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7. Synthesis and evaluation of diphenyl phosphonate esters as inhibitors of the trypsin-like granzymes A and K and mast cell tryptase. Jackson DS, Fraser SA, Ni LM, Kam CM, Winkler U, Johnson DA, Froelich CJ, Hudig D, Powers JC. J Med Chem; 1998 Jun 18; 41(13):2289-301. PubMed ID: 9632362 [Abstract] [Full Text] [Related]
8. Bis(5-amidino-2-benzimidazolyl)methane and related amidines are potent, reversible inhibitors of mast cell tryptases. Caughey GH, Raymond WW, Bacci E, Lombardy RJ, Tidwell RR. J Pharmacol Exp Ther; 1993 Feb 18; 264(2):676-82. PubMed ID: 8437115 [Abstract] [Full Text] [Related]
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12. Dibasic inhibitors of human mast cell tryptase. Part 1: synthesis and optimization of a novel class of inhibitors. Rice KD, Gangloff AR, Kuo EY, Dener JM, Wang VR, Lum R, Newcomb WS, Havel C, Putnam D, Cregar L, Wong M, Warne RL. Bioorg Med Chem Lett; 2000 Oct 16; 10(20):2357-60. PubMed ID: 11055355 [Abstract] [Full Text] [Related]
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14. 1,2-Benzisothiazol-3-one 1,1-dioxide inhibitors of human mast cell tryptase. Combrink KD, Gülgeze HB, Meanwell NA, Pearce BC, Zulan P, Bisacchi GS, Roberts DG, Stanley P, Seiler SM. J Med Chem; 1998 Nov 19; 41(24):4854-60. PubMed ID: 9822554 [Abstract] [Full Text] [Related]
15. Neutrophil myeloperoxidase is a potent and selective inhibitor of mast cell tryptase. Cregar L, Elrod KC, Putnam D, Moore WR. Arch Biochem Biophys; 1999 Jun 01; 366(1):125-30. PubMed ID: 10334872 [Abstract] [Full Text] [Related]
16. Inhibition of human mast cell tryptase by benzamidine derivatives. Stürzebecher J, Prasa D, Sommerhoff CP. Biol Chem Hoppe Seyler; 1992 Oct 01; 373(10):1025-30. PubMed ID: 1418674 [Abstract] [Full Text] [Related]
17. Structure based design of 4-(3-aminomethylphenyl)piperidinyl-1-amides: novel, potent, selective, and orally bioavailable inhibitors of betaII tryptase. Levell J, Astles P, Eastwood P, Cairns J, Houille O, Aldous S, Merriman G, Whiteley B, Pribish J, Czekaj M, Liang G, Maignan S, Guilloteau JP, Dupuy A, Davidson J, Harrison T, Morley A, Watson S, Fenton G, McCarthy C, Romano J, Mathew R, Engers D, Gardyan M, Sides K, Kwong J, Tsay J, Rebello S, Shen L, Wang J, Luo Y, Giardino O, Lim HK, Smith K, Pauls H. Bioorg Med Chem; 2005 Apr 15; 13(8):2859-72. PubMed ID: 15781396 [Abstract] [Full Text] [Related]
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