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Journal Abstract Search

268 related items for PubMed ID: 20922253

  • 1. Selective hydrophobic pocket binding observed within the carbonic anhydrase II active site accommodate different 4-substituted-ureido-benzenesulfonamides and correlate to inhibitor potency.
    Pacchiano F, Aggarwal M, Avvaru BS, Robbins AH, Scozzafava A, McKenna R, Supuran CT.
    Chem Commun (Camb); 2010 Nov 28; 46(44):8371-3. PubMed ID: 20922253
    [Abstract] [Full Text] [Related]

  • 2. Carbonic anhydrase inhibitors. The X-ray crystal structure of human isoform II in adduct with an adamantyl analogue of acetazolamide resides in a less utilized binding pocket than most hydrophobic inhibitors.
    Avvaru BS, Wagner JM, Maresca A, Scozzafava A, Robbins AH, Supuran CT, McKenna R.
    Bioorg Med Chem Lett; 2010 Aug 01; 20(15):4376-81. PubMed ID: 20605094
    [Abstract] [Full Text] [Related]

  • 3. Carbonic anhydrase inhibitors. X-ray crystal studies of the carbonic anhydrase II-trithiocarbonate adduct--an inhibitor mimicking the sulfonamide and urea binding to the enzyme.
    Temperini C, Scozzafava A, Supuran CT.
    Bioorg Med Chem Lett; 2010 Jan 15; 20(2):474-8. PubMed ID: 20005709
    [Abstract] [Full Text] [Related]

  • 4. 4-[N-(substituted 4-pyrimidinyl)amino]benzenesulfonamides as inhibitors of carbonic anhydrase isozymes I, II, VII, and XIII.
    Sūdžius J, Baranauskienė L, Golovenko D, Matulienė J, Michailovienė V, Torresan J, Jachno J, Sukackaitė R, Manakova E, Gražulis S, Tumkevičius S, Matulis D.
    Bioorg Med Chem; 2010 Nov 01; 18(21):7413-21. PubMed ID: 20889345
    [Abstract] [Full Text] [Related]

  • 5. Binding affinity of substituted ureido-benzenesulfonamide ligands to the carbonic anhydrase receptor: a theoretical study of enzyme inhibition.
    Sahu C, Sen K, Pakhira S, Mondal B, Das AK.
    J Comput Chem; 2013 Aug 15; 34(22):1907-16. PubMed ID: 23712937
    [Abstract] [Full Text] [Related]

  • 6. Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II "selective" inhibitor celecoxib.
    Di Fiore A, Pedone C, D'Ambrosio K, Scozzafava A, De Simone G, Supuran CT.
    Bioorg Med Chem Lett; 2006 Jan 15; 16(2):437-42. PubMed ID: 16290146
    [Abstract] [Full Text] [Related]

  • 7. Indapamide-like benzenesulfonamides as inhibitors of carbonic anhydrases I, II, VII, and XIII.
    Čapkauskaitė E, Baranauskienė L, Golovenko D, Manakova E, Gražulis S, Tumkevičius S, Matulis D.
    Bioorg Med Chem; 2010 Nov 01; 18(21):7357-64. PubMed ID: 20926301
    [Abstract] [Full Text] [Related]

  • 8. Carbonic anhydrase inhibitors: inhibition of cytosolic carbonic anhydrase isozymes II and VII with simple aromatic sulfonamides and some azo dyes.
    Carta F, Pothen B, Maresca A, Tiwari M, Singh V, Supuran CT.
    Chem Biol Drug Des; 2009 Aug 01; 74(2):196-202. PubMed ID: 19549076
    [Abstract] [Full Text] [Related]

  • 9. Protein crystal structures with ferrocene and ruthenocene-based enzyme inhibitors.
    Salmon AJ, Williams ML, Hofmann A, Poulsen SA.
    Chem Commun (Camb); 2012 Feb 25; 48(17):2328-30. PubMed ID: 22258283
    [Abstract] [Full Text] [Related]

  • 10. Virtual screening-driven identification of human carbonic anhydrase inhibitors incorporating an original, new pharmacophore.
    Pala N, Dallocchio R, Dessì A, Brancale A, Carta F, Ihm S, Maresca A, Sechi M, Supuran CT.
    Bioorg Med Chem Lett; 2011 Apr 15; 21(8):2515-20. PubMed ID: 21420862
    [Abstract] [Full Text] [Related]

  • 11. QSAR study on para-substituted aromatic sulfonamides as carbonic anhydrase II inhibitors using topological information indices.
    Melagraki G, Afantitis A, Sarimveis H, Igglessi-Markopoulou O, Supuran CT.
    Bioorg Med Chem; 2006 Feb 15; 14(4):1108-14. PubMed ID: 16213737
    [Abstract] [Full Text] [Related]

  • 12. Carbonic anhydrase inhibitors: X-ray crystallographic studies for the binding of N-substituted benzenesulfonamides to human isoform II.
    Di Fiore A, Maresca A, Alterio V, Supuran CT, De Simone G.
    Chem Commun (Camb); 2011 Nov 14; 47(42):11636-8. PubMed ID: 21952494
    [Abstract] [Full Text] [Related]

  • 13. Synthesis of different thio-scaffolds bearing sulfonamide with subnanomolar carbonic anhydrase II and IX inhibitory properties and X-ray investigations for their inhibitory mechanism.
    Angeli A, Tanini D, Capperucci A, Malevolti G, Turco F, Ferraroni M, Supuran CT.
    Bioorg Chem; 2018 Dec 14; 81():642-648. PubMed ID: 30253337
    [Abstract] [Full Text] [Related]

  • 14. Inhibition of β-carbonic anhydrases with ureido-substituted benzenesulfonamides.
    Pacchiano F, Carta F, Vullo D, Scozzafava A, Supuran CT.
    Bioorg Med Chem Lett; 2011 Jan 01; 21(1):102-5. PubMed ID: 21145236
    [Abstract] [Full Text] [Related]

  • 15. Carbonic anhydrase inhibitors: binding of indanesulfonamides to the human isoform II.
    D'Ambrosio K, Masereel B, Thiry A, Scozzafava A, Supuran CT, De Simone G.
    ChemMedChem; 2008 Mar 01; 3(3):473-7. PubMed ID: 18161740
    [Abstract] [Full Text] [Related]

  • 16. Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II.
    Di Fiore A, De Simone G, Menchise V, Pedone C, Casini A, Scozzafava A, Supuran CT.
    Bioorg Med Chem Lett; 2005 Apr 01; 15(7):1937-42. PubMed ID: 15780637
    [Abstract] [Full Text] [Related]

  • 17. Anticonvulsant 4-aminobenzenesulfonamide derivatives with branched-alkylamide moieties: X-ray crystallography and inhibition studies of human carbonic anhydrase isoforms I, II, VII, and XIV.
    Hen N, Bialer M, Yagen B, Maresca A, Aggarwal M, Robbins AH, McKenna R, Scozzafava A, Supuran CT.
    J Med Chem; 2011 Jun 09; 54(11):3977-81. PubMed ID: 21506569
    [Abstract] [Full Text] [Related]

  • 18. Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies.
    De Simone G, Di Fiore A, Menchise V, Pedone C, Antel J, Casini A, Scozzafava A, Wurl M, Supuran CT.
    Bioorg Med Chem Lett; 2005 May 02; 15(9):2315-20. PubMed ID: 15837316
    [Abstract] [Full Text] [Related]

  • 19. Carbonic anhydrase II-induced selection of inhibitors from a dynamic combinatorial library of Schiff's bases.
    Nasr G, Petit E, Supuran CT, Winum JY, Barboiu M.
    Bioorg Med Chem Lett; 2009 Nov 01; 19(21):6014-7. PubMed ID: 19796939
    [Abstract] [Full Text] [Related]

  • 20. QSAR studies on benzene sulfonamide carbonic anhydrase inhibitors: need of hydrophobic parameter for topological modeling of binding constants of sulfonamides to human CA-II.
    Khadikar PV, Sharma V, Karmarkar S, Supuran CT.
    Bioorg Med Chem Lett; 2005 Feb 15; 15(4):923-30. PubMed ID: 15686888
    [Abstract] [Full Text] [Related]

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