255 related articles for article (PubMed ID: 9426470)
1. The benzodiazepine binding site of GABAA receptors.
Sigel E; Buhr A
Trends Pharmacol Sci; 1997 Nov; 18(11):425-9. PubMed ID: 9426470
[TBL] [Abstract][Full Text] [Related]
2. Functional domains of GABAA receptors.
Smith GB; Olsen RW
Trends Pharmacol Sci; 1995 May; 16(5):162-8. PubMed ID: 7624971
[TBL] [Abstract][Full Text] [Related]
3. A closer look at the high affinity benzodiazepine binding site on GABAA receptors.
Sigel E; Lüscher BP
Curr Top Med Chem; 2011; 11(2):241-6. PubMed ID: 21189125
[TBL] [Abstract][Full Text] [Related]
4. Allosteric ligands and their binding sites define γ-aminobutyric acid (GABA) type A receptor subtypes.
Olsen RW
Adv Pharmacol; 2015; 73():167-202. PubMed ID: 25637441
[TBL] [Abstract][Full Text] [Related]
5. Mapping of the benzodiazepine recognition site on GABA(A) receptors.
Sigel E
Curr Top Med Chem; 2002 Aug; 2(8):833-9. PubMed ID: 12171574
[TBL] [Abstract][Full Text] [Related]
6. GABA-induced uncoupling of GABA/benzodiazepine site interactions is mediated by increased GABAA receptor internalization and associated with a change in subunit composition.
Gutiérrez ML; Ferreri MC; Gravielle MC
Neuroscience; 2014 Jan; 257():119-29. PubMed ID: 24215979
[TBL] [Abstract][Full Text] [Related]
7. The Benzodiazepine Binding Sites of GABA
Sigel E; Ernst M
Trends Pharmacol Sci; 2018 Jul; 39(7):659-671. PubMed ID: 29716746
[TBL] [Abstract][Full Text] [Related]
8. Positive modulation of synaptic and extrasynaptic GABAA receptors by an antagonist of the high affinity benzodiazepine binding site.
Middendorp SJ; Maldifassi MC; Baur R; Sigel E
Neuropharmacology; 2015 Aug; 95():459-67. PubMed ID: 25963418
[TBL] [Abstract][Full Text] [Related]
9. A point mutation in the gamma2 subunit of gamma-aminobutyric acid type A receptors results in altered benzodiazepine binding site specificity.
Buhr A; Sigel E
Proc Natl Acad Sci U S A; 1997 Aug; 94(16):8824-9. PubMed ID: 9238062
[TBL] [Abstract][Full Text] [Related]
10. Analysis of γ-aminobutyric acid (GABA) type A receptor subtypes using isosteric and allosteric ligands.
Olsen RW
Neurochem Res; 2014 Oct; 39(10):1924-41. PubMed ID: 25015397
[TBL] [Abstract][Full Text] [Related]
11. Probing the molecular basis for affinity/potency- and efficacy-based subtype-selectivity exhibited by benzodiazepine-site modulators at GABA
Söderhielm PC; Balle T; Bak-Nyhus S; Zhang M; Hansen KM; Ahring PK; Jensen AA
Biochem Pharmacol; 2018 Dec; 158():339-358. PubMed ID: 30121248
[TBL] [Abstract][Full Text] [Related]
12. Relative positioning of classical benzodiazepines to the γ2-subunit of GABAA receptors.
Middendorp SJ; Hurni E; Schönberger M; Stein M; Pangerl M; Trauner D; Sigel E
ACS Chem Biol; 2014 Aug; 9(8):1846-53. PubMed ID: 24918742
[TBL] [Abstract][Full Text] [Related]
13. The effect of subunit composition of rat brain GABAA receptors on channel function.
Sigel E; Baur R; Trube G; Möhler H; Malherbe P
Neuron; 1990 Nov; 5(5):703-11. PubMed ID: 1699569
[TBL] [Abstract][Full Text] [Related]
14. Fishing for allosteric sites on GABA(A) receptors.
Olsen RW; Chang CS; Li G; Hanchar HJ; Wallner M
Biochem Pharmacol; 2004 Oct; 68(8):1675-84. PubMed ID: 15451411
[TBL] [Abstract][Full Text] [Related]
15. GABAA receptor subtypes: autoradiographic comparison of GABA, benzodiazepine, and convulsant binding sites in the rat central nervous system.
Olsen RW; McCabe RT; Wamsley JK
J Chem Neuroanat; 1990; 3(1):59-76. PubMed ID: 2156526
[TBL] [Abstract][Full Text] [Related]
16. The GABAA-BZR complex as target for the development of anxiolytic drugs.
Trincavelli ML; Da Pozzo E; Daniele S; Martini C
Curr Top Med Chem; 2012; 12(4):254-69. PubMed ID: 22204488
[TBL] [Abstract][Full Text] [Related]
17. Cerebellar GABAA receptor selective for a behavioural alcohol antagonist.
Lüddens H; Pritchett DB; Köhler M; Killisch I; Keinänen K; Monyer H; Sprengel R; Seeburg PH
Nature; 1990 Aug; 346(6285):648-51. PubMed ID: 2166916
[TBL] [Abstract][Full Text] [Related]
18. A residue close to α1 loop F disrupts modulation of GABAA receptors by benzodiazepines while their binding is maintained.
Baur R; Lüscher BP; Richter L; Sigel E
J Neurochem; 2010 Dec; 115(6):1478-85. PubMed ID: 20946417
[TBL] [Abstract][Full Text] [Related]
19. Two tyrosine residues on the alpha subunit are crucial for benzodiazepine binding and allosteric modulation of gamma-aminobutyric acidA receptors.
Amin J; Brooks-Kayal A; Weiss DS
Mol Pharmacol; 1997 May; 51(5):833-41. PubMed ID: 9145922
[TBL] [Abstract][Full Text] [Related]
20. Ligands for the benzodiazepine binding site--a survey.
Teuber L; Wätjens F; Jensen LH
Curr Pharm Des; 1999 May; 5(5):317-43. PubMed ID: 10213798
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]