137 related articles for article (PubMed ID: 9754930)
1. Amino acid residue 200 on the alpha1 subunit of GABA(A) receptors affects the interaction with selected benzodiazepine binding site ligands.
Schaerer MT; Buhr A; Baur R; Sigel E
Eur J Pharmacol; 1998 Aug; 354(2-3):283-7. PubMed ID: 9754930
[TBL] [Abstract][Full Text] [Related]
2. Residues at positions 206 and 209 of the alpha1 subunit of gamma-aminobutyric AcidA receptors influence affinities for benzodiazepine binding site ligands.
Buhr A; Schaerer MT; Baur R; Sigel E
Mol Pharmacol; 1997 Oct; 52(4):676-82. PubMed ID: 9380031
[TBL] [Abstract][Full Text] [Related]
3. A point mutation in the gamma2 subunit of gamma-aminobutyric acid type A receptors results in altered benzodiazepine binding site specificity.
Buhr A; Sigel E
Proc Natl Acad Sci U S A; 1997 Aug; 94(16):8824-9. PubMed ID: 9238062
[TBL] [Abstract][Full Text] [Related]
4. Subtle changes in residue 77 of the gamma subunit of alpha1beta2gamma2 GABAA receptors drastically alter the affinity for ligands of the benzodiazepine binding site.
Buhr A; Baur R; Sigel E
J Biol Chem; 1997 May; 272(18):11799-804. PubMed ID: 9115236
[TBL] [Abstract][Full Text] [Related]
5. Cloning and characterization of the human GABAA receptor alpha 4 subunit: identification of a unique diazepam-insensitive binding site.
Yang W; Drewe JA; Lan NC
Eur J Pharmacol; 1995 Nov; 291(3):319-25. PubMed ID: 8719416
[TBL] [Abstract][Full Text] [Related]
6. Identification of a residue in the gamma-aminobutyric acid type A receptor alpha subunit that differentially affects diazepam-sensitive and -insensitive benzodiazepine site binding.
Derry JM; Dunn SM; Davies M
J Neurochem; 2004 Mar; 88(6):1431-8. PubMed ID: 15009644
[TBL] [Abstract][Full Text] [Related]
7. Actions of two GABAA receptor benzodiazepine-site ligands that are mediated via non-γ2-dependent modulation.
Leppä E; Linden AM; Rabe H; Vekovischeva OY; Wulff P; Lüddens H; Wisden W; Korpi ER
Eur J Pharmacol; 2011 Sep; 666(1-3):111-21. PubMed ID: 21616065
[TBL] [Abstract][Full Text] [Related]
8. Two tyrosine residues on the alpha subunit are crucial for benzodiazepine binding and allosteric modulation of gamma-aminobutyric acidA receptors.
Amin J; Brooks-Kayal A; Weiss DS
Mol Pharmacol; 1997 May; 51(5):833-41. PubMed ID: 9145922
[TBL] [Abstract][Full Text] [Related]
9. Point mutations of the alpha 1 beta 2 gamma 2 gamma-aminobutyric acid(A) receptor affecting modulation of the channel by ligands of the benzodiazepine binding site.
Buhr A; Baur R; Malherbe P; Sigel E
Mol Pharmacol; 1996 Jun; 49(6):1080-4. PubMed ID: 8649346
[TBL] [Abstract][Full Text] [Related]
10. Binding of 1,4-benzodiazepines to a novel [3H]Ro15-4513 binding site in the rat spinal cord.
Maguire PA; Davies MF; Loew GH
Eur J Pharmacol; 1995 Jul; 280(2):167-73. PubMed ID: 7589182
[TBL] [Abstract][Full Text] [Related]
11. Structural elements of the gamma-aminobutyric acid type A receptor conferring subtype selectivity for benzodiazepine site ligands.
Renard S; Olivier A; Granger P; Avenet P; Graham D; Sevrin M; George P; Besnard F
J Biol Chem; 1999 May; 274(19):13370-4. PubMed ID: 10224099
[TBL] [Abstract][Full Text] [Related]
12. Affinity of various ligands for GABAA receptors containing alpha 4 beta 3 gamma 2, alpha 4 gamma 2, or alpha 1 beta 3 gamma 2 subunits.
Scholze P; Ebert V; Sieghart W
Eur J Pharmacol; 1996 May; 304(1-3):155-62. PubMed ID: 8813598
[TBL] [Abstract][Full Text] [Related]
13. Affinity of various benzodiazepine site ligands in mice with a point mutation in the GABA(A) receptor gamma2 subunit.
Ogris W; Pöltl A; Hauer B; Ernst M; Oberto A; Wulff P; Höger H; Wisden W; Sieghart W
Biochem Pharmacol; 2004 Oct; 68(8):1621-9. PubMed ID: 15451405
[TBL] [Abstract][Full Text] [Related]
14. Molecular and pharmacological characterization of GABA(A) receptor alpha1 subunit knockout mice.
Kralic JE; Korpi ER; O'Buckley TK; Homanics GE; Morrow AL
J Pharmacol Exp Ther; 2002 Sep; 302(3):1037-45. PubMed ID: 12183661
[TBL] [Abstract][Full Text] [Related]
15. Identification of benzodiazepine binding site residues in the gamma2 subunit of the gamma-aminobutyric acid(A) receptor.
Kucken AM; Wagner DA; Ward PR; Teissére JA; Boileau AJ; Czajkowski C
Mol Pharmacol; 2000 May; 57(5):932-9. PubMed ID: 10779376
[TBL] [Abstract][Full Text] [Related]
16. Alterations of the benzodiazepine site of rat alpha 6 beta 2 gamma 2-GABAA receptor by replacement of several divergent amino-terminal regions with the alpha 1 counterparts.
Im WB; Pregenzer JF; Binder JA; Alberts GL; Im HK
Br J Pharmacol; 1997 Feb; 120(4):559-64. PubMed ID: 9051290
[TBL] [Abstract][Full Text] [Related]
17. Labelling of diazepam-sensitive and -insensitive benzodiazepine receptors with [3H]tert-butyl-8-chloro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo [1,5-a][1,4]benzodiazepine 3-carboxylate (ZG-63).
Wong G; Gu ZQ; de Costa B; Skolnick P
Eur J Pharmacol; 1993 Sep; 247(1):57-63. PubMed ID: 8258361
[TBL] [Abstract][Full Text] [Related]
18. Allosteric modulation by benzodiazepine receptor ligands of the GABAA receptor channel expressed in Xenopus oocytes.
Sigel E; Baur R
J Neurosci; 1988 Jan; 8(1):289-95. PubMed ID: 2448430
[TBL] [Abstract][Full Text] [Related]
19. Characterization of novel ligands for wild-type and natural mutant diazepam-insensitive benzodiazepine receptors.
Wong G; Uusi-Oukari M; Hansen HC; Suzdak PD; Korpi ER
Eur J Pharmacol; 1995 Apr; 289(2):335-42. PubMed ID: 7621907
[TBL] [Abstract][Full Text] [Related]
20. Mechanism of alpha-subunit selectivity of benzodiazepine pharmacology at gamma-aminobutyric acid type A receptors.
Wingrove PB; Safo P; Wheat L; Thompson SA; Wafford KA; Whiting PJ
Eur J Pharmacol; 2002 Feb; 437(1-2):31-9. PubMed ID: 11864636
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]