BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

95 related articles for article (PubMed ID: 8772187)

  • 1. Alkynyl phosphates are potent inhibitors of serine enzyme.
    Segal D; Shalitin C; Shalitin Y; Fischer DR; Stang PJ
    FEBS Lett; 1996 Aug; 392(2):117-20. PubMed ID: 8772187
    [TBL] [Abstract][Full Text] [Related]  

  • 2. The interaction of alkynyl carboxylates with serine enzymes. A potent new class of serine enzyme inhibitors.
    Segal D; Shalitin Y; Wingert H; Kitamura T; Stang PJ
    FEBS Lett; 1989 Apr; 247(2):217-20. PubMed ID: 2714433
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Mechanism-based inactivation of phosphotriesterase by reaction of a critical histidine with a ketene intermediate.
    Banzon JA; Kuo JM; Miles BW; Fischer DR; Stang PJ; Raushel FM
    Biochemistry; 1995 Jan; 34(3):743-9. PubMed ID: 7827032
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Irreversible inhibition of serine proteases by peptidyl derivatives of alpha-aminoalkylphosphonate diphenyl esters.
    Oleksyszyn J; Powers JC
    Biochem Biophys Res Commun; 1989 May; 161(1):143-9. PubMed ID: 2730652
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Irreversible inhibition of serine proteases by peptide derivatives of (alpha-aminoalkyl)phosphonate diphenyl esters.
    Oleksyszyn J; Powers JC
    Biochemistry; 1991 Jan; 30(2):485-93. PubMed ID: 1988040
    [TBL] [Abstract][Full Text] [Related]  

  • 6. The serpin MNEI inhibits elastase-like and chymotrypsin-like serine proteases through efficient reactions at two active sites.
    Cooley J; Takayama TK; Shapiro SD; Schechter NM; Remold-O'Donnell E
    Biochemistry; 2001 Dec; 40(51):15762-70. PubMed ID: 11747453
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Inactivation of chymotrypsin and human skin chymase: kinetics of time-dependent inhibition in the presence of substrate.
    Johnson LA; Moon KE; Eisenberg M
    Biochim Biophys Acta; 1988 Apr; 953(3):269-79. PubMed ID: 2451541
    [TBL] [Abstract][Full Text] [Related]  

  • 8. A comparative study of antichymotryptic and anticholinesterase activity of organophosphorus quasi-substrate inhibitors.
    Rozengart EV
    Dokl Biochem Biophys; 2008; 419():82-7. PubMed ID: 18505164
    [No Abstract]   [Full Text] [Related]  

  • 9. Synthesis and kinetic studies of an amidine-containing phosphonofluoridate: a novel potent inhibitor of trypsin-like enzymes.
    Ni LM; Powers JC
    Bioorg Med Chem; 1998 Oct; 6(10):1767-73. PubMed ID: 9839006
    [TBL] [Abstract][Full Text] [Related]  

  • 10. N-tosyl-L-phenylalanine chloromethyl ketone, a serine protease inhibitor, identifies glutamate 398 at the coenzyme-binding site of human aldehyde dehydrogenase. Evidence for a second "naked anion" at the active site.
    Dryjanski M; Kosley LL; Pietruszko R
    Biochemistry; 1998 Oct; 37(40):14151-6. PubMed ID: 9760251
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Utilization of biotinylated diphenyl phosphonates for disclosure of serine proteases.
    Hawthorne S; Hamilton R; Walker BJ; Walker B
    Anal Biochem; 2004 Mar; 326(2):273-5. PubMed ID: 15003568
    [No Abstract]   [Full Text] [Related]  

  • 12. [Biochemical characteristics of aminostigmine--a new anticholinesterase agent].
    Prozorovskiĭ VB; Rozengart VI; Ardab'eva TV; Kugusheva LI; Suslova IM
    Biokhimiia; 1996 Apr; 61(4):690-6. PubMed ID: 8724787
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Model equations for the kinetics of covalent irreversible enzyme inhibition and spontaneous reactivation: esterases and organophosphorus compounds.
    Estevez J; Vilanova E
    Crit Rev Toxicol; 2009; 39(5):427-48. PubMed ID: 19514915
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Interactions of oxime reactivators with diethylphosphoryl adducts of human acetylcholinesterase and its mutant derivatives.
    Grosfeld H; Barak D; Ordentlich A; Velan B; Shafferman A
    Mol Pharmacol; 1996 Sep; 50(3):639-49. PubMed ID: 8794905
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Novel diphenyl esters of peptidyl alpha-aminoalkylphosphonates as inhibitors of chymotrypsin and subtilisin.
    Pietrusewicz E; Sieńczyk M; Oleksyszyn J
    J Enzyme Inhib Med Chem; 2009 Dec; 24(6):1229-36. PubMed ID: 19912056
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Interactions between acetylcholinesterase, toxic organophosphorus compounds and a short series of structurally related non-oxime reactivators: Analysis of reactivation and inhibition kinetics in vitro.
    Horn G; de Koning MC; van Grol M; Thiermann H; Worek F
    Toxicol Lett; 2018 Dec; 299():218-225. PubMed ID: 30312685
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Dipeptide-derived diphenyl phosphonate esters: mechanism-based inhibitors of dipeptidyl peptidase IV.
    Lambeir AM; Borloo M; De Meester I; Belyaev A; Augustyns K; Hendriks D; Scharpé S; Haemers A
    Biochim Biophys Acta; 1996 May; 1290(1):76-82. PubMed ID: 8645710
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Failure of toxogonin to reactivate soman-inhibited brain acetylcholinesterase in monkeys and regeneration of the enzyme.
    Filbert MG; Fleisher JH; Lochner MA
    Biochim Biophys Acta; 1972 Sep; 284(1):164-74. PubMed ID: 4627450
    [No Abstract]   [Full Text] [Related]  

  • 19. Histidine-254 is essential for the inactivation of phosphotriesterase with the alkynyl phosphate esters and diethyl pyrocarbonate.
    Banzon JA; Kuo JM; Fischer DR; Stang PJ; Raushel FM
    Biochemistry; 1995 Jan; 34(3):750-4. PubMed ID: 7827033
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis and in vitro kinetic study of novel mono-pyridinium oximes as reactivators of organophosphorus (OP) inhibited human acetylcholinesterase (hAChE).
    Valiveti AK; Bhalerao UM; Acharya J; Karade HN; Gundapu R; Halve AK; Kaushik MP
    Chem Biol Interact; 2015 Jul; 237():125-32. PubMed ID: 26070418
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 5.