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4. Conformational restriction of the phenylalanine residue in a cyclic opioid peptide analogue: effects on receptor selectivity and stereospecificity. Schiller PW, Weltrowska G, Nguyen TM, Lemieux C, Chung NN, Marsden BJ, Wilkes BC. J Med Chem; 1991 Oct; 34(10):3125-32. PubMed ID: 1656045 [Abstract] [Full Text] [Related]
5. Conformational features responsible for the binding of cyclic analogues of enkephalin to opioid receptors. III. Probable binding conformations of mu-agonists with phenylalanine in position 3. Shenderovich MD, Nikiforovich GV, Golbraikh AA. Int J Pept Protein Res; 1991 Apr; 37(4):241-51. PubMed ID: 1654306 [Abstract] [Full Text] [Related]
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10. Substitution of aromatic and nonaromatic amino acids for the Phe3 residue in the delta-selective opioid peptide deltorphin I: effects on binding affinity and selectivity. Heyl DL, Schmitter SJ, Bouzit H, Johnson TW, Hepp AM, Kurtz KR, Mousigian C. Int J Pept Protein Res; 1994 Nov; 44(5):420-6. PubMed ID: 7896499 [Abstract] [Full Text] [Related]
11. Design and synthesis of conformationally constrained somatostatin analogues with high potency and specificity for mu opioid receptors. Pelton JT, Kazmierski W, Gulya K, Yamamura HI, Hruby VJ. J Med Chem; 1986 Nov; 29(11):2370-5. PubMed ID: 2878079 [Abstract] [Full Text] [Related]
12. Dermenkephalin (Tyr-D-Met-Phe-His-Leu-Met-Asp-NH2): a potent and fully specific agonist for the delta opioid receptor. Amiche M, Sagan S, Mor A, Delfour A, Nicolas P. Mol Pharmacol; 1989 Jun; 35(6):774-9. PubMed ID: 2543911 [Abstract] [Full Text] [Related]
13. Dermenkephalin and deltorphin I reveal similarities within ligand-binding domains of mu- and delta-opioid receptors and an additional address subsite on the delta-receptor. Charpentier S, Sagan S, Delfour A, Nicolas P. Biochem Biophys Res Commun; 1991 Sep 30; 179(3):1161-8. PubMed ID: 1656944 [Abstract] [Full Text] [Related]
14. Examination of the conformational meaning of "delta-address" in the dermenkephalin sequence. Nikiforovich GV, Hruby VJ. Biochem Biophys Res Commun; 1990 Dec 14; 173(2):521-7. PubMed ID: 1979733 [Abstract] [Full Text] [Related]
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16. Design and synthesis of somatostatin analogues with topographical properties that lead to highly potent and specific mu opioid receptor antagonists with greatly reduced binding at somatostatin receptors. Kazmierski W, Wire WS, Lui GK, Knapp RJ, Shook JE, Burks TF, Yamamura HI, Hruby VJ. J Med Chem; 1988 Nov 09; 31(11):2170-7. PubMed ID: 2903246 [Abstract] [Full Text] [Related]
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18. Solution conformation of mu-selective dermorphin and delta-selective deltorphin-I in phospholipid micelles, studied by NMR spectroscopy and molecular dynamics simulations. Segawa M, Ohno Y, Doi M, Ishida T, Iwashita T. Int J Pept Protein Res; 1995 Jul 09; 46(1):37-46. PubMed ID: 7558595 [Abstract] [Full Text] [Related]
19. Comparative conformational analyses of mu-selective dermorphin and delta-selective deltorphin-II in aqueous solution by 1H-NMR spectroscopy. Segawa M, Ohno Y, Doi M, Inoue M, Ishida T, Iwashita T. Int J Pept Protein Res; 1994 Sep 09; 44(3):295-304. PubMed ID: 7822107 [Abstract] [Full Text] [Related]
20. Molecular determinants of receptor affinity and selectivity of the natural delta-opioid agonist, dermenkephalin. Sagan S, Amiche M, Delfour A, Mor A, Camus A, Nicolas P. J Biol Chem; 1989 Oct 15; 264(29):17100-6. PubMed ID: 2551895 [Abstract] [Full Text] [Related] Page: [Next] [New Search]