96 related articles for article (PubMed ID: 8960547)
1. Anti-inflammatory 17beta-thioalkyl-16alpha,17alpha-ketal and -acetal androstanes: a new class of airway selective steroids for the treatment of asthma.
Ashton MJ; Lawrence C; Karlsson JA; Stuttle KA; Newton CG; Vacher BY; Webber S; Withnall MJ
J Med Chem; 1996 Dec; 39(25):4888-96. PubMed ID: 8960547
[TBL] [Abstract][Full Text] [Related]
2. In vitro anti-inflammatory activities of new steroidal antedrugs: [16alpha,17alpha-d] Isoxazoline and [16alpha,17alpha-d]-3'-hydroxy-iminoformyl isoxazoline derivatives of prednisolone and 9alpha-fluoroprednisolone.
Park KK; Ko DH; You Z; Khan MO; Lee HJ
Steroids; 2006 Mar; 71(3):183-8. PubMed ID: 16309722
[TBL] [Abstract][Full Text] [Related]
3. Novel glucocorticoid antedrugs possessing a 17beta-(gamma-lactone) ring.
Procopiou PA; Biggadike K; English AF; Farrell RM; Hagger GN; Hancock AP; Haase MV; Irving WR; Sareen M; Snowden MA; Solanke YE; Tralau-Stewart CJ; Walton SE; Wood JA
J Med Chem; 2001 Feb; 44(4):602-12. PubMed ID: 11170650
[TBL] [Abstract][Full Text] [Related]
4. Synthesis and pharmacological evaluations of new steroidal anti-inflammatory antedrugs: 9alpha-Fluoro-11beta,17alpha,21-trihydroxy-3,20-dioxo-pregna-1,4-diene-16alpha-carboxylate (FP16CM) and its derivatives.
Park KK; Ko DH; You Z; Heiman AS; Lee HJ
Steroids; 2006 Jan; 71(1):83-9. PubMed ID: 16280144
[TBL] [Abstract][Full Text] [Related]
5. Discovery of betamethasone 17alpha-carbamates as dissociated glucocorticoid receptor modulators in the rat.
Ali A; Balkovec JM; Greenlee M; Hammond ML; Rouen G; Taylor G; Einstein M; Ge L; Harris G; Kelly TM; Mazur P; Pandit S; Santoro J; Sitlani A; Wang C; Williamson J; Forrest MJ; Carballo-Jane E; Luell S; Lowitz K; Visco D
Bioorg Med Chem; 2008 Aug; 16(16):7535-42. PubMed ID: 18691892
[TBL] [Abstract][Full Text] [Related]
6. New steroidal anti-inflammatory antedrugs: methyl 21-desoxy-21-chloro-11beta,17alpha-dihydroxy-3,20-dioxo-1, 4-pregnadiene-16alpha-carboxylate, methyl 21-desoxy-21-chloro-11beta-hydroxy-3,20-dioxo-1, 4-pregnadiene-16alpha-carboxylate, and their 9alpha-fluoro derivatives*.
Ko D; Heiman AS; Chen M; Lee HJ
Steroids; 2000 Apr; 65(4):210-8. PubMed ID: 10713309
[TBL] [Abstract][Full Text] [Related]
7. 7alpha-Iodo and 7alpha-fluoro steroids as androgen receptor-mediated imaging agents.
Labaree DC; Hoyte RM; Nazareth LV; Weigel NL; Hochberg RB
J Med Chem; 1999 Jun; 42(11):2021-34. PubMed ID: 10354410
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and biological properties of novel glucocorticoid androstene C-17 furoate esters.
Sandham DA; Barker L; Beattie D; Beer D; Bidlake L; Bentley D; Butler KD; Craig S; Farr D; Ffoulkes-Jones C; Fozard JR; Haberthuer S; Howes C; Hynx D; Jeffers S; Keller TH; Kirkham PA; Maas JC; Mazzoni L; Nicholls A; Pilgrim GE; Schaebulin E; Spooner GM; Stringer R; Tranter P; Turner KL; Tweed MF; Walker C; Watson SJ; Cuenoud BM
Bioorg Med Chem; 2004 Oct; 12(19):5213-24. PubMed ID: 15351404
[TBL] [Abstract][Full Text] [Related]
9. Nonsteroidal selective glucocorticoid modulators: the effect of C-10 substitution on receptor selectivity and functional potency of 5-allyl-2,5-dihydro-2,2,4-trimethyl-1H-[1]benzopyrano[3,4-f]quinolines.
Kym PR; Kort ME; Coghlan MJ; Moore JL; Tang R; Ratajczyk JD; Larson DP; Elmore SW; Pratt JK; Stashko MA; Falls HD; Lin CW; Nakane M; Miller L; Tyree CM; Miner JN; Jacobson PB; Wilcox DM; Nguyen P; Lane BC
J Med Chem; 2003 Mar; 46(6):1016-30. PubMed ID: 12620078
[TBL] [Abstract][Full Text] [Related]
10. [Protective effects of ketamine on allergen-induced airway inflammatory injure and high airway reactivity in asthma: experiment with rats].
Zhu MM; Qian YN; Zhu W; Xu YM; Rong HB; Ding ZN; Fu CZ
Zhonghua Yi Xue Za Zhi; 2007 May; 87(19):1308-13. PubMed ID: 17727773
[TBL] [Abstract][Full Text] [Related]
11. NTP toxicology and carcinogenesis studies of 3,3',4,4',5-pentachlorobiphenyl (PCB 126) (CAS No. 57465-28-8) in female Harlan Sprague-Dawley rats (Gavage Studies).
National Toxicology Program
Natl Toxicol Program Tech Rep Ser; 2006 Jan; (520):4-246. PubMed ID: 16628245
[TBL] [Abstract][Full Text] [Related]
12. Novel ketal ligands for the glucocorticoid receptor: in vitro and in vivo activity.
Smith CJ; Ali A; Balkovec JM; Graham DW; Hammond ML; Patel GF; Rouen GP; Smith SK; Tata JR; Einstein M; Ge L; Harris GS; Kelly TM; Mazur P; Thompson CM; Wang CF; Williamson JM; Miller DK; Pandit S; Santoro JC; Sitlani A; Yamin TT; O'Neill EA; Zaller DM; Carballo-Jane E; Forrest MJ; Luell S
Bioorg Med Chem Lett; 2005 Jun; 15(11):2926-31. PubMed ID: 15911283
[TBL] [Abstract][Full Text] [Related]
13. Glucocorticoids: mechanisms of action and anti-inflammatory potential in asthma.
van der Velden VH
Mediators Inflamm; 1998; 7(4):229-37. PubMed ID: 9792333
[TBL] [Abstract][Full Text] [Related]
14. Enhanced expression of urocortin in lung tissues of rats with allergic asthma.
Wu Y; Zhou H; Xu Y; Li S
Biochem Biophys Res Commun; 2006 Mar; 341(2):532-40. PubMed ID: 16427607
[TBL] [Abstract][Full Text] [Related]
15. Macrolactonolides: a novel class of anti-inflammatory compounds.
Tomašković L; Komac M; Makaruha Stegić O; Munić V; Ralić J; Stanić B; Banjanac M; Marković S; Hrvačić B; Čipčić Paljetak H; Padovan J; Glojnarić I; Eraković Haber V; Mesić M; Merćep M
Bioorg Med Chem; 2013 Jan; 21(1):321-32. PubMed ID: 23199485
[TBL] [Abstract][Full Text] [Related]
16. Potency and specificity of the pharmacological action of a new, antiasthmatic, topically administered soft steroid, etiprednol dicloacetate (BNP-166).
Kurucz I; Tóth S; Németh K; Török K; Csillik-Perczel V; Pataki A; Salamon C; Nagy Z; Székely JI; Horváth K; Bodor N
J Pharmacol Exp Ther; 2003 Oct; 307(1):83-92. PubMed ID: 12893841
[TBL] [Abstract][Full Text] [Related]
17. Thymic involution in the suspended rat model for weightlessness: decreased glucocorticoid receptor concentration.
Steffen JM; Musacchia XJ
Physiologist; 1984; 27(6 Suppl):S39-40. PubMed ID: 11539011
[TBL] [Abstract][Full Text] [Related]
18. The glucocorticoid receptor is essential for induction of cytochrome P-4502B by steroids but not for drug or steroid induction of CYP3A or P-450 reductase in mouse liver.
Schuetz EG; Schmid W; Schutz G; Brimer C; Yasuda K; Kamataki T; Bornheim L; Myles K; Cole TJ
Drug Metab Dispos; 2000 Mar; 28(3):268-78. PubMed ID: 10681370
[TBL] [Abstract][Full Text] [Related]
19. Selective prostacyclin receptor agonism augments glucocorticoid-induced gene expression in human bronchial epithelial cells.
Wilson SM; Shen P; Rider CF; Traves SL; Proud D; Newton R; Giembycz MA
J Immunol; 2009 Nov; 183(10):6788-99. PubMed ID: 19880449
[TBL] [Abstract][Full Text] [Related]
20. Steroidal C-21 heteroaryl thioethers (Part 2): discovery of orally bioavailable selective glucocorticoid receptor modulators (dissociated steroids).
Biju P; McCormick K; Aslanian R; Berlin M; Solomon D; Wang H; Lee YJ; Bitar R; Prelusky D; McLeod R; Jia Y; Fernandez X; Eckel S; House A; Lieber G; Jimenez J; Kelly G; Chapman R; Phillips J; Anthes J
Bioorg Med Chem Lett; 2012 Jan; 22(2):1086-90. PubMed ID: 22197391
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
