116 related articles for article (PubMed ID: 8915103)
1. Binding of clozapine metabolites and analogues to the histamine H3 receptor in rat brain cortex.
Alves-Rodrigues A; Leurs R; Willems E; Timmerman H
Arch Pharm (Weinheim); 1996; 329(8-9):413-6. PubMed ID: 8915103
[TBL] [Abstract][Full Text] [Related]
2. The moderate affinity of clozapine at H3 receptors is not shared by its two major metabolites and by structurally related and unrelated atypical neuroleptics.
Schlicker E; Marr I
Naunyn Schmiedebergs Arch Pharmacol; 1996 Feb; 353(3):290-4. PubMed ID: 8692283
[TBL] [Abstract][Full Text] [Related]
3. Characterization of the binding of the first selective radiolabelled histamine H3-receptor antagonist, [125I]-iodophenpropit, to rat brain.
Jansen FP; Wu TS; Voss HP; Steinbusch HW; Vollinga RC; Rademaker B; Bast A; Timmerman H
Br J Pharmacol; 1994 Oct; 113(2):355-62. PubMed ID: 7834183
[TBL] [Abstract][Full Text] [Related]
4. Intermediate affinity and potency of clozapine and low affinity of other neuroleptics and of antidepressants at H3 receptors.
Kathmann M; Schlicker E; Göthert M
Psychopharmacology (Berl); 1994 Dec; 116(4):464-8. PubMed ID: 7701050
[TBL] [Abstract][Full Text] [Related]
5. Interaction of clozapine with the histamine H3 receptor in rat brain.
Rodrigues AA; Jansen FP; Leurs R; Timmerman H; Prell GD
Br J Pharmacol; 1995 Apr; 114(8):1523-4. PubMed ID: 7541279
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and in vitro pharmacology of a series of new chiral histamine H3-receptor ligands: 2-(R and S)-Amino-3-(1H-imidazol-4(5)-yl)propyl ether derivatives.
Kovalainen JT; Christiaans JA; Kotisaari S; Laitinen JT; Männistö PT; Tuomisto L; Gynther J
J Med Chem; 1999 Apr; 42(7):1193-202. PubMed ID: 10197963
[TBL] [Abstract][Full Text] [Related]
7. Evaluation of the receptor selectivity of the H3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5-HT3 receptor revealed.
Leurs R; Tulp MT; Menge WM; Adolfs MJ; Zuiderveld OP; Timmerman H
Br J Pharmacol; 1995 Oct; 116(4):2315-21. PubMed ID: 8564266
[TBL] [Abstract][Full Text] [Related]
8. The first radiolabeled histamine H3 receptor antagonist, [125I]iodophenpropit: saturable and reversible binding to rat cortex membranes.
Jansen FP; Rademaker B; Bast A; Timmerman H
Eur J Pharmacol; 1992 Jul; 217(2-3):203-5. PubMed ID: 1330590
[TBL] [Abstract][Full Text] [Related]
9. Discovery of histamine H3 receptor antagonistic property of simple imidazole-free derivatives: Preliminary pharmacological investigation.
Barocelli E; Ballabeni V; Manenti V; Flammini L; Bertoni S; Morini G; Comini M; Impicciatore M
Pharmacol Res; 2006 Mar; 53(3):226-32. PubMed ID: 16364652
[TBL] [Abstract][Full Text] [Related]
10. Chloro-substituted, sterically hindered 5,11-dicarbo analogues of clozapine as potential chiral antipsychotic agents.
Davis DA; de Paulis T; Janowsky A; Smith HE
J Med Chem; 1990 Feb; 33(2):809-14. PubMed ID: 1967652
[TBL] [Abstract][Full Text] [Related]
11. H3-receptor antagonists: synthesis and structure-activity relationships of para- and meta-substituted 4(5)-phenyl-2-[[2-[4(5)-imidazolyl]ethyl]thio]imidazoles.
Mor M; Bordi F; Silva C; Rivara S; Crivori P; Plazzi PV; Ballabeni V; Caretta A; Barocelli E; Impicciatore M; Carrupt PA; Testa B
J Med Chem; 1997 Aug; 40(16):2571-8. PubMed ID: 9258364
[TBL] [Abstract][Full Text] [Related]
12. Non-Imidazole Histamine H3 Ligands. Part VI. Synthesis and Preliminary Pharmacological Investigation of Thiazole-Type Histamine H3-Receptor Antagonists with Lacking a Nitrogen Nucleus in the Side Chain.
Guryn R; Staszewski M; Kopczacki P; Walczyski K
Med Chem; 2016; 13(1):65-76. PubMed ID: 27220560
[TBL] [Abstract][Full Text] [Related]
13. Novel histamine H3 receptor antagonists: synthesis and evaluation of formamidine and S-methylisothiourea derivatives.
Goto T; Sakashita H; Murakami K; Sugiura M; Kondo T; Fukaya C
Chem Pharm Bull (Tokyo); 1997 Feb; 45(2):305-11. PubMed ID: 9118445
[TBL] [Abstract][Full Text] [Related]
14. Pharmacological characterisation of the histamine H3 receptor in the rat hippocampus.
Alves-Rodrigues A; Timmerman H; Willems E; Lemstra S; Zuiderveld OP; Leurs R
Brain Res; 1998 Mar; 788(1-2):179-86. PubMed ID: 9555002
[TBL] [Abstract][Full Text] [Related]
15. [3H]-thioperamide as a radioligand for the histamine H3 receptor in rat cerebral cortex.
Alves-Rodrigues A; Leurs R; Wu TS; Prell GD; Foged C; Timmerman H
Br J Pharmacol; 1996 Aug; 118(8):2045-52. PubMed ID: 8864541
[TBL] [Abstract][Full Text] [Related]
16. Potencies of antagonists chemically related to iodoproxyfan at histamine H3 receptors in mouse brain cortex and guinea-pig ileum: evidence for H3 receptor heterogeneity?
Schlicker E; Kathmann M; Bitschnau H; Marr I; Reidemeister S; Stark H; Schunack W
Naunyn Schmiedebergs Arch Pharmacol; 1996 Apr; 353(5):482-8. PubMed ID: 8740140
[TBL] [Abstract][Full Text] [Related]
17. Novel histamine H3 receptor antagonists: affinities in an H3 receptor binding assay and potencies in two functional H3 receptor models.
Schlicker E; Kathmann M; Reidemeister S; Stark H; Schunack W
Br J Pharmacol; 1994 Aug; 112(4):1043-8. PubMed ID: 7952862
[TBL] [Abstract][Full Text] [Related]
18. Development of FUB 181, a selective histamine H3-receptor antagonist of high oral in vivo potency with 4-(omega-(arylalkyloxy)alkyl)-1H-imidazole structure.
Stark H; Hüls A; Ligneau X; Purand K; Pertz H; Arrang JM; Schwartz JC; Schunack W
Arch Pharm (Weinheim); 1998 Jun; 331(6):211-8. PubMed ID: 9713254
[TBL] [Abstract][Full Text] [Related]
19. Development of trans-2-[1H-imidazol-4-yl] cyclopropane derivatives as new high-affinity histamine H3 receptor ligands.
Tedford CE; Phillips JG; Gregory R; Pawlowski GP; Fadnis L; Khan MA; Ali SM; Handley MK; Yates SL
J Pharmacol Exp Ther; 1999 May; 289(2):1160-8. PubMed ID: 10215700
[TBL] [Abstract][Full Text] [Related]
20. Characterization of histamine H3 receptors in mouse brain using the H3 antagonist [125I]iodophenpropit.
Jansen FP; Mochizuki T; Maeyama K; Leurs R; Timmerman H
Naunyn Schmiedebergs Arch Pharmacol; 2000 Jul; 362(1):60-7. PubMed ID: 10935534
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
