BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

131 related articles for article (PubMed ID: 9767642)

  • 21. Antagonistic effects of novel non-peptide chlorobenzhydryl piperazine compounds on contractile response to bradykinin in the guinea-pig ileum.
    Kam YL; Ro JY; Kim HJ; Choo HY
    Eur J Pharmacol; 2005 Oct; 523(1-3):143-50. PubMed ID: 16226247
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Effects of a nonpeptide bradykinin B2 receptor antagonist, FR167344, on guinea-pig tracheal smooth muscle bradykinin receptors.
    Asano M; Sawai H; Hatori C; Inamura N; Fujiwara T; Nakahara K
    Can J Physiol Pharmacol; 1998; 76(10-11):1051-5. PubMed ID: 10100888
    [TBL] [Abstract][Full Text] [Related]  

  • 23. MEN 11270, A novel selective constrained peptide antagonist with high affinity at the human B2 kinin receptor.
    Meini S; Quartara L; Rizzi A; Patacchini R; Cucchi P; Giolitti A; Calò G; Regoli D; Criscuoli M; Maggi CA
    J Pharmacol Exp Ther; 1999 Jun; 289(3):1250-6. PubMed ID: 10336513
    [TBL] [Abstract][Full Text] [Related]  

  • 24. Nonpeptide bradykinin B2 receptor antagonists: conversion of rodent-selective bradyzide analogues into potent, orally-active human bradykinin B2 receptor antagonists.
    Dziadulewicz EK; Ritchie TJ; Hallett A; Snell CR; Davies JW; Wrigglesworth R; Dunstan AR; Bloomfield GC; Drake GS; McIntyre P; Brown MC; Burgess GM; Lee W; Davis C; Yaqoob M; Phagoo SB; Phillips E; Perkins MN; Campbell EA; Davis AJ; Rang HP
    J Med Chem; 2002 May; 45(11):2160-72. PubMed ID: 12014954
    [TBL] [Abstract][Full Text] [Related]  

  • 25. MEN16132, a novel potent and selective nonpeptide antagonist for the human bradykinin B2 receptor. In vitro pharmacology and molecular characterization.
    Cucchi P; Meini S; Bressan A; Catalani C; Bellucci F; Santicioli P; Lecci A; Faiella A; Rotondaro L; Giuliani S; Giolitti A; Quartara L; Maggi CA
    Eur J Pharmacol; 2005 Dec; 528(1-3):7-16. PubMed ID: 16324696
    [TBL] [Abstract][Full Text] [Related]  

  • 26. MEN16132, a novel potent and selective nonpeptide kinin B2 receptor antagonist: in vivo activity on bradykinin-induced bronchoconstriction and nasal mucosa microvascular leakage in anesthetized guinea pigs.
    Valenti C; Cialdai C; Giuliani S; Lecci A; Tramontana M; Meini S; Quartara L; Maggi CA
    J Pharmacol Exp Ther; 2005 Nov; 315(2):616-23. PubMed ID: 16027229
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Structure-activity relationships of novel peptide agonists of the human bradykinin B2 receptor.
    Bélanger S; Bovenzi V; Côté J; Neugebauer W; Amblard M; Martinez J; Lammek B; Savard M; Gobeil F
    Peptides; 2009 Apr; 30(4):777-87. PubMed ID: 19111586
    [TBL] [Abstract][Full Text] [Related]  

  • 28. Design and synthesis of novel sulfonamide-containing bradykinin hB2 receptor antagonists. 1. Synthesis and SAR of alpha,alpha-dimethylglycine sulfonamides.
    Fattori D; Rossi C; Fincham CI; Berettoni M; Calvani F; Catrambone F; Felicetti P; Gensini M; Terracciano R; Altamura M; Bressan A; Giuliani S; Maggi CA; Meini S; Valenti C; Quartara L
    J Med Chem; 2006 Jun; 49(12):3602-13. PubMed ID: 16759102
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Potent bradykinin B1 receptor antagonists: 4-substituted phenyl cyclohexanes.
    Su DS; Lim JL; Markowitz MK; Wan BL; Murphy KL; Reiss DR; Harrell CM; O'Malley SS; Ransom RW; Chang RS; Pettibone DJ; Tang C; Prueksaritanont T; Freidinger RM; Bock MG
    Bioorg Med Chem Lett; 2007 Jun; 17(11):3006-9. PubMed ID: 17428657
    [TBL] [Abstract][Full Text] [Related]  

  • 30. A non-peptide antagonist unusually selective for the human form of the bradykinin B2 receptor.
    Marceau F; Fortin JP; Morissette G; Dziadulewicz EK
    Int Immunopharmacol; 2003 Oct; 3(10-11):1529-36. PubMed ID: 12946450
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Pharmacological and functional characterization of the guinea-pig B2 bradykinin receptor stably expressed in CHO-K1 cell line.
    Robert C; Pruneau D; Paquet JL
    Br J Pharmacol; 2002 Jan; 135(2):462-8. PubMed ID: 11815382
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Antagonistic effects of FR 173657 on human, pig, rabbit, and guinea pig kinin receptors: an in vitro study.
    Rizzi A; Gobeil F; Bogoni G; Calò G; Campobasso C; Inamura N; Regoli D
    Can J Physiol Pharmacol; 1997 Jun; 75(6):601-8. PubMed ID: 9276136
    [TBL] [Abstract][Full Text] [Related]  

  • 33. LF 16.0335, a novel potent and selective nonpeptide antagonist of the human bradykinin B2 receptor.
    Pruneau D; Luccarini JM; Fouchet C; Defrêne E; Franck RM; Loillier B; Duclos H; Robert C; Cremers B; Bélichard P; Paquet JL
    Br J Pharmacol; 1998 Sep; 125(2):365-72. PubMed ID: 9786510
    [TBL] [Abstract][Full Text] [Related]  

  • 34. In vitro and in vivo effects of the new nonpeptide bradykinin B2 receptor antagonist, LF 16-0335C, on guinea-pig and rat kinin receptors.
    Pruneau D; Luccarini JM; Fouchet C; Defrêne E; Franck RM; Loillier B; Duclos H; Robert C; Cremers B; Bélichard P; Paquet JL
    Fundam Clin Pharmacol; 1999; 13(1):75-83. PubMed ID: 10027091
    [TBL] [Abstract][Full Text] [Related]  

  • 35. Two bradykinin binding sites with picomolar affinities.
    Manning DC; Vavrek R; Stewart JM; Snyder SH
    J Pharmacol Exp Ther; 1986 May; 237(2):504-12. PubMed ID: 2871174
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Novel pseudopeptides with high affinities for the human bradykinin B2 receptor.
    Chakravarty S; Connolly M; Kyle DJ
    Pept Res; 1995; 8(1):16-9. PubMed ID: 7756750
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Pharmacological characterization of ZD6021: a novel, orally active antagonist of the tachykinin receptors.
    Rumsey WL; Aharony D; Bialecki RA; Abbott BM; Barthlow HG; Caccese R; Ghanekar S; Lengel D; McCarthy M; Wenrich B; Undem B; Ohnmacht C; Shenvi A; Albert JS; Brown F; Bernstein PR; Russell K
    J Pharmacol Exp Ther; 2001 Jul; 298(1):307-15. PubMed ID: 11408556
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Bradykinin B2-receptor-mediated modulation of membrane currents in guinea-pig cardiomyocytes.
    Sakamoto N; Uemura H; Hara Y; Saito T; Masuda Y; Nakaya H
    Br J Pharmacol; 1998 Sep; 125(2):283-92. PubMed ID: 9786500
    [TBL] [Abstract][Full Text] [Related]  

  • 39. Design, synthesis, and structure-activity relationships of thieno[2,3-b]pyridin-4-one derivatives as a novel class of potent, orally active, non-peptide luteinizing hormone-releasing hormone receptor antagonists.
    Imada T; Cho N; Imaeda T; Hayase Y; Sasaki S; Kasai S; Harada M; Matsumoto H; Endo S; Suzuki N; Furuya S
    J Med Chem; 2006 Jun; 49(13):3809-25. PubMed ID: 16789738
    [TBL] [Abstract][Full Text] [Related]  

  • 40. SSR240612 [(2R)-2-[((3R)-3-(1,3-benzodioxol-5-yl)-3-[[(6-methoxy-2-naphthyl)sulfonyl]amino]propanoyl)amino]-3-(4-[[2R,6S)-2,6-dimethylpiperidinyl]methyl]phenyl)-N-isopropyl-N-methylpropanamide hydrochloride], a new nonpeptide antagonist of the bradykinin B1 receptor: biochemical and pharmacological characterization.
    Gougat J; Ferrari B; Sarran L; Planchenault C; Poncelet M; Maruani J; Alonso R; Cudennec A; Croci T; Guagnini F; Urban-Szabo K; Martinolle JP; Soubrié P; Finance O; Le Fur G
    J Pharmacol Exp Ther; 2004 May; 309(2):661-9. PubMed ID: 14747609
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 7.