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Journal Abstract Search

134 related items for PubMed ID: 23953070

  • 1. Discovery of potent and selective nonsteroidal indazolyl amide glucocorticoid receptor agonists.
    Sheppeck JE, Gilmore JL, Xiao HY, Dhar TG, Nirschl D, Doweyko AM, Sack JS, Corbett MJ, Malley MF, Gougoutas JZ, Mckay L, Cunningham MD, Habte SF, Dodd JH, Nadler SG, Somerville JE, Barrish JC.
    Bioorg Med Chem Lett; 2013 Oct 01; 23(19):5442-7. PubMed ID: 23953070
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  • 2. Synthesis and structure-activity relationships of novel indazolyl glucocorticoid receptor partial agonists.
    Gilmore JL, Sheppeck JE, Wang J, Dhar TG, Cavallaro C, Doweyko AM, Mckay L, Cunningham MD, Habte SF, Nadler SG, Dodd JH, Somerville JE, Barrish JC.
    Bioorg Med Chem Lett; 2013 Oct 01; 23(19):5448-51. PubMed ID: 23916594
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  • 3. Substituted phenyl as a steroid A-ring mimetic: providing agonist activity to a class of arylsulfonamide nonsteroidal glucocorticoid ligands.
    DiSalvo D, Kuzmich D, Bentzien J, Regan J, Kukulka A, Fadra-Khan T, Nelson R, Harcken C, Thomson D, Nabozny G.
    Bioorg Med Chem Lett; 2013 Dec 15; 23(24):6645-9. PubMed ID: 24239189
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  • 4. Discovery of a potent series of non-steroidal non α-trifluoromethyl carbinol glucocorticoid receptor agonists with reduced lipophilicity.
    Diallo H, Angell DC, Barnett HA, Biggadike K, Coe DM, Cooper TW, Craven A, Gray JR, House D, Jack TI, Keeling SP, Macdonald SJ, McLay IM, Oliver S, Taylor SJ, Uings IJ, Wellaway N.
    Bioorg Med Chem Lett; 2011 Feb 15; 21(4):1126-33. PubMed ID: 21257309
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  • 5. Structure guided design of 5-arylindazole glucocorticoid receptor agonists and antagonists.
    Yates CM, Brown PJ, Stewart EL, Patten C, Austin RJ, Holt JA, Maglich JM, Angell DC, Sasse RZ, Taylor SJ, Uings IJ, Trump RP.
    J Med Chem; 2010 Jun 10; 53(11):4531-44. PubMed ID: 20469868
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  • 6. Non-steroidal glucocorticoid agonists: the discovery of aryl pyrazoles as A-ring mimetics.
    Clackers M, Coe DM, Demaine DA, Hardy GW, Humphreys D, Inglis GG, Johnston MJ, Jones HT, House D, Loiseau R, Minick DJ, Skone PA, Uings I, McLay IM, Macdonald SJ.
    Bioorg Med Chem Lett; 2007 Sep 01; 17(17):4737-45. PubMed ID: 17616395
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  • 9. The first X-ray crystal structure of the glucocorticoid receptor bound to a non-steroidal agonist.
    Madauss KP, Bledsoe RK, Mclay I, Stewart EL, Uings IJ, Weingarten G, Williams SP.
    Bioorg Med Chem Lett; 2008 Dec 01; 18(23):6097-9. PubMed ID: 18952422
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  • 10. Discovery of inhibitors of the mitotic kinase TTK based on N-(3-(3-sulfamoylphenyl)-1H-indazol-5-yl)-acetamides and carboxamides.
    Laufer R, Ng G, Liu Y, Patel NK, Edwards LG, Lang Y, Li SW, Feher M, Awrey DE, Leung G, Beletskaya I, Plotnikova O, Mason JM, Hodgson R, Wei X, Mao G, Luo X, Huang P, Green E, Kiarash R, Lin DC, Harris-Brandts M, Ban F, Nadeem V, Mak TW, Pan GJ, Qiu W, Chirgadze NY, Pauls HW.
    Bioorg Med Chem; 2014 Sep 01; 22(17):4968-97. PubMed ID: 25043312
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  • 11. Discovery and optimization of indazoles as potent and selective interleukin-2 inducible T cell kinase (ITK) inhibitors.
    Pastor RM, Burch JD, Magnuson S, Ortwine DF, Chen Y, De La Torre K, Ding X, Eigenbrot C, Johnson A, Liimatta M, Liu Y, Shia S, Wang X, Wu LC, Pei Z.
    Bioorg Med Chem Lett; 2014 Jun 01; 24(11):2448-52. PubMed ID: 24767842
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  • 12. Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor.
    Biggadike K, Bledsoe RK, Coe DM, Cooper TW, House D, Iannone MA, Macdonald SJ, Madauss KP, McLay IM, Shipley TJ, Taylor SJ, Tran TB, Uings IJ, Weller V, Williams SP.
    Proc Natl Acad Sci U S A; 2009 Oct 27; 106(43):18114-9. PubMed ID: 19822747
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  • 13. Discovery and SAR study of novel dihydroquinoline-containing glucocorticoid receptor agonists.
    Takahashi H, Bekkali Y, Capolino AJ, Gilmore T, Goldrick SE, Kaplita PV, Liu L, Nelson RM, Terenzio D, Wang J, Zuvela-Jelaska L, Proudfoot J, Nabozny G, Thomson D.
    Bioorg Med Chem Lett; 2007 Sep 15; 17(18):5091-5. PubMed ID: 17681466
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  • 17. Discovery of acylurea isosteres of 2-acylaminothiadiazole in the azaxanthene series of glucocorticoid receptor agonists.
    Gong H, Yang M, Xiao Z, Doweyko AM, Cunningham M, Wang J, Habte S, Holloway D, Burke C, Shuster D, Gao L, Carman J, Somerville JE, Nadler SG, Salter-Cid L, Barrish JC, Weinstein DS.
    Bioorg Med Chem Lett; 2014 Aug 01; 24(15):3268-73. PubMed ID: 24980053
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  • 19. Synthesis of novel steroidal agonists, partial agonists, and antagonists for the glucocorticoid receptor.
    Jin Z, Lin H, Srinivasan S, Nwachukwu JC, Bruno N, Griffin PR, Nettles KW, Kamenecka TM.
    Bioorg Med Chem Lett; 2017 Jan 15; 27(2):347-353. PubMed ID: 27919657
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