113 related articles for article (PubMed ID: 9416427)
1. Inhibition of papain with 2-benzyl-3,4-epoxybutanoic acid esters. Mechanistic and stereochemical probe for cysteine protease catalysis.
Kim DH; Jin Y; Ryu CH
Bioorg Med Chem; 1997 Nov; 5(11):2103-8. PubMed ID: 9416427
[TBL] [Abstract][Full Text] [Related]
2. Design of protease inhibitors on the basis of substrate stereospecificity.
Kim DH
Biopolymers; 1999; 51(1):3-8. PubMed ID: 10380348
[TBL] [Abstract][Full Text] [Related]
3. Azapeptides as inhibitors and active site titrants for cysteine proteinases.
Xing R; Hanzlik RP
J Med Chem; 1998 Apr; 41(8):1344-51. PubMed ID: 9548822
[TBL] [Abstract][Full Text] [Related]
4. Syntheses and kinetic evaluation of racemic and optically active 2-benzyl-2-methyl-3,4-epoxybutanoic acids as irreversible inactivators for carboxypeptidase A.
Lee M; Kim DH
Bioorg Med Chem; 2002 Apr; 10(4):913-22. PubMed ID: 11836098
[TBL] [Abstract][Full Text] [Related]
5. Inactivation of cysteine proteases.
Govardhan CP; Abeles RH
Arch Biochem Biophys; 1996 Jun; 330(1):110-4. PubMed ID: 8651683
[TBL] [Abstract][Full Text] [Related]
6. Mechanistic studies on the inactivation of papain by epoxysuccinyl inhibitors.
Meara JP; Rich DH
J Med Chem; 1996 Aug; 39(17):3357-66. PubMed ID: 8765519
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and evaluation of chloromethyl sulfoxides as a new class of selective irreversible cysteine protease inhibitors.
Brouwer AJ; Bunschoten A; Liskamp RM
Bioorg Med Chem; 2007 Nov; 15(22):6985-93. PubMed ID: 17869119
[TBL] [Abstract][Full Text] [Related]
8. New peptidic cysteine protease inhibitors derived from the electrophilic alpha-amino acid aziridine-2,3-dicarboxylic acid.
Schirmeister T
J Med Chem; 1999 Feb; 42(4):560-72. PubMed ID: 10052963
[TBL] [Abstract][Full Text] [Related]
9. Cysteine protease inhibition by azapeptide esters.
Magrath J; Abeles RH
J Med Chem; 1992 Nov; 35(23):4279-83. PubMed ID: 1447732
[TBL] [Abstract][Full Text] [Related]
10. E64 [trans-epoxysuccinyl-L-leucylamido-(4-guanidino)butane] analogues as inhibitors of cysteine proteinases: investigation of S2 subsite interactions.
Gour-Salin BJ; Lachance P; Magny MC; Plouffe C; Ménard R; Storer AC
Biochem J; 1994 Apr; 299 ( Pt 2)(Pt 2):389-92. PubMed ID: 8172599
[TBL] [Abstract][Full Text] [Related]
11. Peptidyl beta-homo-aspartals (3-amino-4-carboxybutyraldehydes): new specific inhibitors of caspases.
Bajusz S; Fauszt I; Németh K; Barabás E; Juhász A; Patthy M; Bauer PI
Biopolymers; 1999; 51(1):109-18. PubMed ID: 10380358
[TBL] [Abstract][Full Text] [Related]
12. Novel aza peptide inhibitors and active-site probes of papain-family cysteine proteases.
Verhelst SH; Witte MD; Arastu-Kapur S; Fonovic M; Bogyo M
Chembiochem; 2006 Jun; 7(6):943-50. PubMed ID: 16607671
[TBL] [Abstract][Full Text] [Related]
13. beta-Lactam derivatives as enzyme inhibitors: 1-peptidyl derivatives of 4-phenylazetidin-2-one as inhibitors of elastase and papain.
Achilles K; Schirmeister T; Otto HH
Arch Pharm (Weinheim); 2000 Aug; 333(8):243-53. PubMed ID: 11008374
[TBL] [Abstract][Full Text] [Related]
14. Peptide alpha-keto ester, alpha-keto amide, and alpha-keto acid inhibitors of calpains and other cysteine proteases.
Li Z; Patil GS; Golubski ZE; Hori H; Tehrani K; Foreman JE; Eveleth DD; Bartus RT; Powers JC
J Med Chem; 1993 Oct; 36(22):3472-80. PubMed ID: 8230139
[TBL] [Abstract][Full Text] [Related]
15. The mechanism of papain inhibition by peptidyl aldehydes.
Shokhen M; Khazanov N; Albeck A
Proteins; 2011 Mar; 79(3):975-85. PubMed ID: 21181719
[TBL] [Abstract][Full Text] [Related]
16. Interactions of papaya proteinase IV with inhibitors.
Buttle DJ; Ritonja A; Dando PM; Abrahamson M; Shaw EN; Wikstrom P; Turk V; Barrett AJ
FEBS Lett; 1990 Mar; 262(1):58-60. PubMed ID: 1690669
[TBL] [Abstract][Full Text] [Related]
17. Structure-activity relationships for inhibition of papain by peptide Michael acceptors.
Liu S; Hanzlik RP
J Med Chem; 1992 Mar; 35(6):1067-75. PubMed ID: 1552501
[TBL] [Abstract][Full Text] [Related]
18. A re-appraisal of the structural basis of stereochemical recognition in papain. Insensitivity of binding-site-catalytic-site signalling to P2-chirality in a time-dependent inhibition.
Templeton W; Kowlessur D; Thomas EW; Topham CM; Brocklehurst K
Biochem J; 1990 Mar; 266(3):645-51. PubMed ID: 2327953
[TBL] [Abstract][Full Text] [Related]
19. New non-peptidic inhibitors of papain derived from etacrynic acid.
Kaeppler U; Schirmeister T
Med Chem; 2005 Jul; 1(4):361-70. PubMed ID: 16789893
[TBL] [Abstract][Full Text] [Related]
20. Clarification of substrate specificity of papain by crystal analyses of complexes with covalent-type inhibitors.
Matsumoto K; Murata M; Sumiya S; Kitamura K; Ishida T
Biochim Biophys Acta; 1994 Oct; 1208(2):268-76. PubMed ID: 7947958
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]