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112 related items for PubMed ID: 22372816

  • 1. Fluorophosphonylated nucleoside derivatives as new series of thymidine phosphorylase multisubstrate inhibitors.
    Diab SA, De Schutter C, Muzard M, Plantier-Royon R, Pfund E, Lequeux T.
    J Med Chem; 2012 Mar 22; 55(6):2758-68. PubMed ID: 22372816
    [Abstract] [Full Text] [Related]

  • 2. Novel multisubstrate inhibitors of mammalian purine nucleoside phosphorylase.
    Toms AV, Wang W, Li Y, Ganem B, Ealick SE.
    Acta Crystallogr D Biol Crystallogr; 2005 Nov 22; 61(Pt 11):1449-58. PubMed ID: 16239721
    [Abstract] [Full Text] [Related]

  • 3. Inhibition of human thymidine phosphorylase by conformationally constrained pyrimidine nucleoside phosphonic acids and their "open-structure" isosteres.
    Košiová I, Šimák O, Panova N, Buděšínský M, Petrová M, Rejman D, Liboska R, Páv O, Rosenberg I.
    Eur J Med Chem; 2014 Mar 03; 74():145-68. PubMed ID: 24462848
    [Abstract] [Full Text] [Related]

  • 4. Nucleoside phosphonic acids in thymidine phosphorylase inhibition: structure-activity relationship.
    Panova N, Kosiová I, Petrová M, Vanĕk V, Liboska R, Kovacková S, Kocalka P, Králíková S, Tocík Z, Páv O, Paces O, Rejman D, Rosenberg I.
    Nucleic Acids Symp Ser (Oxf); 2008 Mar 03; (52):665-6. PubMed ID: 18776555
    [Abstract] [Full Text] [Related]

  • 5. Syntheses of pyrimidine acyclic nucleoside phosphonates as potent inhibitors of thymidine phosphorylase (PD-ECGF) from SD-lymphoma.
    Pomeisl K, Votruba I, Holý A, Pohl R.
    Nucleosides Nucleotides Nucleic Acids; 2007 Mar 03; 26(8-9):1025-8. PubMed ID: 18058530
    [Abstract] [Full Text] [Related]

  • 6. Synthesis and evaluation of multisubstrate bicyclic pyrimidine nucleoside inhibitors of human thymidine phosphorylase.
    Allan AL, Gladstone PL, Price ML, Hopkins SA, Juarez JC, Doñate F, Ternansky RJ, Shaw DE, Ganem B, Li Y, Wang W, Ealick S.
    J Med Chem; 2006 Dec 28; 49(26):7807-15. PubMed ID: 17181163
    [Abstract] [Full Text] [Related]

  • 7. Kinetic analysis of novel multisubstrate analogue inhibitors of thymidine phosphorylase.
    Balzarini J, Degrève B, Esteban-Gamboa A, Esnouf R, De Clercq E, Engelborghs Y, Camarasa MJ, Pérez-Pérez MJ.
    FEBS Lett; 2000 Oct 20; 483(2-3):181-5. PubMed ID: 11042277
    [Abstract] [Full Text] [Related]

  • 8. Synthesis of a new family of acyclic nucleoside phosphonates, analogues of TPases transition states.
    Dayde B, Benzaria S, Pierra C, Gosselin G, Surleraux D, Volle JN, Pirat JL, Virieux D.
    Org Biomol Chem; 2012 May 07; 10(17):3448-54. PubMed ID: 22434259
    [Abstract] [Full Text] [Related]

  • 9. Structural diversity of nucleoside phosphonic acids as a key factor in the discovery of potent inhibitors of rat T-cell lymphoma thymidine phosphorylase.
    Kocalka P, Rejman D, Vanek V, Rinnová M, Tomecková I, Králíková S, Petrová M, Páv O, Pohl R, Budesínský M, Liboska R, Tocík Z, Panova N, Votruba I, Rosenberg I.
    Bioorg Med Chem Lett; 2010 Feb 01; 20(3):862-5. PubMed ID: 20053558
    [Abstract] [Full Text] [Related]

  • 10. 5'-O-tritylated nucleoside derivatives: inhibition of thymidine phosphorylase and angiogenesis.
    Liekens S, Bronckaers A, Hernández AI, Priego EM, Casanova E, Camarasa MJ, Pérez-Pérez MJ, Balzarini J.
    Mol Pharmacol; 2006 Aug 01; 70(2):501-9. PubMed ID: 16675660
    [Abstract] [Full Text] [Related]

  • 11. Design, synthesis, and enzymatic evaluation of multisubstrate analogue inhibitors of Escherichia coli thymidine phosphorylase.
    Esteban-Gamboa A, Balzarini J, Esnouf R, De Clercq E, Camarasa MJ, Pérez-Pérez MJ.
    J Med Chem; 2000 Mar 09; 43(5):971-83. PubMed ID: 10715161
    [Abstract] [Full Text] [Related]

  • 12. 5'-O-tritylinosine and analogues as allosteric inhibitors of human thymidine phosphorylase.
    Casanova E, Hernandez AI, Priego EM, Liekens S, Camarasa MJ, Balzarini J, Pérez-Pérez MJ.
    J Med Chem; 2006 Sep 07; 49(18):5562-70. PubMed ID: 16942029
    [Abstract] [Full Text] [Related]

  • 13. Syntheses of N3-substituted thymine acyclic nucleoside phosphonates and a comparison of their inhibitory effect towards thymidine phosphorylase.
    Pomeisl K, Holý A, Votruba I, Pohl R.
    Bioorg Med Chem Lett; 2008 Feb 15; 18(4):1364-7. PubMed ID: 18221873
    [Abstract] [Full Text] [Related]

  • 14. The nucleoside derivative 5'-O-trityl-inosine (KIN59) suppresses thymidine phosphorylase-triggered angiogenesis via a noncompetitive mechanism of action.
    Liekens S, Hernández AI, Ribatti D, De Clercq E, Camarasa MJ, Pérez-Pérez MJ, Balzarini J.
    J Biol Chem; 2004 Jul 09; 279(28):29598-605. PubMed ID: 15123637
    [Abstract] [Full Text] [Related]

  • 15. Novel antiviral C5-substituted pyrimidine acyclic nucleoside phosphonates selected as human thymidylate kinase substrates.
    Topalis D, Pradère U, Roy V, Caillat C, Azzouzi A, Broggi J, Snoeck R, Andrei G, Lin J, Eriksson S, Alexandre JA, El-Amri C, Deville-Bonne D, Meyer P, Balzarini J, Agrofoglio LA.
    J Med Chem; 2011 Jan 13; 54(1):222-32. PubMed ID: 21128666
    [Abstract] [Full Text] [Related]

  • 16. Syntheses of 1-[2-(Phosphonomethoxy)Alkyl] thymine monophosphates and an evaluation of their inhibitory activity toward human thymidine phosphorylase.
    Pomeisl K, Horská K, Pohl R, Blažek J, Krečmerová M.
    Nucleosides Nucleotides Nucleic Acids; 2012 Jan 13; 31(3):159-71. PubMed ID: 22356232
    [Abstract] [Full Text] [Related]

  • 17. Pyrimidine acyclic nucleoside phosphonates and phosphorylated analogs. Part 2. Syntheses and investigation of their inhibitory effects towards human thymidine phosphorylase.
    Pomeisl K, Holý A, Votruba I.
    Nucleic Acids Symp Ser (Oxf); 2008 Jan 13; (52):657-8. PubMed ID: 18776551
    [Abstract] [Full Text] [Related]

  • 18. Discovery of 5-substituted-6-chlorouracils as efficient inhibitors of human thymidine phosphorylase.
    Nencka R, Votruba I, Hrebabecký H, Jansa P, Tloust'ová E, Horská K, Masojídková M, Holý A.
    J Med Chem; 2007 Nov 29; 50(24):6016-23. PubMed ID: 17963370
    [Abstract] [Full Text] [Related]

  • 19. Substrate specificity of Escherichia coli thymidine phosphorylase.
    Panova NG, Alexeev CS, Kuzmichov AS, Shcheveleva EV, Gavryushov SA, Polyakov KM, Kritzyn AM, Mikhailov SN, Esipov RS, Miroshnikov AI.
    Biochemistry (Mosc); 2007 Jan 29; 72(1):21-8. PubMed ID: 17309433
    [Abstract] [Full Text] [Related]

  • 20. Synthesis, anti-HIV activity, and resistance profiles of ribose modified nucleoside phosphonates.
    Mackman RL, Boojamra CG, Prasad V, Zhang L, Lin KY, Petrakovsky O, Babusis D, Chen J, Douglas J, Grant D, Hui HC, Kim CU, Markevitch DY, Vela J, Ray A, Cihlar T.
    Bioorg Med Chem Lett; 2007 Dec 15; 17(24):6785-9. PubMed ID: 18029175
    [Abstract] [Full Text] [Related]

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