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712 related items for PubMed ID: 24518190

  • 1. 6-Triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrases IX and XII.
    Grandane A, Tanc M, Zalubovskis R, Supuran CT.
    Bioorg Med Chem Lett; 2014 Mar 01; 24(5):1256-60. PubMed ID: 24518190
    [Abstract] [Full Text] [Related]

  • 2. Synthesis of 6-tetrazolyl-substituted sulfocoumarins acting as highly potent and selective inhibitors of the tumor-associated carbonic anhydrase isoforms IX and XII.
    Grandane A, Tanc M, Zalubovskis R, Supuran CT.
    Bioorg Med Chem; 2014 Mar 01; 22(5):1522-8. PubMed ID: 24513186
    [Abstract] [Full Text] [Related]

  • 3. 5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: solution and X-ray crystallographic studies.
    Leitans J, Sprudza A, Tanc M, Vozny I, Zalubovskis R, Tars K, Supuran CT.
    Bioorg Med Chem; 2013 Sep 01; 21(17):5130-8. PubMed ID: 23859774
    [Abstract] [Full Text] [Related]

  • 4. Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII.
    Nocentini A, Carta F, Ceruso M, Bartolucci G, Supuran CT.
    Bioorg Med Chem; 2015 Nov 01; 23(21):6955-66. PubMed ID: 26432607
    [Abstract] [Full Text] [Related]

  • 5. Sulfocoumarin-, Coumarin-, 4-Sulfamoylphenyl-Bearing Indazole-3-carboxamide Hybrids: Synthesis and Selective Inhibition of Tumor-Associated Carbonic Anhydrase Isozymes IX and XII.
    Angapelly S, Sri Ramya PV, Angeli A, Supuran CT, Arifuddin M.
    ChemMedChem; 2017 Oct 09; 12(19):1578-1584. PubMed ID: 28940980
    [Abstract] [Full Text] [Related]

  • 6. Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones.
    Sarikaya B, Ceruso M, Carta F, Supuran CT.
    Bioorg Med Chem; 2014 Nov 01; 22(21):5883-90. PubMed ID: 25267005
    [Abstract] [Full Text] [Related]

  • 7. Synthesis of 6-aryl-substituted sulfocoumarins and investigation of their carbonic anhydrase inhibitory action.
    Grandane A, Tanc M, Žalubovskis R, Supuran CT.
    Bioorg Med Chem; 2015 Apr 01; 23(7):1430-6. PubMed ID: 25753329
    [Abstract] [Full Text] [Related]

  • 8. Coumarins incorporating hydroxy- and chloro-moieties selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the cytosolic ones I and II.
    Maresca A, Supuran CT.
    Bioorg Med Chem Lett; 2010 Aug 01; 20(15):4511-4. PubMed ID: 20580555
    [Abstract] [Full Text] [Related]

  • 9. 7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII.
    Nocentini A, Ceruso M, Carta F, Supuran CT.
    J Enzyme Inhib Med Chem; 2016 Dec 01; 31(6):1226-33. PubMed ID: 26681367
    [Abstract] [Full Text] [Related]

  • 10. Carbonic anhydrase inhibitors. Synthesis, and molecular structure of novel series N-substituted N'-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)guanidines and their inhibition of human cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII.
    Żołnowska B, Sławiński J, Pogorzelska A, Chojnacki J, Vullo D, Supuran CT.
    Eur J Med Chem; 2014 Jan 01; 71():135-47. PubMed ID: 24291567
    [Abstract] [Full Text] [Related]

  • 11. Sulfocoumarins (1,2-benzoxathiine-2,2-dioxides): a class of potent and isoform-selective inhibitors of tumor-associated carbonic anhydrases.
    Tars K, Vullo D, Kazaks A, Leitans J, Lends A, Grandane A, Zalubovskis R, Scozzafava A, Supuran CT.
    J Med Chem; 2013 Jan 10; 56(1):293-300. PubMed ID: 23241068
    [Abstract] [Full Text] [Related]

  • 12. 4-Functionalized 1,3-diarylpyrazoles bearing 6-aminosulfonylbenzothiazole moiety as potent inhibitors of carbonic anhydrase isoforms hCA I, II, IX and XII.
    SitaRam, Ceruso M, Khloya P, Supuran CT, Sharma PK.
    Bioorg Med Chem; 2014 Dec 15; 22(24):6945-52. PubMed ID: 25456084
    [Abstract] [Full Text] [Related]

  • 13. N-β-glycosyl sulfamides are selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII.
    Rodríguez OM, Maresca A, Témpera CA, Bravo RD, Colinas PA, Supuran CT.
    Bioorg Med Chem Lett; 2011 Aug 01; 21(15):4447-50. PubMed ID: 21723123
    [Abstract] [Full Text] [Related]

  • 14. Substituted benzene sulfonamides incorporating 1,3,5-triazinyl moieties potently inhibit human carbonic anhydrases II, IX and XII.
    Saluja AK, Tiwari M, Vullo D, Supuran CT.
    Bioorg Med Chem Lett; 2014 Mar 01; 24(5):1310-4. PubMed ID: 24507918
    [Abstract] [Full Text] [Related]

  • 15. Phenylethynylbenzenesulfonamide regioisomers strongly and selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the cytosolic isoforms I and II.
    Knaus EE, Innocenti A, Scozzafava A, Supuran CT.
    Bioorg Med Chem Lett; 2011 Oct 01; 21(19):5892-6. PubMed ID: 21852133
    [Abstract] [Full Text] [Related]

  • 16. Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isoforms I and II and transmembrane, tumor-associated isoforms IX and XII with boronic acids.
    Winum JY, Innocenti A, Scozzafava A, Montero JL, Supuran CT.
    Bioorg Med Chem; 2009 May 15; 17(10):3649-52. PubMed ID: 19375921
    [Abstract] [Full Text] [Related]

  • 17. Novel coumarins and 2-thioxo-coumarins as inhibitors of the tumor-associated carbonic anhydrases IX and XII.
    Carta F, Maresca A, Scozzafava A, Supuran CT.
    Bioorg Med Chem; 2012 Apr 01; 20(7):2266-73. PubMed ID: 22377674
    [Abstract] [Full Text] [Related]

  • 18. 7,8-disubstituted- but not 6,7-disubstituted coumarins selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the cytosolic ones I and II in the low nanomolar/subnanomolar range.
    Maresca A, Scozzafava A, Supuran CT.
    Bioorg Med Chem Lett; 2010 Dec 15; 20(24):7255-8. PubMed ID: 21067924
    [Abstract] [Full Text] [Related]

  • 19. Carbonic anhydrase inhibitors: synthesis and inhibition of the human cytosolic isozymes I and II and transmembrane isozymes IX, XII (cancer-associated) and XIV with 4-substituted 3-pyridinesulfonamides.
    Brzozowski Z, Sławiński J, Saczewski F, Innocenti A, Supuran CT.
    Eur J Med Chem; 2010 Jun 15; 45(6):2396-404. PubMed ID: 20202722
    [Abstract] [Full Text] [Related]

  • 20. Continued Structural Exploration of Sulfocoumarin as Selective Inhibitor of Tumor-Associated Human Carbonic Anhydrases IX and XII.
    Giovannuzzi S, Capasso C, Nocentini A, Supuran CT.
    Molecules; 2022 Jun 24; 27(13):. PubMed ID: 35807318
    [Abstract] [Full Text] [Related]


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