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Journal Abstract Search

171 related items for PubMed ID: 22337204

  • 21. The effect of substitution patterns on the release rates of opioid peptides DADLE and [Leu(5)]-enkephalin from coumarin prodrug moieties.
    Zych LA, Yang W, Liao Y, Griffin KR, Wang B.
    Bioorg Chem; 2004 Apr; 32(2):109-23. PubMed ID: 14990309
    [Abstract] [Full Text] [Related]

  • 22. Characterization of the efflux transporter(s) responsible for restricting intestinal mucosa permeation of the coumarinic acid-based cyclic prodrug of the opioid peptide DADLE.
    Tang F, Borchardt RT.
    Pharm Res; 2002 Jun; 19(6):787-93. PubMed ID: 12134948
    [Abstract] [Full Text] [Related]

  • 23. A modified coumarinic acid-based cyclic prodrug of an opioid peptide: its enzymatic and chemical stability and cell permeation characteristics.
    Ouyang H, Tang F, Siahaan TJ, Borchardt RT.
    Pharm Res; 2002 Jun; 19(6):794-801. PubMed ID: 12134949
    [Abstract] [Full Text] [Related]

  • 24. Stereoselective evasion of P-glycoprotein, cytochrome P450 3A, and hydrolases by peptide prodrug modification of saquinavir.
    Wang Z, Pal D, Mitra AK.
    J Pharm Sci; 2012 Sep; 101(9):3199-213. PubMed ID: 22611042
    [Abstract] [Full Text] [Related]

  • 25. Characterization of the efflux transporter(s) responsible for restricting intestinal mucosa permeation of an acyloxyalkoxy-based cyclic prodrug of the opioid peptide DADLE.
    Tang F, Borchardt RT.
    Pharm Res; 2002 Jun; 19(6):780-6. PubMed ID: 12134947
    [Abstract] [Full Text] [Related]

  • 26. Esterase-sensitive cyclic prodrugs of peptides: evaluation of an acyloxyalkoxy promoiety in a model hexapeptide.
    Pauletti GM, Gangwar S, Okumu FW, Siahaan TJ, Stella VJ, Borchardt RT.
    Pharm Res; 1996 Nov; 13(11):1615-23. PubMed ID: 8956324
    [Abstract] [Full Text] [Related]

  • 27. Esterase-sensitive cyclic prodrugs of peptides: evaluation of a phenylpropionic acid promoiety in a model hexapeptide.
    Pauletti GM, Gangwar S, Wang B, Borchardt RT.
    Pharm Res; 1997 Jan; 14(1):11-7. PubMed ID: 9034215
    [Abstract] [Full Text] [Related]

  • 28. Synthesis and evaluation of novel coumarin-based esterase-sensitive cyclic prodrugs of peptidomimetic RGD analogs with improved membrane permeability.
    Wang B, Wang W, Camenisch GP, Elmo J, Zhang H, Borchardt RT.
    Chem Pharm Bull (Tokyo); 1999 Jan; 47(1):90-5. PubMed ID: 9987829
    [Abstract] [Full Text] [Related]

  • 29. Physiological models are good tools to predict rat bioavailability of EF5154 prodrugs from in vitro intestinal parameters.
    Nomoto M, Tatebayashi T, Morita J, Suzuki H, Aizawa K, Kurosawa T, Komiya I.
    J Pharm Sci; 2009 Apr; 98(4):1532-44. PubMed ID: 18683862
    [Abstract] [Full Text] [Related]

  • 30. A comparison of the bioconversion rates and the Caco-2 cell permeation characteristics of coumarin-based cyclic prodrugs and methylester-based linear prodrugs of RGD peptidomimetics.
    Camenisch GP, Wang W, Wang B, Borchardt RT.
    Pharm Res; 1998 Aug; 15(8):1174-81. PubMed ID: 9706046
    [Abstract] [Full Text] [Related]

  • 31. Propylene glycol-linked amino acid/dipeptide diester prodrugs of oleanolic acid for PepT1-mediated transport: synthesis, intestinal permeability, and pharmacokinetics.
    Cao F, Gao Y, Wang M, Fang L, Ping Q.
    Mol Pharm; 2013 Apr 01; 10(4):1378-87. PubMed ID: 23339520
    [Abstract] [Full Text] [Related]

  • 32. Bifunctional peptidomimetic prodrugs of didanosine for improved intestinal permeability and enhanced acidic stability: synthesis, transepithelial transport, chemical stability and pharmacokinetics.
    Yan Z, Sun J, Chang Y, Liu Y, Fu Q, Xu Y, Sun Y, Pu X, Zhang Y, Jing Y, Yin S, Zhu M, Wang Y, He Z.
    Mol Pharm; 2011 Apr 04; 8(2):319-29. PubMed ID: 21280612
    [Abstract] [Full Text] [Related]

  • 33. Comparison of permeation enhancing strategies for an oral factor Xa inhibitor using the Caco-2 cell monolayer model.
    Bruesewitz C, Funke A, Kuhland U, Wagner T, Lipp R.
    Eur J Pharm Biopharm; 2006 Oct 04; 64(2):229-37. PubMed ID: 16904877
    [Abstract] [Full Text] [Related]

  • 34. Syntheses of cyclic prodrugs of RGD peptidomimetics with various macrocyclic ring sizes: evaluation of physicochemical, transport and antithrombic properties.
    He HT, Xu CR, Song X, Siahaan TJ.
    J Pept Res; 2003 Jun 04; 61(6):331-42. PubMed ID: 12753380
    [Abstract] [Full Text] [Related]

  • 35. Oxidative activation of acylguanidine prodrugs: intestinal presystemic activation in rats limits absorption and can be inhibited by co-administration of ketoconazole.
    Humphreys WG, Obermeier MT, Chong S, Kimball SD, Das J, Chen P, Moquin R, Han WC, Gedamke R, White RE, Morrison RA.
    Xenobiotica; 2003 Jan 04; 33(1):93-106. PubMed ID: 12519697
    [Abstract] [Full Text] [Related]

  • 36. Enhancing the intestinal membrane permeability of zanamivir: a carrier mediated prodrug approach.
    Gupta SV, Gupta D, Sun J, Dahan A, Tsume Y, Hilfinger J, Lee KD, Amidon GL.
    Mol Pharm; 2011 Dec 05; 8(6):2358-67. PubMed ID: 21905667
    [Abstract] [Full Text] [Related]

  • 37. Ester prodrugs of morphine improve transdermal drug delivery: a mechanistic study.
    Wang JJ, Sung KC, Huang JF, Yeh CH, Fang JY.
    J Pharm Pharmacol; 2007 Jul 05; 59(7):917-25. PubMed ID: 17637185
    [Abstract] [Full Text] [Related]

  • 38.
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  • 39. Lipophilic derivatives of leu-enkephalinamide: in vitro permeability, stability and in vivo nasal delivery.
    Cros CD, Toth I, Blanchfield JT.
    Bioorg Med Chem; 2011 Feb 15; 19(4):1528-34. PubMed ID: 21273080
    [Abstract] [Full Text] [Related]

  • 40. Effect of intestinal first-pass hydrolysis on the oral bioavailability of an ester prodrug of fexofenadine.
    Ohura K, Soejima T, Nogata R, Adachi Y, Ninomiya S, Imai T.
    J Pharm Sci; 2012 Sep 15; 101(9):3264-74. PubMed ID: 22628163
    [Abstract] [Full Text] [Related]

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