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Journal Abstract Search
209 related items for PubMed ID: 19577470
41. 2-amino-4H-3,1-benzoxazin-4-ones as inhibitors of C1r serine protease. Hays SJ, Caprathe BW, Gilmore JL, Amin N, Emmerling MR, Michael W, Nadimpalli R, Nath R, Raser KJ, Stafford D, Watson D, Wang K, Jaen JC. J Med Chem; 1998 Mar 26; 41(7):1060-7. PubMed ID: 9544206 [Abstract] [Full Text] [Related]
42. 1H-pyrrolo[2,3-b]pyridine: A new scaffold for human neutrophil elastase (HNE) inhibitors. Crocetti L, Giovannoni MP, Schepetkin IA, Quinn MT, Khlebnikov AI, Cantini N, Guerrini G, Iacovone A, Teodori E, Vergelli C. Bioorg Med Chem; 2018 Nov 15; 26(21):5583-5595. PubMed ID: 30385225 [Abstract] [Full Text] [Related]
43. Optimization of a series of multi-isoform PI3 kinase inhibitors. Perry B, Beevers R, Bennett G, Buckley G, Crabbe T, Gowers L, James L, Jenkins K, Lock C, Sabin V, Wright S. Bioorg Med Chem Lett; 2008 Oct 01; 18(19):5299-302. PubMed ID: 18774713 [Abstract] [Full Text] [Related]
44. Synthesis of diverse benzo[1,4]oxazin-3-one-based compounds using 1,5-difluoro-2,4-dinitrobenzene. Yuan Y, Liu G, Li L, Wang Z, Wang L. J Comb Chem; 2007 Oct 01; 9(1):158-70. PubMed ID: 17206844 [Abstract] [Full Text] [Related]
46. Benzoxazin-4-ones as novel, easily accessible inhibitors for rhomboid proteases. Yang J, Barniol-Xicota M, Nguyen MTN, Ticha A, Strisovsky K, Verhelst SHL. Bioorg Med Chem Lett; 2018 May 01; 28(8):1423-1427. PubMed ID: 29506958 [Abstract] [Full Text] [Related]
47. Preparation of 1-(3-aminobenzo[d]isoxazol-5-yl)-1H-pyrazolo[4,3-d]pyrimidin-7(6H)-ones as potent, selective, and efficacious inhibitors of coagulation factor Xa. Li YL, Fevig JM, Cacciola J, Buriak J, Rossi KA, Jona J, Knabb RM, Luettgen JM, Wong PC, Bai SA, Wexler RR, Lam PY. Bioorg Med Chem Lett; 2006 Oct 01; 16(19):5176-82. PubMed ID: 16870435 [Abstract] [Full Text] [Related]
50. The crystal structure of the complex of non-peptidic inhibitor of human neutrophil elastase ONO-6818 and porcine pancreatic elastase. Odagaki Y, Ohmoto K, Matsuoka S, Hamanaka N, Nakai H, Toda M, Katsuya Y. Bioorg Med Chem; 2001 Mar 01; 9(3):647-51. PubMed ID: 11310599 [Abstract] [Full Text] [Related]
54. 1-[3-Aminobenzisoxazol-5'-yl]-3-trifluoromethyl-6-[2'-(3-(R)-hydroxy-N-pyrrolidinyl)methyl-[1,1']-biphen-4-yl]-1,4,5,6-tetrahydropyrazolo-[3,4-c]-pyridin-7-one (BMS-740808) a highly potent, selective, efficacious, and orally bioavailable inhibitor of blood coagulation factor Xa. Pinto DJ, Orwat MJ, Quan ML, Han Q, Galemmo RA, Amparo E, Wells B, Ellis C, He MY, Alexander RS, Rossi KA, Smallwood A, Wong PC, Luettgen JM, Rendina AR, Knabb RM, Mersinger L, Kettner C, Bai S, He K, Wexler RR, Lam PY. Bioorg Med Chem Lett; 2006 Aug 01; 16(15):4141-7. PubMed ID: 16730984 [Abstract] [Full Text] [Related]
58. Discovery of inhibitors of the channel-activating protease prostasin (CAP1/PRSS8) utilizing structure-based design. Tully DC, Vidal A, Chatterjee AK, Williams JA, Roberts MJ, Petrassi HM, Spraggon G, Bursulaya B, Pacoma R, Shipway A, Schumacher AM, Danahay H, Harris JL. Bioorg Med Chem Lett; 2008 Nov 15; 18(22):5895-9. PubMed ID: 18752942 [Abstract] [Full Text] [Related]
59. Leucine-phenylalanine dipeptide-based N-mesyloxysuccinimides: synthesis of all four stereoisomers and their assay against serine proteases. Abell AD, Oldham MD. Bioorg Med Chem Lett; 1999 Feb 08; 9(3):497-500. PubMed ID: 10091709 [Abstract] [Full Text] [Related]