; Ishida C; Okuda H; Ozoe Y; Matsuda K
    Invert Neurosci; 2005 Nov; 5(3-4):157-64. PubMed ID: 16195902
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Unique insecticide specificity of human homomeric rho 1 GABA(C) receptor.
    Ratra GS; Erkkila BE; Weiss DS; Casida JE
    Toxicol Lett; 2002 Mar; 129(1-2):47-53. PubMed ID: 11879973
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Bicycloorthocarboxylate convulsants. Potent GABAA receptor antagonists.
    Casida JE; Palmer CJ; Cole LM
    Mol Pharmacol; 1985 Sep; 28(3):246-53. PubMed ID: 2993847
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Chloride channels as tools for developing selective insecticides.
    Bloomquist JR
    Arch Insect Biochem Physiol; 2003 Dec; 54(4):145-56. PubMed ID: 14635176
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.