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Journal Abstract Search

479 related items for PubMed ID: 16414180

  • 21. A 3D QSAR model of 17beta-HSD1 inhibitors based on a thieno[2,3-d]pyrimidin-4(3H)-one core applying molecular dynamics simulations and ligand-protein docking.
    Karkola S, Lilienkampf A, Wähälä K.
    ChemMedChem; 2008 Mar; 3(3):461-72. PubMed ID: 18224704
    [Abstract] [Full Text] [Related]

  • 22. Substituted 6-phenyl-2-naphthols. Potent and selective nonsteroidal inhibitors of 17beta-hydroxysteroid dehydrogenase type 1 (17beta-HSD1): design, synthesis, biological evaluation, and pharmacokinetics.
    Marchais-Oberwinkler S, Kruchten P, Frotscher M, Ziegler E, Neugebauer A, Bhoga U, Bey E, Müller-Vieira U, Messinger J, Thole H, Hartmann RW.
    J Med Chem; 2008 Aug 14; 51(15):4685-98. PubMed ID: 18630892
    [Abstract] [Full Text] [Related]

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  • 24. Bicyclic substituted hydroxyphenylmethanones as novel inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) for the treatment of estrogen-dependent diseases.
    Oster A, Hinsberger S, Werth R, Marchais-Oberwinkler S, Frotscher M, Hartmann RW.
    J Med Chem; 2010 Nov 25; 53(22):8176-86. PubMed ID: 20977238
    [Abstract] [Full Text] [Related]

  • 25. Estrone and estradiol C-16 derivatives as inhibitors of type 1 17beta-hydroxysteroid dehydrogenase.
    Poirier D, Chang HJ, Azzi A, Boivin RP, Lin SX.
    Mol Cell Endocrinol; 2006 Mar 27; 248(1-2):236-8. PubMed ID: 16337735
    [Abstract] [Full Text] [Related]

  • 26. 17beta-hydroxysteroid dehydrogenase Type 1, and not Type 12, is a target for endocrine therapy of hormone-dependent breast cancer.
    Day JM, Foster PA, Tutill HJ, Parsons MF, Newman SP, Chander SK, Allan GM, Lawrence HR, Vicker N, Potter BV, Reed MJ, Purohit A.
    Int J Cancer; 2008 May 01; 122(9):1931-40. PubMed ID: 18183589
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  • 27. A new nonestrogenic steroidal inhibitor of 17β-hydroxysteroid dehydrogenase type I blocks the estrogen-dependent breast cancer tumor growth induced by estrone.
    Ayan D, Maltais R, Roy J, Poirier D.
    Mol Cancer Ther; 2012 Oct 01; 11(10):2096-104. PubMed ID: 22914440
    [Abstract] [Full Text] [Related]

  • 28. Chemical synthesis, characterisation and biological evaluation of furanic-estradiol derivatives as inhibitors of 17β-hydroxysteroid dehydrogenase type 1.
    Farhane S, Laplante Y, Poirier D.
    Med Chem; 2011 Mar 01; 7(2):80-91. PubMed ID: 21222612
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  • 30. Design, synthesis, biological evaluation and pharmacokinetics of bis(hydroxyphenyl) substituted azoles, thiophenes, benzenes, and aza-benzenes as potent and selective nonsteroidal inhibitors of 17beta-hydroxysteroid dehydrogenase type 1 (17beta-HSD1).
    Bey E, Marchais-Oberwinkler S, Werth R, Negri M, Al-Soud YA, Kruchten P, Oster A, Frotscher M, Birk B, Hartmann RW.
    J Med Chem; 2008 Nov 13; 51(21):6725-39. PubMed ID: 18855374
    [Abstract] [Full Text] [Related]

  • 31. Chemical synthesis, characterisation and biological evaluation of lactonic-estradiol derivatives as inhibitors of 17β-hydroxysteroid dehydrogenase type 1.
    Farhane S, Fournier MA, Poirier D.
    J Steroid Biochem Mol Biol; 2013 Sep 13; 137():322-31. PubMed ID: 23685015
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  • 33. C6-(N,N-butyl-methyl-heptanamide) derivatives of estrone and estradiol as inhibitors of type 1 17beta-hydroxysteroid dehydrogenase: Chemical synthesis and biological evaluation.
    Cadot C, Laplante Y, Kamal F, Luu-The V, Poirier D.
    Bioorg Med Chem; 2007 Jan 15; 15(2):714-26. PubMed ID: 17110114
    [Abstract] [Full Text] [Related]

  • 34. Chemical Synthesis and Biological Evaluation of 3-Substituted Estrone/Estradiol Derivatives as 17β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors Acting via a Reverse Orientation of the Natural Substrate Estrone.
    Ngueta AD, Roy J, Maltais R, Poirier D.
    Molecules; 2023 Jan 07; 28(2):. PubMed ID: 36677690
    [Abstract] [Full Text] [Related]

  • 35. Novel and potent 17beta-hydroxysteroid dehydrogenase type 1 inhibitors.
    Lawrence HR, Vicker N, Allan GM, Smith A, Mahon MF, Tutill HJ, Purohit A, Reed MJ, Potter BV.
    J Med Chem; 2005 Apr 21; 48(8):2759-62. PubMed ID: 15828812
    [Abstract] [Full Text] [Related]

  • 36. Triazole ring-opening leads to the discovery of potent nonsteroidal 17β-hydroxysteroid dehydrogenase type 2 inhibitors.
    Xu K, Al-Soud YA, Wetzel M, Hartmann RW, Marchais-Oberwinkler S.
    Eur J Med Chem; 2011 Dec 21; 46(12):5978-90. PubMed ID: 22037253
    [Abstract] [Full Text] [Related]

  • 37. Mammalian lignans and genistein decrease the activities of aromatase and 17beta-hydroxysteroid dehydrogenase in MCF-7 cells.
    Brooks JD, Thompson LU.
    J Steroid Biochem Mol Biol; 2005 Apr 21; 94(5):461-7. PubMed ID: 15876411
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  • 38. Effects of Org OD14 (Livial) and its metabolites on 17 beta-hydroxysteroid dehydrogenase activity in hormone-dependent MCF-7 and T-47D breast cancer cells.
    Chetrite GS, Kloosterboer HJ, Philippe JC, Pasqualini JR.
    Anticancer Res; 1999 Apr 21; 19(1A):261-7. PubMed ID: 10226552
    [Abstract] [Full Text] [Related]

  • 39. Novel estrone mimetics with high 17beta-HSD1 inhibitory activity.
    Oster A, Klein T, Werth R, Kruchten P, Bey E, Negri M, Marchais-Oberwinkler S, Frotscher M, Hartmann RW.
    Bioorg Med Chem; 2010 May 15; 18(10):3494-505. PubMed ID: 20413314
    [Abstract] [Full Text] [Related]

  • 40. Recent insight on the control of enzymes involved in estrogen formation and transformation in human breast cancer.
    Pasqualini JR, Chetrite GS.
    J Steroid Biochem Mol Biol; 2005 Feb 15; 93(2-5):221-36. PubMed ID: 15860265
    [Abstract] [Full Text] [Related]

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