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Journal Abstract Search

163 related items for PubMed ID: 20225862

  • 1. Synthesis, antitubulin, and antiproliferative SAR of analogues of 2-methoxyestradiol-3,17-O,O-bis-sulfamate.
    Jourdan F, Leese MP, Dohle W, Hamel E, Ferrandis E, Newman SP, Purohit A, Reed MJ, Potter BV.
    J Med Chem; 2010 Apr 08; 53(7):2942-51. PubMed ID: 20225862
    [Abstract] [Full Text] [Related]

  • 2. 2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity.
    Leese MP, Leblond B, Smith A, Newman SP, Di Fiore A, De Simone G, Supuran CT, Purohit A, Reed MJ, Potter BV.
    J Med Chem; 2006 Dec 28; 49(26):7683-96. PubMed ID: 17181151
    [Abstract] [Full Text] [Related]

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  • 4. Synthesis, antiproliferative activity and inhibition of tubulin polymerization by anthracenone-based oxime derivatives.
    Surkau G, Böhm KJ, Müller K, Prinz H.
    Eur J Med Chem; 2010 Aug 28; 45(8):3354-64. PubMed ID: 20546980
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  • 6. Structure-activity relationships of C-17 cyano-substituted estratrienes as anticancer agents.
    Leese MP, Jourdan FL, Gaukroger K, Mahon MF, Newman SP, Foster PA, Stengel C, Regis-Lydi S, Ferrandis E, Di Fiore A, De Simone G, Supuran CT, Purohit A, Reed MJ, Potter BV.
    J Med Chem; 2008 Mar 13; 51(5):1295-308. PubMed ID: 18260615
    [Abstract] [Full Text] [Related]

  • 7. 3,17-disubstituted 2-alkylestra-1,3,5(10)-trien-3-ol derivatives: synthesis, in vitro and in vivo anticancer activity.
    Bubert C, Leese MP, Mahon MF, Ferrandis E, Regis-Lydi S, Kasprzyk PG, Newman SP, Ho YT, Purohit A, Reed MJ, Potter BV.
    J Med Chem; 2007 Sep 06; 50(18):4431-43. PubMed ID: 17696419
    [Abstract] [Full Text] [Related]

  • 8. Effects of C-17 heterocyclic substituents on the anticancer activity of 2-ethylestra-1,3,5(10)-triene-3-O-sulfamates: synthesis, in vitro evaluation and computational modelling.
    Jourdan F, Bubert C, Leese MP, Smith A, Ferrandis E, Regis-Lydi S, Newman SP, Purohit A, Reed MJ, Potter BV.
    Org Biomol Chem; 2008 Nov 21; 6(22):4108-19. PubMed ID: 18972041
    [Abstract] [Full Text] [Related]

  • 9. A-ring-substituted estrogen-3-O-sulfamates: potent multitargeted anticancer agents.
    Leese MP, Hejaz HA, Mahon MF, Newman SP, Purohit A, Reed MJ, Potter BV.
    J Med Chem; 2005 Aug 11; 48(16):5243-56. PubMed ID: 16078843
    [Abstract] [Full Text] [Related]

  • 10. Synthesis and biological evaluation of 2-amino-3-(3',4',5'-trimethoxybenzoyl)-5-aryl thiophenes as a new class of potent antitubulin agents.
    Romagnoli R, Baraldi PG, Pavani MG, Tabrizi MA, Preti D, Fruttarolo F, Piccagli L, Jung MK, Hamel E, Borgatti M, Gambari R.
    J Med Chem; 2006 Jun 29; 49(13):3906-15. PubMed ID: 16789746
    [Abstract] [Full Text] [Related]

  • 11. Quinazolinone-Based Anticancer Agents: Synthesis, Antiproliferative SAR, Antitubulin Activity, and Tubulin Co-crystal Structure.
    Dohle W, Jourdan FL, Menchon G, Prota AE, Foster PA, Mannion P, Hamel E, Thomas MP, Kasprzyk PG, Ferrandis E, Steinmetz MO, Leese MP, Potter BVL.
    J Med Chem; 2018 Feb 08; 61(3):1031-1044. PubMed ID: 29227648
    [Abstract] [Full Text] [Related]

  • 12. Synthesis and structure-activity profiles of A-homoestranes, the estratropones.
    Miller TA, Bulman AL, Thompson CD, Garst ME, Macdonald TL.
    J Med Chem; 1997 Nov 07; 40(23):3836-41. PubMed ID: 9371249
    [Abstract] [Full Text] [Related]

  • 13. Synthesis, antiproliferative activity and inhibition of tubulin polymerization by 1,5- and 1,8-disubstituted 10H-anthracen-9-ones bearing a 10-benzylidene or 10-(2-oxo-2-phenylethylidene) moiety.
    Nickel HC, Schmidt P, Böhm KJ, Baasner S, Müller K, Gerlach M, Unger E, Günther EG, Prinz H.
    Eur J Med Chem; 2010 Aug 07; 45(8):3420-38. PubMed ID: 20537765
    [Abstract] [Full Text] [Related]

  • 14. Synthesis of 2-substituted 17β-hydroxy/17-methylene estratrienes and their in vitro cytotoxicity in human cancer cell cultures.
    Panchapakesan G, Dhayalan V, Dhatchana Moorthy N, Saranya N, Mohanakrishnan AK.
    Steroids; 2011 Dec 11; 76(13):1491-504. PubMed ID: 21872616
    [Abstract] [Full Text] [Related]

  • 15. Design, synthesis, and biological evaluation of thiophene analogues of chalcones.
    Romagnoli R, Baraldi PG, Carrion MD, Cara CL, Cruz-Lopez O, Preti D, Tolomeo M, Grimaudo S, Di Cristina A, Zonta N, Balzarini J, Brancale A, Sarkar T, Hamel E.
    Bioorg Med Chem; 2008 May 15; 16(10):5367-76. PubMed ID: 18440234
    [Abstract] [Full Text] [Related]

  • 16. Synthesis and SAR of C12-C13-oxazoline derivatives of epothilone A.
    Pfeiffer B, Hauenstein K, Merz P, Gertsch J, Altmann KH.
    Bioorg Med Chem Lett; 2009 Jul 15; 19(14):3760-3. PubMed ID: 19433359
    [Abstract] [Full Text] [Related]

  • 17. Synthesis, cytotoxic effects and tubulin polymerization inhibition of 1,4-disubstituted 1,2,3-triazole analogs of 2-methoxyestradiol.
    Solum EJ, Vik A, Hansen TV.
    Steroids; 2014 Sep 15; 87():46-53. PubMed ID: 24923521
    [Abstract] [Full Text] [Related]

  • 18. Exploring the effect of 2,3,4-trimethoxy-phenyl moiety as a component of indolephenstatins.
    Alvarez C, Alvarez R, Corchete P, Pérez-Melero C, Peláez R, Medarde M.
    Eur J Med Chem; 2010 Feb 15; 45(2):588-97. PubMed ID: 19939521
    [Abstract] [Full Text] [Related]

  • 19. 4- and 5-aroylindoles as novel classes of potent antitubulin agents.
    Liou JP, Wu CY, Hsieh HP, Chang CY, Chen CM, Kuo CC, Chang JY.
    J Med Chem; 2007 Sep 06; 50(18):4548-52. PubMed ID: 17685504
    [Abstract] [Full Text] [Related]

  • 20. Generation of ligand-based pharmacophore model and virtual screening for identification of novel tubulin inhibitors with potent anticancer activity.
    Chiang YK, Kuo CC, Wu YS, Chen CT, Coumar MS, Wu JS, Hsieh HP, Chang CY, Jseng HY, Wu MH, Leou JS, Song JS, Chang JY, Lyu PC, Chao YS, Wu SY.
    J Med Chem; 2009 Jul 23; 52(14):4221-33. PubMed ID: 19507860
    [Abstract] [Full Text] [Related]

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