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Journal Abstract Search

117 related items for PubMed ID: 24471437

  • 1. Synthesis, structure-activity relationships and brain uptake of a novel series of benzopyran inhibitors of insulin-regulated aminopeptidase.
    Mountford SJ, Albiston AL, Charman WN, Ng L, Holien JK, Parker MW, Nicolazzo JA, Thompson PE, Chai SY.
    J Med Chem; 2014 Feb 27; 57(4):1368-77. PubMed ID: 24471437
    [Abstract] [Full Text] [Related]

  • 2. Identification and characterization of a new cognitive enhancer based on inhibition of insulin-regulated aminopeptidase.
    Albiston AL, Morton CJ, Ng HL, Pham V, Yeatman HR, Ye S, Fernando RN, De Bundel D, Ascher DB, Mendelsohn FA, Parker MW, Chai SY.
    FASEB J; 2008 Dec 27; 22(12):4209-17. PubMed ID: 18716029
    [Abstract] [Full Text] [Related]

  • 3. Synthesis and structure-activity relationships of dehydroaltenusin derivatives as selective DNA polymerase alpha inhibitors.
    Kuramochi K, Fukudome K, Kuriyama I, Takeuchi T, Sato Y, Kamisuki S, Tsubaki K, Sugawara F, Yoshida H, Mizushina Y.
    Bioorg Med Chem; 2009 Oct 15; 17(20):7227-38. PubMed ID: 19767211
    [Abstract] [Full Text] [Related]

  • 4. Synthesis, pharmacological evaluation, and structure-activity relationships of benzopyran derivatives with potent SERM activity.
    Amari G, Armani E, Ghirardi S, Delcanale M, Civelli M, Caruso PL, Galbiati E, Lipreri M, Rivara S, Lodola A, Mor M.
    Bioorg Med Chem; 2004 Jul 15; 12(14):3763-82. PubMed ID: 15210143
    [Abstract] [Full Text] [Related]

  • 5. Structure-based parallel medicinal chemistry approach to improve metabolic stability of benzopyran COX-2 inhibitors.
    Xing L, Hamper BC, Fletcher TR, Wendling JM, Carter J, Gierse JK, Liao S.
    Bioorg Med Chem Lett; 2011 Feb 01; 21(3):993-6. PubMed ID: 21215625
    [Abstract] [Full Text] [Related]

  • 6. Phenylalanine-544 plays a key role in substrate and inhibitor binding by providing a hydrophobic packing point at the active site of insulin-regulated aminopeptidase.
    Albiston AL, Pham V, Ye S, Ng L, Lew RA, Thompson PE, Holien JK, Morton CJ, Parker MW, Chai SY.
    Mol Pharmacol; 2010 Oct 01; 78(4):600-7. PubMed ID: 20628006
    [Abstract] [Full Text] [Related]

  • 7. Novel selective inhibitors of aminopeptidases that generate antigenic peptides.
    Papakyriakou A, Zervoudi E, Theodorakis EA, Saveanu L, Stratikos E, Vourloumis D.
    Bioorg Med Chem Lett; 2013 Sep 01; 23(17):4832-6. PubMed ID: 23916253
    [Abstract] [Full Text] [Related]

  • 8. Synthesis and structure activity relationships of novel non-peptidic metallo-aminopeptidase inhibitors.
    Albrecht S, Defoin A, Salomon E, Tarnus C, Wetterholm A, Haeggström JZ.
    Bioorg Med Chem; 2006 Nov 01; 14(21):7241-57. PubMed ID: 16844380
    [Abstract] [Full Text] [Related]

  • 9. Beta-homo-amino acid scan of angiotensin IV.
    Lukaszuk A, Demaegdt H, Szemenyei E, Tóth G, Tymecka D, Misicka A, Karoyan P, Vanderheyden P, Vauquelin G, Tourwé D.
    J Med Chem; 2008 Apr 10; 51(7):2291-6. PubMed ID: 18386881
    [Abstract] [Full Text] [Related]

  • 10. 1-Benzopyran-4-one antioxidants as aldose reductase inhibitors.
    Costantino L, Rastelli G, Gamberini MC, Vinson JA, Bose P, Iannone A, Staffieri M, Antolini L, Del Corso A, Mura U, Albasini A.
    J Med Chem; 1999 Jun 03; 42(11):1881-93. PubMed ID: 10354396
    [Abstract] [Full Text] [Related]

  • 11. Rapid and efficient synthesis of a novel series of substituted aminobenzosuberone derivatives as potent, selective, non-peptidic neutral aminopeptidase inhibitors.
    Albrecht S, Salomon E, Defoin A, Tarnus C.
    Bioorg Med Chem; 2012 Aug 15; 20(16):4942-53. PubMed ID: 22796349
    [Abstract] [Full Text] [Related]

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  • 13. Protein kinase C-zeta phosphorylates insulin-responsive aminopeptidase in vitro at Ser-80 and Ser-91.
    Ryu J, Hah JS, Park JS, Lee W, Rampal AL, Jung CY.
    Arch Biochem Biophys; 2002 Jul 01; 403(1):71-82. PubMed ID: 12061804
    [Abstract] [Full Text] [Related]

  • 14. Structure-activity study of LVV-hemorphin-7: angiotensin AT4 receptor ligand and inhibitor of insulin-regulated aminopeptidase.
    Lee J, Mustafa T, McDowall SG, Mendelsohn FA, Brennan M, Lew RA, Albiston AL, Chai SY.
    J Pharmacol Exp Ther; 2003 Apr 01; 305(1):205-11. PubMed ID: 12649370
    [Abstract] [Full Text] [Related]

  • 15. Binding to and Inhibition of Insulin-Regulated Aminopeptidase by Macrocyclic Disulfides Enhances Spine Density.
    Diwakarla S, Nylander E, Grönbladh A, Vanga SR, Khan YS, Gutiérrez-de-Terán H, Ng L, Pham V, Sävmarker J, Lundbäck T, Jenmalm-Jensen A, Andersson H, Engen K, Rosenström U, Larhed M, Åqvist J, Chai SY, Hallberg M.
    Mol Pharmacol; 2016 Apr 01; 89(4):413-24. PubMed ID: 26769413
    [Abstract] [Full Text] [Related]

  • 16. 3-Nitro-2H-chromenes as a new class of inhibitors against thioredoxin reductase and proliferation of cancer cells.
    Xiao GQ, Liang BX, Chen SH, Ou TM, Bu XZ, Yan M.
    Arch Pharm (Weinheim); 2012 Oct 01; 345(10):767-70. PubMed ID: 22836584
    [Abstract] [Full Text] [Related]

  • 17. Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Benzopyran-Based Inhibitors.
    Vanga SR, Åqvist J, Hallberg A, Gutiérrez-de-Terán H.
    Front Mol Biosci; 2021 Oct 01; 8():625274. PubMed ID: 33869280
    [Abstract] [Full Text] [Related]

  • 18. Disulfide cyclized tripeptide analogues of angiotensin IV as potent and selective inhibitors of insulin-regulated aminopeptidase (IRAP).
    Andersson H, Demaegdt H, Vauquelin G, Lindeberg G, Karlén A, Hallberg M, Erdélyi M, Hallberg A.
    J Med Chem; 2010 Nov 25; 53(22):8059-71. PubMed ID: 21047126
    [Abstract] [Full Text] [Related]

  • 19. Structure activity relationship studies of tricyclic bispyran sulfone γ-secretase inhibitors.
    Wu WL, Asberom T, Bara T, Bennett C, Burnett DA, Clader J, Domalski M, Greenlee WJ, Josien H, McBriar M, Rajagopalan M, Vicarel M, Xu R, Hyde LA, Del Vecchio RA, Cohen-Williams ME, Song L, Lee J, Terracina G, Zhang Q, Nomeir A, Parker EM, Zhang L.
    Bioorg Med Chem Lett; 2013 Feb 01; 23(3):844-9. PubMed ID: 23265892
    [Abstract] [Full Text] [Related]

  • 20. Development of potent and selective inhibitors of ecto-5'-nucleotidase based on an anthraquinone scaffold.
    Baqi Y, Lee SY, Iqbal J, Ripphausen P, Lehr A, Scheiff AB, Zimmermann H, Bajorath J, Müller CE.
    J Med Chem; 2010 Mar 11; 53(5):2076-86. PubMed ID: 20146483
    [Abstract] [Full Text] [Related]

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