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244 related items for PubMed ID: 27117428
1. 1-Sulfonyl-6-Piperazinyl-7-Azaindoles as potent and pseudo-selective 5-HT6 receptor antagonists. Fabritius CH, Pesonen U, Messinger J, Horvath R, Salo H, Gałęzowski M, Galek M, Stefańska K, Szeremeta-Spisak J, Olszak-Płachta M, Buda A, Adamczyk J, Król M, Prusis P, Sieprawska-Lupa M, Mikulski M, Kuokkanen K, Chapman H, Obuchowicz R, Korjamo T, Jalava N, Nowak M. Bioorg Med Chem Lett; 2016 Jun 01; 26(11):2610-5. PubMed ID: 27117428 [Abstract] [Full Text] [Related]
13. New 1-arylindoles based serotonin 5-HT7 antagonists. Synthesis and binding evaluation studies. Sagnes C, Fournet G, Satala G, Bojarski AJ, Joseph B. Eur J Med Chem; 2014 Mar 21; 75():159-68. PubMed ID: 24531229 [Abstract] [Full Text] [Related]
14. Synthesis of substituted diphenyl sulfones and their structure-activity relationship with the antagonism of 5-НТ6 receptors. Ivachtchenko A, Golovina E, Kadieva M, Mitkin O, Tkachenko S, Okun I. Bioorg Med Chem; 2013 Aug 01; 21(15):4614-27. PubMed ID: 23787290 [Abstract] [Full Text] [Related]
16. Influence of the 5-HT6 receptor on acetylcholine release in the cortex: pharmacological characterization of 4-(2-bromo-6-pyrrolidin-1-ylpyridine-4-sulfonyl)phenylamine, a potent and selective 5-HT6 receptor antagonist. Riemer C, Borroni E, Levet-Trafit B, Martin JR, Poli S, Porter RH, Bös M. J Med Chem; 2003 Mar 27; 46(7):1273-6. PubMed ID: 12646038 [Abstract] [Full Text] [Related]
17. Discovery and Development of 1-[(2-Bromophenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dimesylate Monohydrate (SUVN-502): A Novel, Potent, Selective and Orally Active Serotonin 6 (5-HT6) Receptor Antagonist for Potential Treatment of Alzheimer's Disease. Nirogi R, Shinde A, Kambhampati RS, Mohammed AR, Saraf SK, Badange RK, Bandyala TR, Bhatta V, Bojja K, Reballi V, Subramanian R, Benade V, Palacharla RC, Bhyrapuneni G, Jayarajan P, Goyal V, Jasti V. J Med Chem; 2017 Mar 09; 60(5):1843-1859. PubMed ID: 28212021 [Abstract] [Full Text] [Related]
18. Optimization of (arylpiperazinylbutyl)oxindoles exhibiting selective 5-HT₇ receptor antagonist activity. Volk B, Gacsályi I, Pallagi K, Poszávácz L, Gyönös I, Szabó E, Bakó T, Spedding M, Simig G, Szénási G. J Med Chem; 2011 Oct 13; 54(19):6657-69. PubMed ID: 21859099 [Abstract] [Full Text] [Related]
19. Effects of 5-HT6 antagonists, Ro-4368554 and SB-258585, in tests used for the detection of cognitive enhancement and antipsychotic-like activity. Gravius A, Laszy J, Pietraszek M, Sághy K, Nagel J, Chambon C, Wegener N, Valastro B, Danysz W, Gyertyán I. Behav Pharmacol; 2011 Apr 13; 22(2):122-35. PubMed ID: 21301322 [Abstract] [Full Text] [Related]