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Journal Abstract Search

214 related items for PubMed ID: 11714875

  • 1. Constitutive activity of histamine h(3) receptors stably expressed in SK-N-MC cells: display of agonism and inverse agonism by H(3) antagonists.
    Wieland K, Bongers G, Yamamoto Y, Hashimoto T, Yamatodani A, Menge WM, Timmerman H, Lovenberg TW, Leurs R.
    J Pharmacol Exp Ther; 2001 Dec; 299(3):908-14. PubMed ID: 11714875
    [Abstract] [Full Text] [Related]

  • 2. G protein-dependent pharmacology of histamine H3 receptor ligands: evidence for heterogeneous active state receptor conformations.
    Krueger KM, Witte DG, Ireland-Denny L, Miller TR, Baranowski JL, Buckner S, Milicic I, Esbenshade TA, Hancock AA.
    J Pharmacol Exp Ther; 2005 Jul; 314(1):271-81. PubMed ID: 15821027
    [Abstract] [Full Text] [Related]

  • 3. The histamine H3 receptor antagonist clobenpropit enhances GABA release to protect against NMDA-induced excitotoxicity through the cAMP/protein kinase A pathway in cultured cortical neurons.
    Dai H, Fu Q, Shen Y, Hu W, Zhang Z, Timmerman H, Leurs R, Chen Z.
    Eur J Pharmacol; 2007 Jun 01; 563(1-3):117-23. PubMed ID: 17350613
    [Abstract] [Full Text] [Related]

  • 4. Generation and characterization of highly constitutive active histamine H3 receptors.
    Takahashi K, Tokita S, Kotani H.
    J Pharmacol Exp Ther; 2003 Oct 01; 307(1):213-8. PubMed ID: 12954820
    [Abstract] [Full Text] [Related]

  • 5. Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives.
    Gbahou F, Vincent L, Humbert-Claude M, Tardivel-Lacombe J, Chabret C, Arrang JM.
    Br J Pharmacol; 2006 Apr 01; 147(7):744-54. PubMed ID: 16432504
    [Abstract] [Full Text] [Related]

  • 6. High constitutive activity of native H3 receptors regulates histamine neurons in brain.
    Morisset S, Rouleau A, Ligneau X, Gbahou F, Tardivel-Lacombe J, Stark H, Schunack W, Ganellin CR, Schwartz JC, Arrang JM.
    Nature; 2000 Dec 14; 408(6814):860-4. PubMed ID: 11130725
    [Abstract] [Full Text] [Related]

  • 7. Effects of betahistine at histamine H3 receptors: mixed inverse agonism/agonism in vitro and partial inverse agonism in vivo.
    Gbahou F, Davenas E, Morisset S, Arrang JM.
    J Pharmacol Exp Ther; 2010 Sep 01; 334(3):945-54. PubMed ID: 20530654
    [Abstract] [Full Text] [Related]

  • 8. Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.
    Rouleau A, Ligneau X, Tardivel-Lacombe J, Morisset S, Gbahou F, Schwartz JC, Arrang JM.
    Br J Pharmacol; 2002 Jan 01; 135(2):383-92. PubMed ID: 11815373
    [Abstract] [Full Text] [Related]

  • 9. Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: synthesis, pharmacological evaluation, and cross-target QSAR studies.
    Lim HD, Istyastono EP, van de Stolpe A, Romeo G, Gobbi S, Schepers M, Lahaye R, Menge WM, Zuiderveld OP, Jongejan A, Smits RA, Bakker RA, Haaksma EE, Leurs R, de Esch IJ.
    Bioorg Med Chem; 2009 Jun 01; 17(11):3987-94. PubMed ID: 19414267
    [Abstract] [Full Text] [Related]

  • 10. Cloning of rat histamine H(3) receptor reveals distinct species pharmacological profiles.
    Lovenberg TW, Pyati J, Chang H, Wilson SJ, Erlander MG.
    J Pharmacol Exp Ther; 2000 Jun 01; 293(3):771-8. PubMed ID: 10869375
    [Abstract] [Full Text] [Related]

  • 11. Constitutive activity of the histamine H3 receptor.
    Arrang JM, Morisset S, Gbahou F.
    Trends Pharmacol Sci; 2007 Jul 01; 28(7):350-7. PubMed ID: 17573125
    [Abstract] [Full Text] [Related]

  • 12. Two novel and selective nonimidazole histamine H3 receptor antagonists A-304121 and A-317920: I. In vitro pharmacological effects.
    Esbenshade TA, Krueger KM, Miller TR, Kang CH, Denny LI, Witte DG, Yao BB, Fox GB, Faghih R, Bennani YL, Williams M, Hancock AA.
    J Pharmacol Exp Ther; 2003 Jun 01; 305(3):887-96. PubMed ID: 12606603
    [Abstract] [Full Text] [Related]

  • 13. Comparison of the binding distribution of agonist and antagonist ligands for histamine H3 receptors in pig brain by quantitative autoradiography.
    Mezzomo K, Cumming P, Minuzzi L.
    Eur J Pharmacol; 2007 Jun 14; 564(1-3):75-9. PubMed ID: 17350614
    [Abstract] [Full Text] [Related]

  • 14. Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonist.
    Esbenshade TA, Fox GB, Krueger KM, Baranowski JL, Miller TR, Kang CH, Denny LI, Witte DG, Yao BB, Pan JB, Faghih R, Bennani YL, Williams M, Hancock AA.
    Biochem Pharmacol; 2004 Sep 01; 68(5):933-45. PubMed ID: 15294456
    [Abstract] [Full Text] [Related]

  • 15. The human histamine H3 receptor couples to GIRK channels in Xenopus oocytes.
    Sahlholm K, Nilsson J, Marcellino D, Fuxe K, Arhem P.
    Eur J Pharmacol; 2007 Jul 19; 567(3):206-10. PubMed ID: 17537431
    [Abstract] [Full Text] [Related]

  • 16. Protean agonism at histamine H3 receptors in vitro and in vivo.
    Gbahou F, Rouleau A, Morisset S, Parmentier R, Crochet S, Lin JS, Ligneau X, Tardivel-Lacombe J, Stark H, Schunack W, Ganellin CR, Schwartz JC, Arrang JM.
    Proc Natl Acad Sci U S A; 2003 Sep 16; 100(19):11086-91. PubMed ID: 12960366
    [Abstract] [Full Text] [Related]

  • 17. Synthesis and structure-activity relationships of conformationally constrained histamine H(3) receptor agonists.
    Kitbunnadaj R, Zuiderveld OP, De Esch IJ, Vollinga RC, Bakker R, Lutz M, Spek AL, Cavoy E, Deltent MF, Menge WM, Timmerman H, Leurs R.
    J Med Chem; 2003 Dec 04; 46(25):5445-57. PubMed ID: 14640553
    [Abstract] [Full Text] [Related]

  • 18. Detection of multiple H3 receptor affinity states utilizing [3H]A-349821, a novel, selective, non-imidazole histamine H3 receptor inverse agonist radioligand.
    Witte DG, Yao BB, Miller TR, Carr TL, Cassar S, Sharma R, Faghih R, Surber BW, Esbenshade TA, Hancock AA, Krueger KM.
    Br J Pharmacol; 2006 Jul 04; 148(5):657-70. PubMed ID: 16715122
    [Abstract] [Full Text] [Related]

  • 19. Cloning and characterization of a novel human histamine receptor.
    Morse KL, Behan J, Laz TM, West RE, Greenfeder SA, Anthes JC, Umland S, Wan Y, Hipkin RW, Gonsiorek W, Shin N, Gustafson EL, Qiao X, Wang S, Hedrick JA, Greene J, Bayne M, Monsma FJ.
    J Pharmacol Exp Ther; 2001 Mar 04; 296(3):1058-66. PubMed ID: 11181941
    [Abstract] [Full Text] [Related]

  • 20. Detailed pharmacological characterization of GT-2331 for the rat histamine H3 receptor.
    Ito S, Yoshimoto R, Miyamoto Y, Mitobe Y, Nakamura T, Ishihara A, MacNeil DJ, Kanatani A, Tokita S.
    Eur J Pharmacol; 2006 Jan 04; 529(1-3):40-6. PubMed ID: 16316645
    [Abstract] [Full Text] [Related]

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