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  • Title: Synthesis and evaluation of amides surrogates of dopamine D3 receptor ligands.
    Author: Jean M, Renault J, Levoin N, Danvy D, Calmels T, Berrebi-Bertrand I, Robert P, Schwartz JC, Lecomte JM, Uriac P, Capet M.
    Journal: Bioorg Med Chem Lett; 2010 Sep 15; 20(18):5376-9. PubMed ID: 20708933.
    Abstract:
    Isosteric replacement of the amide function and modulation of the arylpiperazine moiety of known dopamine D3 receptor ligands led to potent and selective compounds. Enhanced bioavailability and preferential brain distribution make compound 6c a good candidate for pharmacological and clinical evaluation.
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