These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

126 related articles for article (PubMed ID: 9421405)

  • 1. EM-800, a novel antiestrogen, acts as a pure antagonist of the transcriptional functions of estrogen receptors alpha and beta.
    Tremblay A; Tremblay GB; Labrie C; Labrie F; Giguère V
    Endocrinology; 1998 Jan; 139(1):111-8. PubMed ID: 9421405
    [TBL] [Abstract][Full Text] [Related]  

  • 2. The interaction of raloxifene and the active metabolite of the antiestrogen EM-800 (SC 5705) with the human estrogen receptor.
    Schafer JI; Liu H; Tonetti DA; Jordan VC
    Cancer Res; 1999 Sep; 59(17):4308-13. PubMed ID: 10485477
    [TBL] [Abstract][Full Text] [Related]  

  • 3. EM-652 (SCH 57068), a third generation SERM acting as pure antiestrogen in the mammary gland and endometrium.
    Labrie F; Labrie C; Bélanger A; Simard J; Gauthier S; Luu-The V; Mérand Y; Giguere V; Candas B; Luo S; Martel C; Singh SM; Fournier M; Coquet A; Richard V; Charbonneau R; Charpenet G; Tremblay A; Tremblay G; Cusan L; Veilleux R
    J Steroid Biochem Mol Biol; 1999; 69(1-6):51-84. PubMed ID: 10418981
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Comparison of the effects of the new orally active antiestrogen EM-800 with ICI 182 780 and toremifene on estrogen-sensitive parameters in the ovariectomized mouse.
    Martel C; Labrie C; Bélanger A; Gauthier S; Mérand Y; Li X; Provencher L; Candas B; Labrie F
    Endocrinology; 1998 May; 139(5):2486-92. PubMed ID: 9564862
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Cloning, chromosomal localization, and functional analysis of the murine estrogen receptor beta.
    Tremblay GB; Tremblay A; Copeland NG; Gilbert DJ; Jenkins NA; Labrie F; Giguère V
    Mol Endocrinol; 1997 Mar; 11(3):353-65. PubMed ID: 9058381
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Human estrogen receptor ligand activity inversion mutants: receptors that interpret antiestrogens as estrogens and estrogens as antiestrogens and discriminate among different antiestrogens.
    Montano MM; Ekena K; Krueger KD; Keller AL; Katzenellenbogen BS
    Mol Endocrinol; 1996 Mar; 10(3):230-42. PubMed ID: 8833652
    [TBL] [Abstract][Full Text] [Related]  

  • 7. EM-652 (SCH57068), a pure SERM having complete antiestrogenic activity in the mammary gland and endometrium.
    Labrie F; Labrie C; Bélanger A; Simard J; Giguère V; Tremblay A; Tremblay G
    J Steroid Biochem Mol Biol; 2001 Dec; 79(1-5):213-25. PubMed ID: 11850228
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Ligand-, cell-, and estrogen receptor subtype (alpha/beta)-dependent activation at GC-rich (Sp1) promoter elements.
    Saville B; Wormke M; Wang F; Nguyen T; Enmark E; Kuiper G; Gustafsson JA; Safe S
    J Biol Chem; 2000 Feb; 275(8):5379-87. PubMed ID: 10681512
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Analysis of estrogen receptor transcriptional enhancement by a nuclear hormone receptor coactivator.
    McInerney EM; Tsai MJ; O'Malley BW; Katzenellenbogen BS
    Proc Natl Acad Sci U S A; 1996 Sep; 93(19):10069-73. PubMed ID: 8816752
    [TBL] [Abstract][Full Text] [Related]  

  • 10. The carboxy-terminal F domain of the human estrogen receptor: role in the transcriptional activity of the receptor and the effectiveness of antiestrogens as estrogen antagonists.
    Montano MM; Müller V; Trobaugh A; Katzenellenbogen BS
    Mol Endocrinol; 1995 Jul; 9(7):814-25. PubMed ID: 7476965
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Binding characteristics of novel nonsteroidal antiestrogens to the rat uterine estrogen receptors.
    Martel C; Provencher L; Li X; St Pierre A; Leblanc G; Gauthier S; Mérand Y; Labrie F
    J Steroid Biochem Mol Biol; 1998 Feb; 64(3-4):199-205. PubMed ID: 9605415
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Blockade of the stimulatory effect of estrogens, OH-tamoxifen, OH-toremifene, droloxifene, and raloxifene on alkaline phosphatase activity by the antiestrogen EM-800 in human endometrial adenocarcinoma Ishikawa cells.
    Simard J; Sanchez R; Poirier D; Gauthier S; Singh SM; Merand Y; Belanger A; Labrie C; Labrie F
    Cancer Res; 1997 Aug; 57(16):3494-7. PubMed ID: 9270018
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Estrogen and antiestrogen effects on neonatal ovine uterine development.
    Carpenter KD; Gray CA; Bryan TM; Welsh TH; Spencer TE
    Biol Reprod; 2003 Aug; 69(2):708-17. PubMed ID: 12700189
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Cooperative activation of gene expression by agonists and antagonists mediated by estrogen receptor heteroligand dimer complexes.
    Liu S; Han SJ; Smith CL
    Mol Pharmacol; 2013 May; 83(5):1066-77. PubMed ID: 23462505
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Pure antiestrogens and breast cancer.
    Elkak AE; Mokbel K
    Curr Med Res Opin; 2001; 17(4):282-9. PubMed ID: 11922402
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Novel estrogenic action of the pesticide residue beta-hexachlorocyclohexane in human breast cancer cells.
    Steinmetz R; Young PC; Caperell-Grant A; Gize EA; Madhukar BV; Ben-Jonathan N; Bigsby RM
    Cancer Res; 1996 Dec; 56(23):5403-9. PubMed ID: 8968093
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Effect of twenty-four-week treatment with the antiestrogen EM-800 on estrogen-sensitive parameters in intact and ovariectomized mice.
    Luo S; Sourla A; Labrie C; Gauthier S; Merand Y; Belanger A; Labrie F
    Endocrinology; 1998 May; 139(5):2645-56. PubMed ID: 9564882
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Characterization of the effects of the novel non-steroidal antiestrogen EM-800 on basal and estrogen-induced proliferation of T-47D, ZR-75-1 and MCF-7 human breast cancer cells in vitro.
    Simard J; Labrie C; Bélanger A; Gauthier S; Singh SM; Mérand Y; Labrie F
    Int J Cancer; 1997 Sep; 73(1):104-12. PubMed ID: 9334816
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synergistic activation of estrogen receptor-mediated transcription by estradiol and protein kinase activators.
    Cho H; Katzenellenbogen BS
    Mol Endocrinol; 1993 Mar; 7(3):441-52. PubMed ID: 7683375
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Specific transcriptional response of four blockers of estrogen receptors on estradiol-modulated genes in the mouse mammary gland.
    Calvo E; Luu-The V; Belleau P; Martel C; Labrie F
    Breast Cancer Res Treat; 2012 Jul; 134(2):625-47. PubMed ID: 22678160
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.