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3. Only in the presence of immunophilins can cyclosporin and FK506 disrupt in vivo binding of calcineurin A to its autoinhibitory domain yet strengthen interaction between calcineurin A and B subunits. Chaudhuri B; Stephan C Biochem Biophys Res Commun; 1995 Oct; 215(2):781-90. PubMed ID: 7488022 [TBL] [Abstract][Full Text] [Related]
4. The complex of FK506-binding protein 12 and FK506 inhibits calcineurin phosphatase activity and IgE activation-induced cytokine transcripts, but not exocytosis, in mouse mast cells. Fruman DA; Bierer BE; Benes JE; Burakoff SJ; Austen KF; Katz HR J Immunol; 1995 Feb; 154(4):1846-51. PubMed ID: 7530743 [TBL] [Abstract][Full Text] [Related]
5. Competitive and slow-binding inhibition of calcineurin by drug x immunophilin complexes. Salowe SP; Hermes JD Arch Biochem Biophys; 1998 Jul; 355(2):165-74. PubMed ID: 9675023 [TBL] [Abstract][Full Text] [Related]
6. FKBP12-Dependent Inhibition of Calcineurin Mediates Immunosuppressive Antifungal Drug Action in Ianiri G; Applen Clancey S; Lee SC; Heitman J mBio; 2017 Oct; 8(5):. PubMed ID: 29066552 [TBL] [Abstract][Full Text] [Related]
7. FAP48, a new protein that forms specific complexes with both immunophilins FKBP59 and FKBP12. Prevention by the immunosuppressant drugs FK506 and rapamycin. Chambraud B; Radanyi C; Camonis JH; Shazand K; Rajkowski K; Baulieu EE J Biol Chem; 1996 Dec; 271(51):32923-9. PubMed ID: 8955134 [TBL] [Abstract][Full Text] [Related]
8. The immunosuppressant FK506 and its nonimmunosuppressive analog L-685,818 are toxic to Cryptococcus neoformans by inhibition of a common target protein. Odom A; Del Poeta M; Perfect J; Heitman J Antimicrob Agents Chemother; 1997 Jan; 41(1):156-61. PubMed ID: 8980772 [TBL] [Abstract][Full Text] [Related]
9. Design and synthesis of a rapamycin-based high affinity binding FKBP12 ligand. Chakraborty TK; Weber HP; Nicolaou KC Chem Biol; 1995 Mar; 2(3):157-61. PubMed ID: 9383417 [TBL] [Abstract][Full Text] [Related]
11. Structure-activity profiles of macrolactam immunosuppressant FK-506 analogues. Kawai M; Lane BC; Hsieh GC; Mollison KW; Carter GW; Luly JR FEBS Lett; 1993 Jan; 316(2):107-13. PubMed ID: 7678400 [TBL] [Abstract][Full Text] [Related]
12. Three-dimensional structure and actions of immunosuppressants and their immunophilins. Braun W; Kallen J; Mikol V; Walkinshaw MD; Wüthrich K FASEB J; 1995 Jan; 9(1):63-72. PubMed ID: 7529736 [TBL] [Abstract][Full Text] [Related]
13. Discovery of less nephrotoxic FK506 analogs and determining immunophilin dependence of immunosuppressant nephrotoxicity with a novel single-dose rat cisplatin potentiation assay. Mollison KW; Fey TA; Krause RA; Andrews JM; Bretheim PT; Brandt JA; Kawai M; Wagner R; Hsieh GC; Luly JR J Pharmacol Exp Ther; 1997 Dec; 283(3):1509-19. PubMed ID: 9400028 [TBL] [Abstract][Full Text] [Related]
14. Structure comparison of native and mutant human recombinant FKBP12 complexes with the immunosuppressant drug FK506 (tacrolimus). Itoh S; Navia MA Protein Sci; 1995 Nov; 4(11):2261-8. PubMed ID: 8563622 [TBL] [Abstract][Full Text] [Related]
15. Interaction of tacrolimus(FK506) and its metabolites with FKBP and calcineurin. Tamura K; Fujimura T; Iwasaki K; Sakuma S; Fujitsu T; Nakamura K; Shimomura K; Kuno T; Tanaka C; Kobayashi M Biochem Biophys Res Commun; 1994 Jul; 202(1):437-43. PubMed ID: 7518678 [TBL] [Abstract][Full Text] [Related]
16. 32-Ascomycinyloxyacetic acid derived immunosuppressants. Independence of immunophilin binding and immunosuppressive potency. Wagner R; Rhoades TA; Or YS; Lane BC; Hsieh G; Mollison KW; Luly JR J Med Chem; 1998 May; 41(11):1764-76. PubMed ID: 9599228 [TBL] [Abstract][Full Text] [Related]
17. Modeling the interaction between FK506 and FKBP12: a mechanism for formation of the calcineurin inhibitory complex. Ivery MT; Weiler L Bioorg Med Chem; 1997 Feb; 5(2):217-32. PubMed ID: 9061187 [TBL] [Abstract][Full Text] [Related]
19. Three distinct messenger RNAs can encode the human immunosuppressant-binding protein FKBP12. Peattie DA; Hsiao K; Benasutti M; Lippke JA Gene; 1994 Dec; 150(2):251-7. PubMed ID: 7529739 [TBL] [Abstract][Full Text] [Related]
20. FK506 binding protein 12 mediates sensitivity to both FK506 and rapamycin in murine mast cells. Fruman DA; Wood MA; Gjertson CK; Katz HR; Burakoff SJ; Bierer BE Eur J Immunol; 1995 Feb; 25(2):563-71. PubMed ID: 7533090 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]