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Journal Abstract Search

108 related items for PubMed ID: 15727846

  • 1. Novel acetylcholinesterase inhibitor as increasing agent on rhythmic bladder contractions: SAR of 8-{3-[1-(3-fluorobenzyl)piperidin-4-yl]propanoyl}-1,2,5,6-tetrahydro-4H-pyrrolo[3,2,1-ij]quinolin-4-one (TAK-802) and related compounds.
    Ishichi Y, Sasaki M, Setoh M, Tsukamoto T, Miwatashi S, Nagabukuro H, Okanishi S, Imai S, Saikawa R, Doi T, Ishihara Y.
    Bioorg Med Chem; 2005 Mar 15; 13(6):1901-11. PubMed ID: 15727846
    [Abstract] [Full Text] [Related]

  • 2. Effects of TAK-802, a novel acetylcholinesterase inhibitor, on distension-induced rhythmic bladder contractions in rats and guinea pigs.
    Nagabukuro H, Okanishi S, Imai S, Ishichi Y, Ishihara Y, Doi T.
    Eur J Pharmacol; 2004 Feb 06; 485(1-3):299-305. PubMed ID: 14757154
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  • 3. Effects of TAK-802, a novel acetylcholinesterase inhibitor, and various cholinomimetics on the urodynamic characteristics in anesthetized guinea pigs.
    Nagabukuro H, Okanishi S, Doi T.
    Eur J Pharmacol; 2004 Jun 28; 494(2-3):225-32. PubMed ID: 15212979
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  • 4. Differential effects of TAK-802, a selective acetylcholinesterase inhibitor, and carbamate acetylcholinesterase inhibitors on contraction of the detrusor smooth muscle of the guinea pig.
    Nagabukuro H, Doi T.
    Life Sci; 2005 Nov 12; 77(26):3276-86. PubMed ID: 15978636
    [Abstract] [Full Text] [Related]

  • 5. Effects of the selective acetylcholinesterase inhibitor TAK-802 on the voiding behavior and bladder mass increase in rats with partial bladder outlet obstruction.
    Hashimoto T, Nagabukuro H, Doi T.
    J Urol; 2005 Sep 12; 174(3):1137-41. PubMed ID: 16094081
    [Abstract] [Full Text] [Related]

  • 6. Synthesis and evaluation of novel 4-[(3H,3aH,6aH)-3-phenyl)-4,6-dioxo-2-phenyldihydro-2H-pyrrolo[3,4-d]isoxazol-5(3H,6H,6aH)-yl]benzoic acid derivatives as potent acetylcholinesterase inhibitors and anti-amnestic agents.
    Anand P, Singh B.
    Bioorg Med Chem; 2012 Jan 01; 20(1):521-30. PubMed ID: 22172310
    [Abstract] [Full Text] [Related]

  • 7. Synthesis and structure-activity relationships of a novel series of 2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-dioxide K(ATP) channel openers: discovery of (-)-(9S)-9-(3-bromo-4-fluorophenyl)-2,3,5,6,7,9- hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-dioxide (A-278637), a potent K(ATP) opener that selectively inhibits spontaneous bladder contractions.
    Carroll WA, Altenbach RJ, Bai H, Brioni JD, Brune ME, Buckner SA, Cassidy C, Chen Y, Coghlan MJ, Daza AV, Drizin I, Fey TA, Fitzgerald M, Gopalakrishnan M, Gregg RJ, Henry RF, Holladay MW, King LL, Kort ME, Kym PR, Milicic I, Tang R, Turner SC, Whiteaker KL, Yi L, Zhang H, Sullivan JP.
    J Med Chem; 2004 Jun 03; 47(12):3163-79. PubMed ID: 15163196
    [Abstract] [Full Text] [Related]

  • 8. An atom economic synthesis and AChE inhibitory activity of novel dispiro 7-aryltetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole and 4-aryloctahydroindolizine N-methylpiperidin-4-one hybrid heterocycles.
    Sivakumar S, Ranjith Kumar R, Ali MA, Choon TS.
    Eur J Med Chem; 2013 Jul 03; 65():240-8. PubMed ID: 23721952
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  • 10. One-pot microwave assisted stereoselective synthesis of novel dihydro-2'H-spiro[indene-2,1'-pyrrolo-[3,4-c]pyrrole]-tetraones and evaluation of their antimycobacterial activity and inhibition of AChE.
    Bharkavi C, Vivek Kumar S, Ashraf Ali M, Osman H, Muthusubramanian S, Perumal S.
    Bioorg Med Chem Lett; 2017 Jul 15; 27(14):3071-3075. PubMed ID: 28552337
    [Abstract] [Full Text] [Related]

  • 11. (-)-(9S)-9-(3-Bromo-4-fluorophenyl)-2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-dioxide (A-278637): a novel ATP-sensitive potassium channel opener efficacious in suppressing urinary bladder contractions. I. In vitro characterization.
    Gopalakrishnan M, Buckner SA, Whiteaker KL, Shieh CC, Molinari EJ, Milicic I, Daza AV, Davis-Taber R, Scott VE, Sellers D, Chess-Williams R, Chapple CR, Liu Y, Liu D, Brioni JD, Sullivan JP, Williams M, Carroll WA, Coghlan MJ.
    J Pharmacol Exp Ther; 2002 Oct 15; 303(1):379-86. PubMed ID: 12235274
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  • 14. Inhibition of acetylcholinesterase by two arylderivatives: 3a-Acetoxy-5H-pyrrolo (1,2-a) (3, 1)benzoxazin- 1,5-(3aH)-dione and cis-N-p-Acetoxy-phenylisomaleimide.
    Correa-Basurto J, Espinosa-Raya J, González-May M, Espinoza-Fonseca LM, Vázquez-Alcántara I, Trujillo-Ferrara J.
    J Enzyme Inhib Med Chem; 2006 Apr 15; 21(2):133-8. PubMed ID: 16789426
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  • 15. Novel Tacrine-Based Pyrano[3',4':5,6]pyrano[2,3-b]quinolinones: Synthesis and Cholinesterase Inhibitory Activity.
    Hariri R, Afshar Z, Mahdavi M, Safavi M, Saeedi M, Najafi Z, Sabourian R, Karimpour-Razkenari E, Edraki N, Moghadam FH, Shafiee A, Khanavi M, Akbarzadeh T.
    Arch Pharm (Weinheim); 2016 Dec 15; 349(12):915-924. PubMed ID: 27910192
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  • 17. Conscious voiding during bladder obstruction in guinea pigs correlates with contractile activity of isolated bladders.
    Nicholas S, Keightley L, Brookes S, Costa M, Gibbins I, Zagorodnyuk V.
    Auton Neurosci; 2015 Dec 15; 193():74-83. PubMed ID: 26282433
    [Abstract] [Full Text] [Related]

  • 18. Design, synthesis and evaluation of flavonoid derivatives as potent AChE inhibitors.
    Sheng R, Lin X, Zhang J, Chol KS, Huang W, Yang B, He Q, Hu Y.
    Bioorg Med Chem; 2009 Sep 15; 17(18):6692-8. PubMed ID: 19692250
    [Abstract] [Full Text] [Related]

  • 19. The role of cholinesterases in rat urinary bladder contractility.
    Nakahara T, Kubota Y, Sakamoto K, Ishii K.
    Urol Res; 2003 Jul 15; 31(3):223-6. PubMed ID: 12736766
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  • 20. Synthesis and anti-cholinesterase activity of new 7-hydroxycoumarin derivatives.
    Alipour M, Khoobi M, Moradi A, Nadri H, Homayouni Moghadam F, Emami S, Hasanpour Z, Foroumadi A, Shafiee A.
    Eur J Med Chem; 2014 Jul 23; 82():536-44. PubMed ID: 24941128
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