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2. New synthetic routes to chain-extended selenium, sulfur, and nitrogen analogues of the naturally occurring glucosidase inhibitor salacinol and their inhibitory activities against recombinant human maltase glucoamylase. Liu H, Nasi R, Jayakanthan K, Sim L, Heipel H, Rose DR, Pinto BM. J Org Chem; 2007 Aug 17; 72(17):6562-72. PubMed ID: 17658854 [Abstract] [Full Text] [Related]
3. New chain-extended analogues of salacinol and blintol and their glycosidase inhibitory activities. Mapping the active-site requirements of human maltase glucoamylase. Nasi R, Sim L, Rose DR, Pinto BM. J Org Chem; 2007 Jan 05; 72(1):180-6. PubMed ID: 17194097 [Abstract] [Full Text] [Related]
4. Synthesis of a biologically active isomer of kotalanol, a naturally occurring glucosidase inhibitor. Eskandari R, Jayakanthan K, Kuntz DA, Rose DR, Pinto BM. Bioorg Med Chem; 2010 Apr 15; 18(8):2829-35. PubMed ID: 20363144 [Abstract] [Full Text] [Related]
5. Synthesis of analogues of salacinol containing a carboxylate inner salt and their inhibitory activities against human maltase glucoamylase. Chen W, Sim L, Rose DR, Pinto BM. Carbohydr Res; 2007 Sep 03; 342(12-13):1661-7. PubMed ID: 17597595 [Abstract] [Full Text] [Related]
6. A new class of glucosidase inhibitor: analogues of the naturally occurring glucosidase inhibitor salacinol with different ring heteroatom substituents and acyclic chain extension. Liu H, Sim L, Rose DR, Pinto BM. J Org Chem; 2006 Apr 14; 71(8):3007-13. PubMed ID: 16599595 [Abstract] [Full Text] [Related]
7. Structure proof and synthesis of kotalanol and de-O-sulfonated kotalanol, glycosidase inhibitors isolated from an herbal remedy for the treatment of type-2 diabetes. Jayakanthan K, Mohan S, Pinto BM. J Am Chem Soc; 2009 Apr 22; 131(15):5621-6. PubMed ID: 19331410 [Abstract] [Full Text] [Related]
8. Synthesis of 2-deoxy-2-fluoro and 1,2-ene derivatives of the naturally occurring glycosidase inhibitor, salacinol, and their inhibitory activities against recombinant human maltase glucoamylase. Choubdar N, Sim L, Rose DR, Pinto BM. Carbohydr Res; 2008 Apr 07; 343(5):951-6. PubMed ID: 18295754 [Abstract] [Full Text] [Related]
9. Synthesis of D-lyxitol and D-ribitol analogues of the naturally occurring glycosidase inhibitor salacinol. Kumar NS, Pinto BM. Carbohydr Res; 2005 Dec 12; 340(17):2612-9. PubMed ID: 16198322 [Abstract] [Full Text] [Related]
10. Synthesis and glycosidase inhibitory activities of chain-modified analogues of the glycosidase inhibitors salacinol and blintol. Nasi R, Sim L, Rose DR, Pinto BM. Carbohydr Res; 2007 Sep 03; 342(12-13):1888-94. PubMed ID: 17359953 [Abstract] [Full Text] [Related]
11. Synthesis and biological evaluation of heteroanalogues of kotalanol and de-O-sulfonated kotalanol. Mohan S, Jayakanthan K, Nasi R, Kuntz DA, Rose DR, Pinto BM. Org Lett; 2010 Mar 05; 12(5):1088-91. PubMed ID: 20143790 [Abstract] [Full Text] [Related]
12. Probing the active-site requirements of human intestinal N-terminal maltase-glucoamylase: Synthesis and enzyme inhibitory activities of a six-membered ring nitrogen analogue of kotalanol and its de-O-sulfonated derivative. Mohan S, Sim L, Rose DR, Pinto BM. Bioorg Med Chem; 2010 Nov 15; 18(22):7794-8. PubMed ID: 20970346 [Abstract] [Full Text] [Related]
13. Synthesis of phosphate derivatives related to the glycosidase inhibitor salacinol. Bhat RG, Kumar NS, Pinto BM. Carbohydr Res; 2007 Sep 03; 342(12-13):1934-42. PubMed ID: 17572396 [Abstract] [Full Text] [Related]
14. Synthesis, enzymatic activity, and X-ray crystallography of an unusual class of amino acids. Chen W, Kuntz DA, Hamlet T, Sim L, Rose DR, Mario Pinto B. Bioorg Med Chem; 2006 Dec 15; 14(24):8332-40. PubMed ID: 17010621 [Abstract] [Full Text] [Related]
15. Inhibition of recombinant human maltase glucoamylase by salacinol and derivatives. Rossi EJ, Sim L, Kuntz DA, Hahn D, Johnston BD, Ghavami A, Szczepina MG, Kumar NS, Sterchi EE, Nichols BL, Pinto BM, Rose DR. FEBS J; 2006 Jun 15; 273(12):2673-83. PubMed ID: 16817895 [Abstract] [Full Text] [Related]
16. Synthesis of a salacinol analogue and its alpha-glucosidase inhibitory activity. Shao Y, Osamu M, Kazuya Y, Yoshiharu M, Eriko Y, Toshie M, Genzoh T, Hisashi M, Masayuki Y, You QD. Yao Xue Xue Bao; 2006 Jul 15; 41(7):647-53. PubMed ID: 17007358 [Abstract] [Full Text] [Related]
17. Synthesis and biological evaluation of deoxy salacinols, the role of polar substituents in the side chain on the alpha-glucosidase inhibitory activity. Muraoka O, Yoshikai K, Takahashi H, Minematsu T, Lu G, Tanabe G, Wang T, Matsuda H, Yoshikawa M. Bioorg Med Chem; 2006 Jan 15; 14(2):500-9. PubMed ID: 16198577 [Abstract] [Full Text] [Related]
19. Synthesis of 2-amido, 2-amino, and 2-azido derivatives of the nitrogen analogue of the naturally occurring glycosidase inhibitor salacinol and their inhibitory activities against O-GlcNAcase and NagZ enzymes. Choubdar N, Bhat RG, Stubbs KA, Yuzwa S, Pinto BM. Carbohydr Res; 2008 Jul 21; 343(10-11):1766-77. PubMed ID: 18358456 [Abstract] [Full Text] [Related]
20. Role of the side chain stereochemistry in the α-glucosidase inhibitory activity of kotalanol, a potent natural α-glucosidase inhibitor. Xie W, Tanabe G, Matsuoka K, Amer MF, Minematsu T, Wu X, Yoshikawa M, Muraoka O. Bioorg Med Chem; 2011 Apr 01; 19(7):2252-62. PubMed ID: 21420866 [Abstract] [Full Text] [Related] Page: [Next] [New Search]