239 related articles for article (PubMed ID: 9836615)
21. Synthesis and transporter binding properties of 3 beta-(4'-alkyl-, 4'-alkenyl-, and 4'-alkynylphenyl)nortropane-2 beta-carboxylic acid methyl esters: serotonin transporter selective analogs.
Blough BE; Abraham P; Lewin AH; Kuhar MJ; Boja JW; Carroll FI
J Med Chem; 1996 Sep; 39(20):4027-35. PubMed ID: 8831768
[TBL] [Abstract][Full Text] [Related]
22. Synthesis, biodistribution, and primate imaging of fluorine-18 labeled 2beta-carbo-1'-fluoro-2-propoxy-3beta-(4-chlorophenyl)tr opanes. Ligands for the imaging of dopamine transporters by positron emission tomography.
Xing D; Chen P; Keil R; Kilts CD; Shi B; Camp VM; Malveaux G; Ely T; Owens MJ; Votaw J; Davis M; Hoffman JM; BaKay RA; Subramanian T; Watts RL; Goodman MM
J Med Chem; 2000 Feb; 43(4):639-48. PubMed ID: 10691690
[TBL] [Abstract][Full Text] [Related]
23. Structure-activity relationships at monoamine transporters and muscarinic receptors for N-substituted-3alpha-(3'-chloro-, 4'-chloro-, and 4',4''-dichloro-substituted-diphenyl)methoxytropanes.
Newman AH; Robarge MJ; Howard IM; Wittkopp SL; George C; Kopajtic T; Izenwasser S; Katz JL
J Med Chem; 2001 Feb; 44(4):633-40. PubMed ID: 11170654
[TBL] [Abstract][Full Text] [Related]
24. Synthesis and biological evaluation of tropane-like 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR 12909) analogues.
Zhang Y; Joseph DB; Bowen WD; Flippen-Anderson JL; Dersch CM; Rothman RB; Jacobson AE; Rice KC
J Med Chem; 2001 Nov; 44(23):3937-45. PubMed ID: 11689080
[TBL] [Abstract][Full Text] [Related]
25. Synthesis and evaluation of dopamine and serotonin transporter inhibition by oxacyclic and carbacyclic analogues of methylphenidate.
Meltzer PC; Wang P; Blundell P; Madras BK
J Med Chem; 2003 Apr; 46(8):1538-45. PubMed ID: 12672255
[TBL] [Abstract][Full Text] [Related]
26. Synthesis and transporter binding properties of bridged piperazine analogues of 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR 12909).
Zhang Y; Rothman RB; Dersch CM; de Costa BR; Jacobson AE; Rice KC
J Med Chem; 2000 Dec; 43(25):4840-9. PubMed ID: 11123994
[TBL] [Abstract][Full Text] [Related]
27. Synthesis of 2beta-acyl-3beta-(substituted naphthyl)-8-azabicyclo[3.2.1]octanes and their binding affinities at dopamine and serotonin transport sites.
Davies HM; Gilliatt V; Kuhn LA; Saikali E; Ren P; Hammond PS; Sexton T; Childers SR
J Med Chem; 2001 May; 44(10):1509-15. PubMed ID: 11334561
[TBL] [Abstract][Full Text] [Related]
28. Synthesis, dopamine transporter affinity, dopamine uptake inhibition, and locomotor stimulant activity of 2-substituted 3 beta-phenyltropane derivatives.
Xu L; Kelkar SV; Lomenzo SA; Izenwasser S; Katz JL; Kline RH; Trudell ML
J Med Chem; 1997 Mar; 40(6):858-63. PubMed ID: 9083474
[TBL] [Abstract][Full Text] [Related]
29. Structure-activity relationship studies on a novel series of (S)-2beta-substituted 3alpha-[bis(4-fluoro- or 4-chlorophenyl)methoxy]tropane analogues for in vivo investigation.
Zou MF; Cao J; Kopajtic T; Desai RI; Katz JL; Newman AH
J Med Chem; 2006 Oct; 49(21):6391-9. PubMed ID: 17034144
[TBL] [Abstract][Full Text] [Related]
30. Synthesis, monoamine transporter binding, properties, and functional monoamine uptake activity of 3beta-[4-methylphenyl and 4-chlorophenyl]-2 beta-[5-(substituted phenyl)thiazol-2-yl]tropanes.
Gong PK; Blough BE; Brieaddy LE; Huang X; Kuhar MJ; Navarro HA; Carroll FI
J Med Chem; 2007 Jul; 50(15):3686-95. PubMed ID: 17602602
[TBL] [Abstract][Full Text] [Related]
31. Chemical synthesis and pharmacology of 6- and 7-hydroxylated 2-carbomethoxy-3-(p-tolyl)tropanes: antagonism of cocaine's locomotor stimulant effects.
Zhao L; Johnson KM; Zhang M; Flippen-Anderson J; Kozikowski AP
J Med Chem; 2000 Aug; 43(17):3283-94. PubMed ID: 10966747
[TBL] [Abstract][Full Text] [Related]
32. Synthesis and monoamine transporter affinity of 2beta-carbomethoxy-3beta-(2''-, 3''- or 4''-substituted) biphenyltropanes.
Tamagnan G; Baldwin RM; Kula NS; Baldessarini RJ; Innis RB
Bioorg Med Chem Lett; 2000 Aug; 10(16):1783-5. PubMed ID: 10969967
[TBL] [Abstract][Full Text] [Related]
33. Synthesis and pharmacology of site specific cocaine abuse treatment agents: 8-substituted isotropane (3-azabicyclo[3.2.1]octane) dopamine uptake inhibitors.
Kim DI; Schweri MM; Deutsch HM
J Med Chem; 2003 Apr; 46(8):1456-64. PubMed ID: 12672245
[TBL] [Abstract][Full Text] [Related]
34. Synthesis and monoamine transporter affinity of new 2beta-carbomethoxy-3beta-[4-(substituted thiophenyl)]phenyltropanes: discovery of a selective SERT antagonist with picomolar potency.
Tamagnan G; Alagille D; Fu X; Kula NS; Baldessarini RJ; Innis RB; Baldwin RM
Bioorg Med Chem Lett; 2005 Feb; 15(4):1131-3. PubMed ID: 15686927
[TBL] [Abstract][Full Text] [Related]
35. An enantioselective synthesis and biobehavioral evaluation of 7-fluoro-3-(p-fluorophenyl)-2-propyltropanes.
Prakash KR; Trzcinska M; Johnson KM; Kozikowski AP
Bioorg Med Chem Lett; 2000 Jul; 10(13):1443-6. PubMed ID: 10888328
[TBL] [Abstract][Full Text] [Related]
36. Highly selective chiral N-substituted 3alpha-[bis(4'-fluorophenyl)methoxy]tropane analogues for the dopamine transporter: synthesis and comparative molecular field analysis.
Robarge MJ; Agoston GE; Izenwasser S; Kopajtic T; George C; Katz JL; Newman AH
J Med Chem; 2000 Mar; 43(6):1085-93. PubMed ID: 10737741
[TBL] [Abstract][Full Text] [Related]
37. Synthesis and receptor binding properties of 2beta-alkynyl and 2beta-(1,2,3-triazol)substituted 3beta-(substituted phenyl)tropane derivatives.
Jin C; Navarro HA; Carroll FI
Bioorg Med Chem; 2008 May; 16(10):5529-35. PubMed ID: 18434164
[TBL] [Abstract][Full Text] [Related]
38. Synthesis and monoamine transporter binding of 2-(diarylmethoxymethyl)-3 beta-aryltropane derivatives.
Xu L; Kulkarni SS; Izenwasser S; Katz JL; Kopajtic T; Lomenzo SA; Newman AH; Trudell ML
J Med Chem; 2004 Mar; 47(7):1676-82. PubMed ID: 15027858
[TBL] [Abstract][Full Text] [Related]
39. Further structurally constrained analogues of cis-(6-benzhydrylpiperidin-3-yl)benzylamine with elucidation of bioactive conformation: discovery of 1,4-diazabicyclo[3.3.1]nonane derivatives and evaluation of their biological properties for the monoamine transporters.
Kolhatkar R; Cook CD; Ghorai SK; Deschamps J; Beardsley PM; Reith ME; Dutta AK
J Med Chem; 2004 Oct; 47(21):5101-13. PubMed ID: 15456254
[TBL] [Abstract][Full Text] [Related]
40. Cocaine and 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid ester and amide analogues. New high-affinity and selective compounds for the dopamine transporter.
Carroll FI; Kotian P; Dehghani A; Gray JL; Kuzemko MA; Parham KA; Abraham P; Lewin AH; Boja JW; Kuhar MJ
J Med Chem; 1995 Jan; 38(2):379-88. PubMed ID: 7830281
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
