138 related articles for article (PubMed ID: 9372593)
61. High affinity central benzodiazepine receptor ligands: synthesis and biological evaluation of a series of phenyltriazolobenzotriazindione derivatives.
Primofiore G; Da Settimo F; Taliani S; Salerno S; Novellino E; Greco G; Cosimelli B; Besnard F; Costa B; Montali M; Martini C
J Med Chem; 2005 Apr; 48(8):2936-43. PubMed ID: 15828832
[TBL] [Abstract][Full Text] [Related]
62. Asymmetric synthesis of beta-amino-gamma-substituted-gamma-butyrolactones: double diastereoselective conjugate addition of homochiral lithium amides to homochiral alpha,beta-unsaturated esters.
Cailleau T; Cooke JW; Davies SG; Ling KB; Naylor A; Nicholson RL; Price PD; Roberts PM; Russell AJ; Smith AD; Thomson JE
Org Biomol Chem; 2007 Dec; 5(24):3922-31. PubMed ID: 18043795
[TBL] [Abstract][Full Text] [Related]
63. A novel class of adenosine A3 receptor ligands. 2. Structure affinity profile of a series of isoquinoline and quinazoline compounds.
van Muijlwijk-Koezen JE; Timmerman H; Link R; van der Goot H; Ijzerman AP
J Med Chem; 1998 Oct; 41(21):3994-4000. PubMed ID: 9767637
[TBL] [Abstract][Full Text] [Related]
64. Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423) at wild type and recombinant GABAA receptors.
Cox ED; Diaz-Arauzo H; Huang Q; Reddy MS; Ma C; Harris B; McKernan R; Skolnick P; Cook JM
J Med Chem; 1998 Jul; 41(14):2537-52. PubMed ID: 9651158
[TBL] [Abstract][Full Text] [Related]
65. Doubly diastereoselective conjugate addition of homochiral lithium amides to homochiral alpha,beta-unsaturated esters containing cis- and trans-dioxolane units.
Davies SG; Durbin MJ; Goddard EC; Kelly PM; Kurosawa W; Lee JA; Nicholson RL; Price PD; Roberts PM; Russell AJ; Scott PM; Smith AD
Org Biomol Chem; 2009 Feb; 7(4):761-76. PubMed ID: 19194592
[TBL] [Abstract][Full Text] [Related]
66. Comparative quantitative structure-activity relationship studies (QSAR) on non-benzodiazepine compounds binding to benzodiazepine receptor (BzR).
Hadjipavlou-Litina D; Garg R; Hansch C
Chem Rev; 2004 Sep; 104(9):3751-94. PubMed ID: 15352779
[No Abstract] [Full Text] [Related]
67. Synthesis and serotonin receptor affinities of a series of trans-2-(indol-3-yl)cyclopropylamine derivatives.
Vangveravong S; Kanthasamy A; Lucaites VL; Nelson DL; Nichols DE
J Med Chem; 1998 Dec; 41(25):4995-5001. PubMed ID: 9836617
[TBL] [Abstract][Full Text] [Related]
68. 6,3'-dibromoflavone and 6-nitro-3'-bromoflavone: new additions to the 6,3'-disubstituted flavone family of high-affinity ligands of the brain benzodiazepine binding site with agonistic properties.
Viola H; Marder M; Wasowski C; Giorgi O; Paladini AC; Medina JH
Biochem Biophys Res Commun; 2000 Jul; 273(2):694-8. PubMed ID: 10873666
[TBL] [Abstract][Full Text] [Related]
69. Study on affinity profile toward native human and bovine adenosine receptors of a series of 1,8-naphthyridine derivatives.
Ferrarini PL; Betti L; Cavallini T; Giannaccini G; Lucacchini A; Manera C; Martinelli A; Ortore G; Saccomanni G; Tuccinardi T
J Med Chem; 2004 Jun; 47(12):3019-31. PubMed ID: 15163184
[TBL] [Abstract][Full Text] [Related]
70. Preparation, properties, reactions, and adenosine receptor affinities of sulfophenylxanthine nitrophenyl esters: toward the development of sulfonic acid prodrugs with peroral bioavailability.
Yan L; Müller CE
J Med Chem; 2004 Feb; 47(4):1031-43. PubMed ID: 14761205
[TBL] [Abstract][Full Text] [Related]
71. Substituted benzylaminoalkylindoles with preference for the sigma2 binding site.
Mamolo MG; Zampieri D; Zanette C; Florio C; Collina S; Urbano M; Azzolina O; Vio L
Eur J Med Chem; 2008 Oct; 43(10):2073-81. PubMed ID: 18069094
[TBL] [Abstract][Full Text] [Related]
72. [Reactions of 4,5-dihydro-4-oxo-1H-pyrido(3,2-b)indol-2-carboxylic acid ester].
Görlitzer K; Kramer C
Pharmazie; 2000 Apr; 55(4):273-81. PubMed ID: 10798240
[TBL] [Abstract][Full Text] [Related]
73. Isoindol-1-one analogues of 4-(2'-methoxyphenyl)-1-[2'-[N-(2"-pyridyl)-p-iodobenzamido]ethyl]pipera zine (p-MPPI) as 5-HT1A receptor ligands.
Zhuang ZP; Kung MP; Mu M; Kung HF
J Med Chem; 1998 Jan; 41(2):157-66. PubMed ID: 9457239
[TBL] [Abstract][Full Text] [Related]
74. Effects of propofol and pentobarbital on ligand binding to GABAA receptors suggest a similar mechanism of action.
Davies M; Thuynsma RP; Dunn SM
Can J Physiol Pharmacol; 1998 Jan; 76(1):46-52. PubMed ID: 9564548
[TBL] [Abstract][Full Text] [Related]
75. The importance of the amide bond nearest the thiol group in enzymatic reactions of coenzyme A.
Xun J; Huang H; Vogel KW; Drueckhammer DG
Bioorg Chem; 2005 Apr; 33(2):90-107. PubMed ID: 15788165
[TBL] [Abstract][Full Text] [Related]
76. p-tert-Butyl thiacalix[4]arenes functionalized at the lower rim by amide, hydroxyl and ester groups as anion receptors.
Stoikov II; Yantemirova AA; Nosov RV; Rizvanov IKh; Julmetov AR; Klochkov VV; Antipin IS; Konovalov AI; Zharov I
Org Biomol Chem; 2011 May; 9(9):3225-34. PubMed ID: 21423989
[TBL] [Abstract][Full Text] [Related]
77. Analysis of structure-activity relationships with the N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea template for vanilloid receptor 1 antagonism.
Lee J; Kim SY; Lee J; Kang M; Kil MJ; Choi HK; Jin MK; Wang Y; Toth A; Pearce LV; Lundberg DJ; Tran R; Blumberg PM
Bioorg Med Chem; 2004 Jul; 12(13):3411-20. PubMed ID: 15186827
[TBL] [Abstract][Full Text] [Related]
78. Potent 4-aryl- or 4-arylalkyl-substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.
Frølund B; Jensen LS; Guandalini L; Canillo C; Vestergaard HT; Kristiansen U; Nielsen B; Stensbøl TB; Madsen C; Krogsgaard-Larsen P; Liljefors T
J Med Chem; 2005 Jan; 48(2):427-39. PubMed ID: 15658856
[TBL] [Abstract][Full Text] [Related]
79. Design, synthesis, and structure-affinity relationship studies in NK1 receptor ligands based on azole-fused quinolinecarboxamide moieties.
Cappelli A; Giuliani G; Anzini M; Riitano D; Giorgi G; Vomero S
Bioorg Med Chem; 2008 Jul; 16(14):6850-9. PubMed ID: 18554914
[TBL] [Abstract][Full Text] [Related]
80. Contribution of specific binding to the central benzodiazepine site to the brain concentrations of two novel benzodiazepine site ligands.
Pike A; Cook SM; Watt AP; Scott-Stevens P; Rosahl TW; McKernan RM; Pym LJ; Guiblin A; Moyes C; Sohal B; Atack JR
Biopharm Drug Dispos; 2007 Sep; 28(6):275-82. PubMed ID: 17570124
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
