158 related articles for article (PubMed ID: 9240344)
1. Synthesis and nicotinic acetylcholine receptor binding properties of exo-2-(2'-fluoro-5'-pyridinyl)-7-azabicyclo-[2.2.1]heptane: a new positron emission tomography ligand for nicotinic receptors.
Liang F; Navarro HA; Abraham P; Kotian P; Ding YS; Fowler J; Volkow N; Kuhar MJ; Carroll FI
J Med Chem; 1997 Jul; 40(15):2293-5. PubMed ID: 9240344
[No Abstract] [Full Text] [Related]
2. Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 2-exo-2-(2'-substituted-3'-phenyl-5'-pyridinyl)-7-azabicyclo[2.2.1]heptanes. Novel nicotinic antagonist.
Carroll FI; Lee JR; Navarro HA; Brieaddy LE; Abraham P; Damaj MI; Martin BR
J Med Chem; 2001 Nov; 44(24):4039-41. PubMed ID: 11708907
[TBL] [Abstract][Full Text] [Related]
3. Derivatives of (-)-7-methyl-2-(5-(pyridinyl)pyridin-3-yl)-7-azabicyclo[2.2.1]heptane are potential ligands for positron emission tomography imaging of extrathalamic nicotinic acetylcholine receptors.
Gao Y; Horti AG; Kuwabara H; Ravert HT; Hilton J; Holt DP; Kumar A; Alexander M; Endres CJ; Wong DF; Dannals RF
J Med Chem; 2007 Aug; 50(16):3814-24. PubMed ID: 17629263
[TBL] [Abstract][Full Text] [Related]
4. Preparation of a bromine-76 labelled analogue of epibatidine: a potent ligand for nicotinic acetylcholine receptor studies.
Kassiou M; Loc'h C; Dolle F; Musachio JL; Dolci L; Crouzel C; Dannals RF; Mazière B
Appl Radiat Isot; 2002 Nov; 57(5):713-7. PubMed ID: 12433046
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and binding studies of epibatidine analogues as ligands for the nicotinic acetylcholine receptors.
Mu L; Drandarov K; Bisson WH; Schibig A; Wirz C; Schubiger PA; Westera G
Eur J Med Chem; 2006 May; 41(5):640-50. PubMed ID: 16545497
[TBL] [Abstract][Full Text] [Related]
6. Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 2'-fluoro-3'-(substituted phenyl)deschloroepibatidine analogues. Novel nicotinic antagonist.
Carroll FI; Ware R; Brieaddy LE; Navarro HA; Damaj MI; Martin BR
J Med Chem; 2004 Aug; 47(18):4588-94. PubMed ID: 15317468
[TBL] [Abstract][Full Text] [Related]
7. New synthesis and evaluation of enantiomers of 7-methyl-2-exo-(3'-iodo-5'-pyridinyl)-7-azabicyclo[2.2.1]heptane as stereoselective ligands for PET imaging of nicotinic acetylcholine receptors.
Gao Y; Horti AG; Kuwabara H; Ravert HT; Holt DP; Kumar A; Alexander M; Wong DF; Dannals RF
Bioorg Med Chem Lett; 2008 Dec; 18(23):6168-70. PubMed ID: 18930397
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and pharmacological characterization of exo-2-(2'-chloro-5-pyridinyl)-7-(endo and exo)-aminobicyclo[2.2.1]heptanes as novel epibatidine analogues.
Carroll FI; Brieaddy LE; Navarro HA; Damaj MI; Martin BR
J Med Chem; 2005 Nov; 48(23):7491-5. PubMed ID: 16279810
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and nicotinic acetylcholine receptor binding properties of bridged and fused ring analogues of epibatidine.
Carroll FI; Robinson TP; Brieaddy LE; Atkinson RN; Mascarella SW; Damaj MI; Martin BR; Navarro HA
J Med Chem; 2007 Dec; 50(25):6383-91. PubMed ID: 17994682
[TBL] [Abstract][Full Text] [Related]
10. Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 3'-substituted deschloroepibatidine analogues. Novel nicotinic antagonists.
Carroll FI; Ma W; Yokota Y; Lee JR; Brieaddy LE; Navarro HA; Damaj MI; Martin BR
J Med Chem; 2005 Feb; 48(4):1221-8. PubMed ID: 15715488
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and evaluation of N-[11C]methylated analogues of epibatidine as tracers for positron emission tomographic studies of nicotinic acetylcholine receptors.
Horti AG; Scheffel U; Kimes AS; Musachio JL; Ravert HT; Mathews WB; Zhan Y; Finley PA; London ED; Dannals RF
J Med Chem; 1998 Oct; 41(22):4199-206. PubMed ID: 9784094
[TBL] [Abstract][Full Text] [Related]
12. Synthesis, nicotinic acetylcholine receptor binding, and pharmacological properties of 3'-(substituted phenyl)deschloroepibatidine analogs.
Ivy Carroll F; Yokota Y; Ma W; Lee JR; Brieaddy LE; Burgess JP; Navarro HA; Damaj MI; Martin BR
Bioorg Med Chem; 2008 Jan; 16(2):746-54. PubMed ID: 17964169
[TBL] [Abstract][Full Text] [Related]
13. Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 2-exo-2-(2',3'-disubstituted 5'-pyridinyl)-7-azabicyclo[2.2.1]heptanes: epibatidine analogues.
Carroll FI; Lee JR; Navarro HA; Ma W; Brieaddy LE; Abraham P; Damaj MI; Martin BR
J Med Chem; 2002 Oct; 45(21):4755-61. PubMed ID: 12361403
[TBL] [Abstract][Full Text] [Related]
14. Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 2-exo-2-(2'-substituted 5'-pyridinyl)-7-azabicyclo[2.2.1]heptanes. Epibatidine analogues.
Carroll FI; Liang F; Navarro HA; Brieaddy LE; Abraham P; Damaj MI; Martin BR
J Med Chem; 2001 Jun; 44(13):2229-37. PubMed ID: 11405659
[TBL] [Abstract][Full Text] [Related]
15. Epibatidine analogues as selective ligands for the alpha(x)beta2-containing subtypes of nicotinic acetylcholine receptors.
Huang Y; Zhu Z; Xiao Y; Laruelle M
Bioorg Med Chem Lett; 2005 Oct; 15(19):4385-8. PubMed ID: 16039849
[TBL] [Abstract][Full Text] [Related]
16. Functionalization of the alicyclic skeleton of epibatidine: synthesis and nicotinic acetylcholine receptor binding affinities of epibatidine analogues.
Wei ZL; Xiao Y; George C; Kellar KJ; Kozikowski AP
Org Biomol Chem; 2003 Nov; 1(22):3878-81. PubMed ID: 14664377
[TBL] [Abstract][Full Text] [Related]
17. Discovery of (-)-7-methyl-2-exo-[3'-(6-[18F]fluoropyridin-2-yl)-5'-pyridinyl]-7-azabicyclo[2.2.1]heptane, a radiolabeled antagonist for cerebral nicotinic acetylcholine receptor (alpha4beta2-nAChR) with optimal positron emission tomography imaging properties.
Gao Y; Kuwabara H; Spivak CE; Xiao Y; Kellar K; Ravert HT; Kumar A; Alexander M; Hilton J; Wong DF; Dannals RF; Horti AG
J Med Chem; 2008 Aug; 51(15):4751-64. PubMed ID: 18605717
[TBL] [Abstract][Full Text] [Related]
18. Synthesis of a fluorine-18 labeled derivative of epibatidine for in vivo nicotinic acetylcholine receptor PET imaging.
Dolci L; Dolle F; Valette H; Vaufrey F; Fuseau C; Bottlaender M; Crouzel C
Bioorg Med Chem; 1999 Mar; 7(3):467-79. PubMed ID: 10220033
[TBL] [Abstract][Full Text] [Related]
19. In vivo labeling of nicotinic acetylcholine receptors in brain with [3H]epibatidine.
London ED; Scheffel U; Kimes AS; Kellar KJ
Eur J Pharmacol; 1995 May; 278(1):R1-2. PubMed ID: 7664806
[TBL] [Abstract][Full Text] [Related]
20. Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 2'-fluoro-3'-(substituted pyridinyl)-7-deschloroepibatidine analogues.
Ondachi PW; Castro AH; Bartkowiak JM; Luetje CW; Damaj MI; Mascarella SW; Navarro HA; Carroll FI
J Med Chem; 2014 Feb; 57(3):836-48. PubMed ID: 24428686
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
