These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

374 related articles for article (PubMed ID: 8848011)

  • 1. beta-Carboline gamma-aminobutyric acidA receptor inverse agonists modulate gamma-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site.
    Stevenson A; Wingrove PB; Whiting PJ; Wafford KA
    Mol Pharmacol; 1995 Dec; 48(6):965-9. PubMed ID: 8848011
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Interaction of beta-carboline inverse agonists for the benzodiazepine site with another site on GABAA receptors.
    Im HK; Im WB; Carter DB; McKinley DD
    Br J Pharmacol; 1995 Mar; 114(5):1040-4. PubMed ID: 7780638
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Pharmacology of the human gamma-aminobutyric acidA receptor alpha 4 subunit expressed in Xenopus laevis oocytes.
    Whittemore ER; Yang W; Drewe JA; Woodward RM
    Mol Pharmacol; 1996 Nov; 50(5):1364-75. PubMed ID: 8913369
    [TBL] [Abstract][Full Text] [Related]  

  • 4. The modulatory action of loreclezole at the gamma-aminobutyric acid type A receptor is determined by a single amino acid in the beta 2 and beta 3 subunit.
    Wingrove PB; Wafford KA; Bain C; Whiting PJ
    Proc Natl Acad Sci U S A; 1994 May; 91(10):4569-73. PubMed ID: 8183949
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Actions of two GABAA receptor benzodiazepine-site ligands that are mediated via non-γ2-dependent modulation.
    Leppä E; Linden AM; Rabe H; Vekovischeva OY; Wulff P; Lüddens H; Wisden W; Korpi ER
    Eur J Pharmacol; 2011 Sep; 666(1-3):111-21. PubMed ID: 21616065
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Pharmacological modulation of the diazepam-insensitive recombinant gamma-aminobutyric acidA receptors alpha 4 beta 2 gamma 2 and alpha 6 beta 2 gamma 2.
    Knoflach F; Benke D; Wang Y; Scheurer L; Lüddens H; Hamilton BJ; Carter DB; Mohler H; Benson JA
    Mol Pharmacol; 1996 Nov; 50(5):1253-61. PubMed ID: 8913357
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Direct activation of GABAA receptors by loreclezole, an anticonvulsant drug with selectivity for the beta-subunit.
    Sanna E; Murgia A; Casula A; Usala M; Maciocco E; Tuligi G; Biggio G
    Neuropharmacology; 1996; 35(12):1753-60. PubMed ID: 9076754
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Cerebellar gamma-aminobutyric acid type A receptors: pharmacological subtypes revealed by mutant mouse lines.
    Mäkelä R; Uusi-Oukari M; Homanics GE; Quinlan JJ; Firestone LL; Wisden W; Korpi ER
    Mol Pharmacol; 1997 Sep; 52(3):380-8. PubMed ID: 9281599
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Functional characterization of human gamma-aminobutyric acidA receptors containing the alpha 4 subunit.
    Wafford KA; Thompson SA; Thomas D; Sikela J; Wilcox AS; Whiting PJ
    Mol Pharmacol; 1996 Sep; 50(3):670-8. PubMed ID: 8794909
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Functional GABAA receptor heterogeneity of acutely dissociated hippocampal CA1 pyramidal cells.
    Tietz EI; Kapur J; Macdonald RL
    J Neurophysiol; 1999 Apr; 81(4):1575-86. PubMed ID: 10200193
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Key amino acids in the gamma subunit of the gamma-aminobutyric acidA receptor that determine ligand binding and modulation at the benzodiazepine site.
    Wingrove PB; Thompson SA; Wafford KA; Whiting PJ
    Mol Pharmacol; 1997 Nov; 52(5):874-81. PubMed ID: 9351978
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Differences in the negative allosteric modulation of gamma-aminobutyric acid receptors elicited by 4'-chlorodiazepam and by a beta-carboline-3-carboxylate ester: a study with natural and reconstituted receptors.
    Puia G; Santi MR; Vicini S; Pritchett DB; Seeburg PH; Costa E
    Proc Natl Acad Sci U S A; 1989 Sep; 86(18):7275-9. PubMed ID: 2476816
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Loreclezole modulates [35S]t-butylbicyclophosphorothionate and [3H]flunitrazepam binding via a distinct site on the GABAA receptor complex.
    Xue BG; Friend JM; Gee KW
    Eur J Pharmacol; 1996 Apr; 300(1-2):125-30. PubMed ID: 8741177
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Functional comparison of the role of gamma subunits in recombinant human gamma-aminobutyric acidA/benzodiazepine receptors.
    Wafford KA; Bain CJ; Whiting PJ; Kemp JA
    Mol Pharmacol; 1993 Aug; 44(2):437-42. PubMed ID: 8102787
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Dual mode of stimulation by the beta-carboline ZK 91085 of recombinant GABA(A) receptor currents: molecular determinants affecting its action.
    Thomet U; Baur R; Scholze P; Sieghart W; Sigel E
    Br J Pharmacol; 1999 Jul; 127(5):1231-9. PubMed ID: 10455270
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Behavioral evidence for the role of noradrenaline in the putative anxiogenic actions of the inverse benzodiazepine receptor agonist methyl-4-ethyl-6,7-dimethoxy-beta-carboline-3-carboxylate.
    Yang XM; Luo ZP; Zhou JH
    J Pharmacol Exp Ther; 1989 Jul; 250(1):358-63. PubMed ID: 2545863
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Allosteric modulators affect the efficacy of partial agonists for recombinant GABA(A) receptors.
    Maksay G; Thompson SA; Wafford KA
    Br J Pharmacol; 2000 Apr; 129(8):1794-800. PubMed ID: 10780988
    [TBL] [Abstract][Full Text] [Related]  

  • 18. A novel allosteric modulatory site on the GABAA receptor beta subunit.
    Wafford KA; Bain CJ; Quirk K; McKernan RM; Wingrove PB; Whiting PJ; Kemp JA
    Neuron; 1994 Apr; 12(4):775-82. PubMed ID: 8161449
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Benzodiazepine agonist and inverse agonist actions on GABAA receptor-operated chloride channels. II. Chronic effects of ethanol.
    Buck KJ; Harris RA
    J Pharmacol Exp Ther; 1990 May; 253(2):713-9. PubMed ID: 2160008
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Benzodiazepine site inverse agonists can selectively inhibit subtypes of the GABAA receptor.
    White G; Gurley D
    Neuroreport; 1995 Jun; 6(9):1313-6. PubMed ID: 7669993
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 19.