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PUBMED FOR HANDHELDS

Journal Abstract Search


515 related items for PubMed ID: 18578473

  • 1. From phenothiazine to 3-phenyl-1,4-benzothiazine derivatives as inhibitors of the Staphylococcus aureus NorA multidrug efflux pump.
    Sabatini S, Kaatz GW, Rossolini GM, Brandini D, Fravolini A.
    J Med Chem; 2008 Jul 24; 51(14):4321-30. PubMed ID: 18578473
    [Abstract] [Full Text] [Related]

  • 2. Evolution from a natural flavones nucleus to obtain 2-(4-Propoxyphenyl)quinoline derivatives as potent inhibitors of the S. aureus NorA efflux pump.
    Sabatini S, Gosetto F, Manfroni G, Tabarrini O, Kaatz GW, Patel D, Cecchetti V.
    J Med Chem; 2011 Aug 25; 54(16):5722-36. PubMed ID: 21751791
    [Abstract] [Full Text] [Related]

  • 3. Re-evolution of the 2-phenylquinolines: ligand-based design, synthesis, and biological evaluation of a potent new class of Staphylococcus aureus NorA efflux pump inhibitors to combat antimicrobial resistance.
    Sabatini S, Gosetto F, Iraci N, Barreca ML, Massari S, Sancineto L, Manfroni G, Tabarrini O, Dimovska M, Kaatz GW, Cecchetti V.
    J Med Chem; 2013 Jun 27; 56(12):4975-89. PubMed ID: 23710549
    [Abstract] [Full Text] [Related]

  • 4. Piperine analogs as potent Staphylococcus aureus NorA efflux pump inhibitors.
    Sangwan PL, Koul JL, Koul S, Reddy MV, Thota N, Khan IA, Kumar A, Kalia NP, Qazi GN.
    Bioorg Med Chem; 2008 Nov 15; 16(22):9847-57. PubMed ID: 18848780
    [Abstract] [Full Text] [Related]

  • 5. Efflux-mediated response of Staphylococcus aureus exposed to ethidium bromide.
    Couto I, Costa SS, Viveiros M, Martins M, Amaral L.
    J Antimicrob Chemother; 2008 Sep 15; 62(3):504-13. PubMed ID: 18511413
    [Abstract] [Full Text] [Related]

  • 6. Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues.
    Felicetti T, Cannalire R, Burali MS, Massari S, Manfroni G, Barreca ML, Tabarrini O, Schindler BD, Sabatini S, Kaatz GW, Cecchetti V.
    ChemMedChem; 2017 Aug 22; 12(16):1293-1302. PubMed ID: 28598572
    [Abstract] [Full Text] [Related]

  • 7. Novel structural analogues of piperine as inhibitors of the NorA efflux pump of Staphylococcus aureus.
    Kumar A, Khan IA, Koul S, Koul JL, Taneja SC, Ali I, Ali F, Sharma S, Mirza ZM, Kumar M, Sangwan PL, Gupta P, Thota N, Qazi GN.
    J Antimicrob Chemother; 2008 Jun 22; 61(6):1270-6. PubMed ID: 18334493
    [Abstract] [Full Text] [Related]

  • 8. Citral derived amides as potent bacterial NorA efflux pump inhibitors.
    Thota N, Koul S, Reddy MV, Sangwan PL, Khan IA, Kumar A, Raja AF, Andotra SS, Qazi GN.
    Bioorg Med Chem; 2008 Jul 01; 16(13):6535-43. PubMed ID: 18524600
    [Abstract] [Full Text] [Related]

  • 9. Capsaicin, a novel inhibitor of the NorA efflux pump, reduces the intracellular invasion of Staphylococcus aureus.
    Kalia NP, Mahajan P, Mehra R, Nargotra A, Sharma JP, Koul S, Khan IA.
    J Antimicrob Chemother; 2012 Oct 01; 67(10):2401-8. PubMed ID: 22807321
    [Abstract] [Full Text] [Related]

  • 10. Pyrazolo[4,3-c][1,2]benzothiazines 5,5-dioxide: a promising new class of Staphylococcus aureus NorA efflux pump inhibitors.
    Sabatini S, Gosetto F, Serritella S, Manfroni G, Tabarrini O, Iraci N, Brincat JP, Carosati E, Villarini M, Kaatz GW, Cecchetti V.
    J Med Chem; 2012 Apr 12; 55(7):3568-72. PubMed ID: 22432682
    [Abstract] [Full Text] [Related]

  • 11. Substituted dihydronaphthalenes as efflux pump inhibitors of Staphylococcus aureus.
    Thota N, Reddy MV, Kumar A, Khan IA, Sangwan PL, Kalia NP, Koul JL, Koul S.
    Eur J Med Chem; 2010 Sep 12; 45(9):3607-16. PubMed ID: 20605275
    [Abstract] [Full Text] [Related]

  • 12. Chalcone inhibitors of the NorA efflux pump in Staphylococcus aureus whole cells and enriched everted membrane vesicles.
    Holler JG, Slotved HC, Mølgaard P, Olsen CE, Christensen SB.
    Bioorg Med Chem; 2012 Jul 15; 20(14):4514-21. PubMed ID: 22682300
    [Abstract] [Full Text] [Related]

  • 13. Boronic species as promising inhibitors of the Staphylococcus aureus NorA efflux pump: study of 6-substituted pyridine-3-boronic acid derivatives.
    Fontaine F, Héquet A, Voisin-Chiret AS, Bouillon A, Lesnard A, Cresteil T, Jolivalt C, Rault S.
    Eur J Med Chem; 2015 May 05; 95():185-98. PubMed ID: 25817769
    [Abstract] [Full Text] [Related]

  • 14. Synthesis of amides from (E)-3-(1-chloro-3,4-dihydronaphthalen-2-yl)acrylic acid and substituted amino acid esters as NorA efflux pump inhibitors of Staphylococcus aureus.
    Rath SK, Singh S, Kumar S, Wani NA, Rai R, Koul S, Khan IA, Sangwan PL.
    Bioorg Med Chem; 2019 Jan 15; 27(2):343-353. PubMed ID: 30552006
    [Abstract] [Full Text] [Related]

  • 15. Amino acid amides of piperic acid (PA) and 4-ethylpiperic acid (EPA) as NorA efflux pump inhibitors of Staphylococcus aureus.
    Wani NA, Singh S, Farooq S, Shankar S, Koul S, Khan IA, Rai R.
    Bioorg Med Chem Lett; 2016 Sep 01; 26(17):4174-8. PubMed ID: 27503686
    [Abstract] [Full Text] [Related]

  • 16. First identification of boronic species as novel potential inhibitors of the Staphylococcus aureus NorA efflux pump.
    Fontaine F, Hequet A, Voisin-Chiret AS, Bouillon A, Lesnard A, Cresteil T, Jolivalt C, Rault S.
    J Med Chem; 2014 Mar 27; 57(6):2536-48. PubMed ID: 24499135
    [Abstract] [Full Text] [Related]

  • 17. 1-(1H-indol-3-yl)ethanamine derivatives as potent Staphylococcus aureus NorA efflux pump inhibitors.
    Hequet A, Burchak ON, Jeanty M, Guinchard X, Le Pihive E, Maigre L, Bouhours P, Schneider D, Maurin M, Paris JM, Denis JN, Jolivalt C.
    ChemMedChem; 2014 Jul 27; 9(7):1534-45. PubMed ID: 24677763
    [Abstract] [Full Text] [Related]

  • 18. Synthesis and evaluation of new arylbenzo[b]thiophene and diarylthiophene derivatives as inhibitors of the NorA multidrug transporter of Staphylococcus aureus.
    Fournier Dit Chabert J, Marquez B, Neville L, Joucla L, Broussous S, Bouhours P, David E, Pellet-Rostaing S, Marquet B, Moreau N, Lemaire M.
    Bioorg Med Chem; 2007 Jul 01; 15(13):4482-97. PubMed ID: 17498961
    [Abstract] [Full Text] [Related]

  • 19. Synthesis of functionalized 2-aryl-5-nitro-1H-indoles and their activity as bacterial NorA efflux pump inhibitors.
    Samosorn S, Bremner JB, Ball A, Lewis K.
    Bioorg Med Chem; 2006 Feb 01; 14(3):857-65. PubMed ID: 16203150
    [Abstract] [Full Text] [Related]

  • 20. Discovery of novel inhibitors of the NorA multidrug transporter of Staphylococcus aureus.
    Brincat JP, Carosati E, Sabatini S, Manfroni G, Fravolini A, Raygada JL, Patel D, Kaatz GW, Cruciani G.
    J Med Chem; 2011 Jan 13; 54(1):354-65. PubMed ID: 21141825
    [Abstract] [Full Text] [Related]


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