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Journal Abstract Search


224 related items for PubMed ID: 12869657

  • 1. Tiotidine, a histamine H2 receptor inverse agonist that binds with high affinity to an inactive G-protein-coupled form of the receptor. Experimental support for the cubic ternary complex model.
    Monczor F, Fernandez N, Legnazzi BL, Riveiro ME, Baldi A, Shayo C, Davio C.
    Mol Pharmacol; 2003 Aug; 64(2):512-20. PubMed ID: 12869657
    [Abstract] [Full Text] [Related]

  • 2. Mechanisms of inverse agonism at histamine H(2) receptors - potential benefits and concerns.
    Monczor F.
    Inflammopharmacology; 2006 Mar; 14(1-2):89-96. PubMed ID: 16835719
    [Abstract] [Full Text] [Related]

  • 3. Similar apparent constitutive activity of human histamine H(2)-receptor fused to long and short splice variants of G(salpha).
    Wenzel-Seifert K, Kelley MT, Buschauer A, Seifert R.
    J Pharmacol Exp Ther; 2001 Dec; 299(3):1013-20. PubMed ID: 11714890
    [Abstract] [Full Text] [Related]

  • 4. Theoretical studies on the histamine H2 receptor: molecular mechanism of action of antagonists.
    Giraldo J, Martín M, Campillo M, Pardo L.
    Mol Pharmacol; 1992 Aug; 42(2):373-81. PubMed ID: 1355265
    [Abstract] [Full Text] [Related]

  • 5. Tiotidine, a classical H2-antagonist, presents characteristics of an inverse agonist in U937 cell line.
    Monczor F, Legnazzi BL, Rivera E, Davio C.
    Inflamm Res; 1998 Aug; 47 Suppl 1():S42-3. PubMed ID: 9561408
    [No Abstract] [Full Text] [Related]

  • 6. Expression of histamine H2 receptor in Chinese hamster ovary cells: a probe to study the desensitization mechanism.
    Fukushima Y, Matsuhashi N, Saitoh T, Mori H, Kodama T, Sugano K, Yazaki Y.
    J Gastroenterol; 1994 Jul; 29 Suppl 7():68-72. PubMed ID: 7921157
    [Abstract] [Full Text] [Related]

  • 7. Mutations of Cys-17 and Ala-271 in the human histamine H2 receptor determine the species selectivity of guanidine-type agonists and increase constitutive activity.
    Preuss H, Ghorai P, Kraus A, Dove S, Buschauer A, Seifert R.
    J Pharmacol Exp Ther; 2007 Jun; 321(3):975-82. PubMed ID: 17347323
    [Abstract] [Full Text] [Related]

  • 8. Is [3H]-tiotidine a specific ligand for the H2-receptor?
    Batzri S, Harmon JW.
    Pharmacology; 1986 Jun; 32(5):241-7. PubMed ID: 2872690
    [Abstract] [Full Text] [Related]

  • 9. Heterologous expression of rat epitope-tagged histamine H2 receptors in insect Sf9 cells.
    Beukers MW, Klaassen CH, De Grip WJ, Verzijl D, Timmerman H, Leurs R.
    Br J Pharmacol; 1997 Nov; 122(5):867-74. PubMed ID: 9384502
    [Abstract] [Full Text] [Related]

  • 10. Desensitization of canine histamine H2 receptor expressed in Chinese hamster ovary cells.
    Fukushima Y, Oka Y, Katagiri H, Saitoh T, Asano T, Ishihara H, Matsuhashi N, Kodama T, Yazaki Y, Sugano K.
    Biochem Biophys Res Commun; 1993 Feb 15; 190(3):1149-55. PubMed ID: 8382488
    [Abstract] [Full Text] [Related]

  • 11. Histamine H2 receptor trafficking: role of arrestin, dynamin, and clathrin in histamine H2 receptor internalization.
    Fernandez N, Monczor F, Baldi A, Davio C, Shayo C.
    Mol Pharmacol; 2008 Oct 15; 74(4):1109-18. PubMed ID: 18617631
    [Abstract] [Full Text] [Related]

  • 12. Alteration of intracellular histamine H2 receptor cycling precedes antagonist-induced upregulation.
    Osawa S, Kajimura M, Yamamoto S, Ikuma M, Mochizuki C, Iwasaki H, Hishida A, Terakawa S.
    Am J Physiol Gastrointest Liver Physiol; 2005 Nov 15; 289(5):G880-9. PubMed ID: 15961859
    [Abstract] [Full Text] [Related]

  • 13. G protein-linked receptors labeled by [3H]histamine in guinea pig cerebral cortex. II. Mechanistic basis for multiple states of affinity [corrected].
    Sinkins WG, Wells JW.
    Mol Pharmacol; 1993 Apr 15; 43(4):583-94. PubMed ID: 8097275
    [Abstract] [Full Text] [Related]

  • 14. The cardiac pharmacology of tiotidine (LCL 125, 211): a new histamine H2-receptor antagonist.
    Trzeciakowski JP, Levi R.
    J Pharmacol Exp Ther; 1980 Sep 15; 214(3):629-34. PubMed ID: 6105207
    [Abstract] [Full Text] [Related]

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  • 16. Histamine H2 receptor desensitization in HL-60 human promyelocytic leukemia cells.
    Sawutz DG, Kalinyak K, Whitsett JA, Johnson CL.
    J Pharmacol Exp Ther; 1984 Oct 15; 231(1):1-7. PubMed ID: 6208354
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  • 19. Interaction of the new histamine H2-receptor antagonist pibutidine hydrochloride with canine cloned H2-receptor expressed cells.
    Kaku S, Isobe Y, Kiuchi Y, Tanaka M, Muramatsu M, Higuchi S.
    Arzneimittelforschung; 1999 Jan 15; 49(1):67-71. PubMed ID: 10028383
    [Abstract] [Full Text] [Related]

  • 20. Molecular properties of central and peripheral histamine H1 and H2 receptors.
    Carman-Krzan M, Lipnik-Stangelj M.
    Pflugers Arch; 2000 Jan 15; 439(3 Suppl):R131-2. PubMed ID: 10653166
    [Abstract] [Full Text] [Related]


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