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5. NS1643 interacts around L529 of hERG to alter voltage sensor movement on the path to activation. Guo J, Cheng YM, Lees-Miller JP, Perissinotti LL, Claydon TW, Hull CM, Thouta S, Roach DE, Durdagi S, Noskov SY, Duff HJ. Biophys J; 2015 Mar 24; 108(6):1400-1413. PubMed ID: 25809253 [Abstract] [Full Text] [Related]
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9. Effects of the small molecule HERG activator NS1643 on Kv11.3 channels. Bilet A, Bauer CK. PLoS One; 2012 Aug 24; 7(11):e50886. PubMed ID: 23226420 [Abstract] [Full Text] [Related]
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15. NS1643 enhances ionic currents in a G604S-WT hERG co-expression system associated with long QT syndrome 2. Huo J, Guo X, Lu Q, Qiang H, Liu P, Bai L, Huang CL, Zhang Y, Ma A. Clin Exp Pharmacol Physiol; 2017 Nov 24; 44(11):1125-1133. PubMed ID: 28741726 [Abstract] [Full Text] [Related]
16. Extracellular potassium effects are conserved within the rat erg K+ channel family. Sturm P, Wimmers S, Schwarz JR, Bauer CK. J Physiol; 2005 Apr 15; 564(Pt 2):329-45. PubMed ID: 15705650 [Abstract] [Full Text] [Related]